Target Details
| UniProt AC | P13612 |
|---|---|
| Gene Symbol | ITGA4 |
| Protein Name | Integrin alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 1,260
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Intestinal immune network for IgA production
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Yersinia infection
Active Molecules (1,260)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RJGXUVWHSRSSMR
|
8.3 | IC50 | 2 | — | |
GERYTDGNULKRJC
|
8.3 | IC50 | 2 | — | |
GLAVTOUIMCZWGE
|
8.3 | IC50 | 2 | — | |
PMVDOKGCDYKXLD
|
8.3 | IC50 | 2 | — | |
CVBUCTGSDPYFLF
|
8.3 | IC50 | 2 | — | |
FHNQKWOESOPUGN
|
8.3 | IC50 | 2 | — | |
JEBRWBXEAHSNTF
|
8.3 | Ki | 2 | — | |
MREBBDFKXMXJBV
|
8.3 | IC50 | 2 | — | |
OHOJPZUGJPTYSY
|
8.3 | Ki | 2 | — | |
NCNWVDNQQKXAAM
|
8.3 | IC50 | 2 | — | |
NIBDXGIMKZXWGB
|
8.3 | IC50 | 2 | — | |
PXIBPFAADDDFDQ
|
8.3 | IC50 | 3 | — | |
UERMUNMPBXMBHT
|
8.3 | IC50 | 3 | — | |
XHZIKHVYHSVYCX
|
8.3 | IC50 | 2 | — | |
HNZUOEFJYXSXOO
|
8.3 | IC50 | 2 | — | |
UPEGZTKVOGNGIP
|
8.3 | IC50 | 2 | — | |
FETXIQQMXPIQAE
|
8.3 | IC50 | 2 | — | |
HWTDZVDHOSKTML
|
8.3 | IC50 | 3 | — | |
IXDDZIVBYAEUTN
|
8.3 | IC50 | 3 | — | |
UIQZHYNNPYXEGY
|
8.3 | IC50 | 2 | — | |
UNDDSOFKUNBHJW
|
8.3 | IC50 | 2 | — | |
WIADTCNCIOEKBT
|
8.3 | IC50 | 2 | — | |
XYRKHQUYEVMHKJ
|
8.3 | IC50 | 3 | — | |
HISUKZFCUMSJFG
|
8.2 | IC50 | 3 | — | |
RBEBHTTXTRLDHD
|
8.2 | IC50 | 2 | — | |
MMUKITGTIBVSEA
|
8.2 | IC50 | 2 | — | |
PINULNVBCYPIJX
|
8.2 | IC50 | 2 | — | |
SCAJVSZKETYPPT
|
8.2 | IC50 | 3 | — | |
XNQLPNVBNWPOSH
|
8.2 | IC50 | 2 | — | |
YXQXXMDLCXXTGF
|
8.2 | IC50 | 2 | — | |
AZIOXOMBBGKKBJ
|
8.2 | IC50 | 3 | — | |
IGRGIQWZKAUHDT
|
8.2 | IC50 | 3 | — | |
SMZRAZWAVQZBEC
|
8.2 | IC50 | 3 | — | |
AWKHKGQMQBSIES
|
8.2 | IC50 | 2 | — | |
BNOQGDSGXBBSTB
|
8.2 | IC50 | 2 | — | |
HLILWKBIJYBQOQ
|
8.2 | IC50 | 2 | — | |
RROLERMMZPCBCQ
|
8.2 | IC50 | 2 | — | |
XCYVGOOLNFZXSG
|
8.2 | IC50 | 2 | — | |
XINCANZSFCTALF
|
8.2 | IC50 | 2 | — | |
ZRZRMFPBYJFMQN
|
8.2 | IC50 | 2 | — | |
SSYLLNMYBQFPCH
|
8.2 | IC50 | 3 | — | |
XVQHEIYCHWOYSM
|
8.2 | IC50 | 2 | — | |
ADRBWUVQHKFVMS
|
8.2 | IC50 | 3 | — | |
BVWQVEZQIWSUFK
|
8.2 | IC50 | 2 | — | |
HHXMIWYEGYZWLB
|
8.2 | IC50 | 2 | — | |
LLUIOBYSYMDPBN
|
8.2 | IC50 | 2 | — | |
PYGLVDAJIZZAIX
|
8.2 | IC50 | 2 | — | |
QYKCSJNOQZFASB
|
8.2 | IC50 | 2 | — | |
SUJIFZABSRZWCR
|
8.2 | Ki | 2 | — | |
YEJVFAXMJIJZFP
|
8.2 | Ki | 2 | — |