Target Details
| UniProt AC | P13922 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Bifunctional dihydrofolate reductase-thymidylate synthase |
| Organism | Plasmodium falciparum (isolate K1 / Thailand) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00186 (DHFR_1) PF00303 (Thymidylat_synt) |
Summary
- Multi-target molecules 62
- Clinical molecules 0
- Avg pChEMBL 8.14
Active Molecules (62)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QBQZTCRZECEEGK
|
7.2 | Ki | 3 | — | |
XARRNBRDTOCYPU
|
7.1 | IC50 | 3 | — | |
AXIUXECRTOGILY
|
7.0 | Ki | 4 | — | |
YMGUVTBVYOGUFZ
|
7.0 | Ki | 3 | — | |
WHWDLTBBQLJYCJ
|
6.9 | Ki | 2 | — | |
NTVMHTFWSNGDLC
|
6.9 | Ki | 4 | — | |
VMVKLCXTXSSZSI
|
6.8 | Ki | 3 | — | |
UZPCXRZSRCSFOL
|
6.8 | Ki | 2 | — | |
RLKGBZALMDTISP
|
6.8 | Ki | 2 | — | |
VZUPZCGJBVZOJK
|
6.8 | Ki | 2 | — | |
IFLSKJWEERCMHE
|
6.8 | Ki | 3 | — | |
KNUBCZHIBGZRJT
|
6.6 | IC50 | 2 | — |