Target Details
| UniProt AC | P13995 |
|---|---|
| Gene Symbol | MTHFD2 |
| Protein Name | Bifunctional methylenetetrahydrofolate dehydrogenase/cyclohydrolase, mitochondrial |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00763 (THF_DHG_CYH) PF02882 (THF_DHG_CYH_C) |
Summary
- Multi-target molecules 36
- Clinical molecules 0
- Avg pChEMBL 7.43
KEGG Pathways (3)
Active Molecules (36)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LAURHQVPQVDMSE
|
8.5 | IC50 | 2 | — | |
RJOHVYDADFTSGL
|
8.5 | IC50 | 2 | — | |
TWNUURIDPRMGCQ
|
8.3 | IC50 | 2 | — | |
OQKAKSSZSQPTDZ
|
8.2 | IC50 | 2 | — | |
SKXNALRRMLGLTB
|
8.1 | IC50 | 2 | — | |
NQGWTLFTUAIYKI
|
8.0 | IC50 | 2 | — | |
WLOOYRBZXKXBLF
|
8.0 | IC50 | 2 | — | |
PMGGZFQJUNWXHA
|
7.9 | IC50 | 2 | — | |
JYNZHPFQYPGQAU
|
7.9 | IC50 | 2 | — | |
SAGKQACQLIZPHJ
|
7.8 | IC50 | 2 | — | |
PCJRTTAQGIPBCR
|
7.8 | IC50 | 2 | — | |
OBBLNVHONCLMSM
|
7.8 | IC50 | 2 | — | |
ILAJKRNAEDQPJD
|
7.7 | IC50 | 2 | — | |
QZBDXJBFDOMBLV
|
7.6 | IC50 | 2 | — | |
WJFBLUPWTGDTOZ
|
7.6 | IC50 | 2 | — | |
JKGSWFFLWSOSSE
|
7.5 | IC50 | 2 | — | |
SNHBFWZJOMVDAT
|
7.5 | IC50 | 2 | — | |
LFVRYVOEGGEFDY
|
7.4 | IC50 | 2 | — | |
JKGSWFFLWSOSSE
|
7.4 | IC50 | 2 | — | |
RWVGZRQLIUEYLA
|
7.4 | IC50 | 2 | — | |
XHAIEKQWEJVFLR
|
7.3 | IC50 | 2 | — | |
ALGPVOJFIGPPPX
|
7.3 | IC50 | 2 | — | |
IEPPNKJTYOVPIQ
|
7.3 | IC50 | 2 | — | |
DMYPIJTXBLLWKR
|
7.2 | IC50 | 2 | — | |
GWYJKHAXXXCOHZ
|
7.2 | IC50 | 2 | — | |
DFAHDLXDZDHCOO
|
7.2 | IC50 | 2 | — | |
ZEVWGOXXSTYHQO
|
7.1 | IC50 | 2 | — | |
KRRMKRRVEYGMPU
|
7.0 | IC50 | 2 | — | |
UCMLONNULHLOIN
|
7.0 | IC50 | 2 | — | |
ZAVKHZGVZLDXOI
|
7.0 | IC50 | 2 | — | |
NSAOCQMFXKCLMJ
|
6.8 | IC50 | 2 | — | |
AKZZELKECDEBFM
|
6.7 | IC50 | 2 | — | |
UTFFVIDGGZNLGQ
|
6.5 | IC50 | 2 | — | |
OSZOXAOEGYVBLJ
|
6.5 | IC50 | 2 | — | |
JSNFRYBHBVDHSG
|
6.2 | IC50 | 2 | — | |
NYRWPFRWINKGPS
|
6.0 | IC50 | 2 | — |