Target Details
| UniProt AC | P13612 |
|---|---|
| Gene Symbol | ITGA4 |
| Protein Name | Integrin alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 1,260
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Intestinal immune network for IgA production
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Yersinia infection
Active Molecules (1,260)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UQZSJSAYODPZDI
|
8.4 | IC50 | 2 | — | |
VWGXMPUNQZIEBK
|
8.4 | IC50 | 2 | — | |
WEVSHWPVGKQWOF
|
8.4 | IC50 | 2 | — | |
BWEJBCQAWORYOW
|
8.4 | IC50 | 2 | — | |
NSGJGOWVFDUULW
|
8.4 | Ki | 2 | — | |
QTTOUXZPHJSBFZ
|
8.4 | IC50 | 2 | — | |
ROXYEKDRUFPSTJ
|
8.4 | IC50 | 2 | — | |
SGNBDDWCPLULSJ
|
8.4 | Ki | 2 | — | |
WGSFNDOOBOZLMA
|
8.4 | IC50 | 3 | — | |
ZMHRAQMRFBHOKH
|
8.4 | IC50 | 2 | — | |
ZZQVVTQOTXKPIG
|
8.4 | IC50 | 2 | — | |
NRCSJBQFSDHCEF
|
8.4 | IC50 | 2 | — | |
SKOXRBVQVPASFS
|
8.4 | IC50 | 2 | — | |
UHGBRBWWHMGFEZ
|
8.4 | IC50 | 2 | — | |
VARBGWCQRGTWAS
|
8.4 | IC50 | 2 | — | |
DLLGQRYZARKEBS
|
8.4 | IC50 | 3 | — | |
HGEHCBNZQHVLJS
|
8.4 | IC50 | 3 | — | |
LWCMKXYMIBQWPV
|
8.4 | IC50 | 2 | — | |
CPBOFXSFJQORHL
|
8.4 | IC50 | 2 | — | |
NVVGCQABIHSJSQ
|
8.4 | IC50 | 2 | — | |
OCIRIHRFAHXBIT
|
8.4 | IC50 | 3 | — | |
WTUXQGQYRAGZCP
|
8.4 | IC50 | 3 | — | |
AAQGLFLATBVJPM
|
8.4 | IC50 | 3 | — | |
GCESVLHCMHNRBV
|
8.4 | IC50 | 2 | — | |
GJFNKTYJRCAGCV
|
8.4 | IC50 | 3 | — | |
IAXOAOUFMTWSPG
|
8.4 | IC50 | 3 | — | |
ITXAAOWFOURIHK
|
8.4 | IC50 | 2 | — | |
ITXAAOWFOURIHK
|
8.4 | IC50 | 2 | — | |
POLDUUDTCKSSFP
|
8.4 | IC50 | 3 | — | |
QSVHEGNXLMFWSO
|
8.4 | IC50 | 3 | — | |
SUPGBSSFNJDXNH
|
8.4 | IC50 | 2 | — | |
TXGCBKLXHVSCNM
|
8.4 | IC50 | 2 | — | |
GGRFOSOSNAVBNN
|
8.3 | IC50 | 2 | — | |
IUEVXNMBIIQKAS
|
8.3 | IC50 | 2 | — | |
ZRKHLKCFHURIEZ
|
8.3 | IC50 | 2 | — | |
ZYGZRMMSJAKXOS
|
8.3 | IC50 | 2 | — | |
ZYGZRMMSJAKXOS
|
8.3 | IC50 | 2 | — | |
JOGCJPQFIJVLJJ
|
8.3 | IC50 | 2 | — | |
RBTXBEVPBKTAJE
|
8.3 | IC50 | 2 | — | |
PYDWJUFRRXINNH
|
8.3 | IC50 | 2 | — | |
UFHRTJXQBDQBIP
|
8.3 | IC50 | 2 | — | |
UKDPVOZZLJCIKT
|
8.3 | IC50 | 3 | — | |
WTQCOABHBBAPPQ
|
8.3 | IC50 | 2 | — | |
ZEAGMKZBQHJQAR
|
8.3 | IC50 | 2 | — | |
ADUOFHJYAVYDCK
|
8.3 | IC50 | 2 | — | |
GNBZNYOXBLSXKD
|
8.3 | IC50 | 3 | — | |
MAUMVJHUMXPCFT
|
8.3 | IC50 | 2 | — | |
MIQVLHFYIZFKSQ
|
8.3 | IC50 | 2 | — | |
NNTGHJBTOUDOGY
|
8.3 | IC50 | 2 | — | |
NVVGCQABIHSJSQ
|
8.3 | IC50 | 6 | — |