Target Details
| UniProt AC | P13955 |
|---|---|
| Gene Symbol | dfrA |
| Protein Name | Dihydrofolate reductase type 1 from Tn4003 |
| Organism | Staphylococcus aureus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00186 (DHFR_1) |
Summary
- Multi-target molecules 7
- Clinical molecules 0
- Avg pChEMBL 6.44
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NQHZOWBSMCFILX
|
6.7 | IC50 | 4 | — | |
OKJCHFXBCVXSIZ
|
6.6 | IC50 | 6 | — | |
NQHZOWBSMCFILX
|
6.5 | IC50 | 4 | — | |
NQHZOWBSMCFILX
|
6.5 | IC50 | 4 | — | |
GCDLAOPKRFVDHQ
|
6.4 | IC50 | 4 | — | |
OKJCHFXBCVXSIZ
|
6.4 | IC50 | 6 | — | |
VLQRVOAJCWFFQG
|
6.0 | IC50 | 5 | — |