Target Details
| UniProt AC | P13631 |
|---|---|
| Gene Symbol | RARG |
| Protein Name | Retinoic acid receptor gamma |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 121
- Clinical molecules 0
- Avg pChEMBL 7.66
Active Molecules (121)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HCERSGNVDIKWSP
|
6.8 | Ki | 3 | — | |
BNVDMMYUHOFRII
|
6.7 | Kd | 3 | — | |
SIQAHEVWLUDACF
|
6.6 | Kd | 2 | — | |
GRBBADRHKWHVML
|
6.6 | Kd | 3 | — | |
JVJDJWBKWUKBOF
|
6.6 | IC50 | 6 | — | |
KFOYZMZJCMAUGA
|
6.5 | IC50 | 2 | — | |
RREMNJZTZUKGKQ
|
6.5 | IC50 | 3 | — | |
FICUSZQKSIPECZ
|
6.4 | Ki | 2 | — | |
HPPASAIRMDHNEE
|
6.4 | Kd | 2 | — | |
KKVUNMOPDLOPLN
|
6.4 | Kd | 2 | — | |
APXNUGHTPSKBAO
|
6.4 | Ki | 2 | — | |
UPVFFMLTSPBEBW
|
6.4 | Ki | 6 | — | |
WJVKVKNDLOYKSA
|
6.3 | Ki | 2 | — | |
PBTJHWPJNWIKLF
|
6.3 | Kd | 5 | — | |
AJYSMFOKGBZPCF
|
6.2 | IC50 | 4 | — | |
ACTPLOYOROGJBM
|
6.1 | IC50 | 2 | — | |
AYAJZQYENGWICE
|
6.1 | Kd | 2 | — | |
OYWXZUTUIPXTRD
|
6.1 | Ki | 2 | — | |
ITECTFOHDPZGJZ
|
6.1 | Kd | 3 | — | |
SPARUJQOIBYQHO
|
6.0 | Kd | 6 | — | |
TUTOEKVFOVDKCV
|
6.0 | Kd | 3 | — |