Target Details
UniProt ACP13922
Gene SymbolN/A
Protein NameBifunctional dihydrofolate reductase-thymidylate synthase
OrganismPlasmodium falciparum (isolate K1 / Thailand)
Entry Name
Organism Category Pathogen
Pfam Domains PF00186 (DHFR_1) PF00303 (Thymidylat_synt)
Summary
  • Multi-target molecules 62
  • Clinical molecules 0
  • Avg pChEMBL 8.14
Top Co-occurrence Targets
Active Molecules (62)
InChIKey pChEMBL Type Targets Clinical
OGSBUKJUDHAQEA 10.9 Ki 5
ORJSMNCGGWKWPM 9.8 Ki 2
LZUNMUXBUPPNFI 9.7 Ki 2
KNRZVDGLNIKBGJ 9.6 Ki 2
BRMZTVKOQXSVAI 9.6 Ki 2
BZWMZSPIVLREMK 9.6 Ki 2
PBILNIRICBBFGH 9.6 Ki 2
YWTRUQFQFAKVEB 9.6 Ki 2
WMTJVURUENODST 9.6 Ki 2
SVZPEOABUWMNSO 9.5 Ki 2
TXHFCRNTZQVBKZ 9.5 Ki 2
ZQYDKYDSKVGDJP 9.4 IC50 2
HYEFEHCIXMVHSP 9.3 Ki 2
UJIGCJXGPGPAHE 9.2 Ki 2
HKCOVOSTNGKHNF 9.2 Ki 2
GUZBZPCNAJDYMO 9.2 IC50 2
MJZJYWCQPMNPRM 9.1 IC50 2
BXUVNXVYAMXINP 9.0 Ki 2
FPULLBVUFHTKQQ 9.0 Ki 3
LLRTYNPSGQWCLZ 9.0 Ki 2
VDGXZSSDCDPCRF 8.9 IC50 2
IVICPTLSOMKNRU 8.8 Ki 2
XBSGVDWRRWPQPP 8.8 Ki 2
KYIIICAIZHTXJE 8.6 Ki 2
POHPGOJAYHKLEL 8.4 Ki 2
ZBPANFPFKDRDTA 8.3 Ki 2
ZEOIMTZUCPVMBV 8.3 Ki 2
XJLXINKUBYWONI 8.1 Ki 3
CXDXEQLVIUNPDR 8.0 Ki 2
QMNFFXRFOJIOKZ 7.9 Ki 3
KTIIBCZDEGUAEF 7.8 Ki 2
SCNQDTMQBLHLJC 7.7 Ki 2
KEBULEDONBRZLH 7.7 Ki 2
VWHBREVXFNULBX 7.6 Ki 2
WUZZGEOZQYQDRK 7.6 Ki 2
JVSPLIKLKSADIK 7.6 Ki 2
MQLILUAGVVAVMX 7.5 Ki 2
KKGMSFFTFBDNOR 7.5 Ki 2
ZDMBJEAMVDIKJQ 7.5 Ki 2
XMMWXKISOBGJLA 7.4 Ki 2
VNPFRENABXECQF 7.3 Ki 2
JOIGYABBXVVXCW 7.3 Ki 2
LDBTVAXGKYIFHO 7.3 Ki 4
BRKLJPVCTPAPFG 7.2 Ki 2
PUMGLGGVAIIWCB 7.2 Ki 4
CIFOWUCVXDSKSU 7.2 Ki 2
KRZXDTYOZAQOGL 7.2 Ki 3
NEIHFQUJLSUWCY 7.2 Ki 2
NEBFMAAUKXSAAC 7.2 Ki 2
VKYOSIISWISQAN 7.2 Ki 2
2D structure