Target Details
| UniProt AC | P13612 |
|---|---|
| Gene Symbol | ITGA4 |
| Protein Name | Integrin alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 1,260
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Intestinal immune network for IgA production
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Yersinia infection
Active Molecules (1,260)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VFYLHJRNSIZWQQ
|
8.5 | IC50 | 3 | — | |
WEBZMJPCAJJKTN
|
8.5 | IC50 | 2 | — | |
WEXUEGAYHTYTGF
|
8.5 | IC50 | 2 | — | |
WQKGOLGYPXZSSX
|
8.5 | IC50 | 2 | — | |
XWFOQFNTOYPKSS
|
8.5 | IC50 | 2 | — | |
YXFDUNGSOONFHY
|
8.5 | IC50 | 2 | — | |
ZVKDMVSDTFKHRE
|
8.5 | IC50 | 3 | — | |
ZWYAVCQGXAHVLZ
|
8.5 | IC50 | 2 | — | |
CPBOFXSFJQORHL
|
8.5 | IC50 | 2 | — | |
DBRVODXNNJOQHW
|
8.5 | IC50 | 2 | — | |
FXNGYKSGVMSVJB
|
8.5 | IC50 | 2 | — | |
JTHRYJJUORFXHX
|
8.5 | IC50 | 2 | — | |
USYYNLPEWBGIMJ
|
8.5 | IC50 | 2 | — | |
XMUQMOVIUQVKPD
|
8.5 | IC50 | 2 | — | |
BADDGEGOMPMKGI
|
8.5 | IC50 | 2 | — | |
CPADDNAHPXAQNL
|
8.5 | IC50 | 2 | — | |
ONTULEYBHLEJBB
|
8.5 | IC50 | 2 | — | |
QVXKEVCSWQRIDQ
|
8.5 | IC50 | 2 | — | |
UMIUGDHVXREPOA
|
8.5 | IC50 | 2 | — | |
XWZXOSXSUDVTSY
|
8.5 | IC50 | 3 | — | |
BESXQTSZSXTMFO
|
8.5 | IC50 | 2 | — | |
CYRASILRFNUMJX
|
8.5 | IC50 | 3 | — | |
FSPHAJMHUWEJGX
|
8.5 | IC50 | 2 | — | |
FWAKVVZHVYRXIX
|
8.5 | IC50 | 2 | — | |
ONYGTDLGUGFMPT
|
8.5 | IC50 | 2 | — | |
RQFGLPBPADHEDL
|
8.5 | IC50 | 2 | — | |
YGJLELVDLMNGTP
|
8.5 | IC50 | 3 | — | |
LKNNQWMGOZFFKT
|
8.5 | IC50 | 3 | — | |
ZMSHCQNPVJGYNG
|
8.5 | IC50 | 2 | — | |
QQSLHONKFQQQNS
|
8.5 | IC50 | 2 | — | |
CRLQMBSOODURJR
|
8.4 | IC50 | 3 | — | |
DWDDWGYZNYHOGW
|
8.4 | IC50 | 2 | — | |
HAFRWCGZNZNVIH
|
8.4 | IC50 | 3 | — | |
KKZBAYODMNBMQJ
|
8.4 | IC50 | 3 | — | |
LYBFJWLDWYPLFI
|
8.4 | IC50 | 2 | — | |
NVSCTWCNVXBLQP
|
8.4 | IC50 | 3 | — | |
PRAQNLQOJOFZRC
|
8.4 | IC50 | 2 | — | |
VVKWSNOGZODKEQ
|
8.4 | IC50 | 3 | — | |
XMJDMDBLEIGQSK
|
8.4 | IC50 | 3 | — | |
LKUHHZPYAGRQJR
|
8.4 | IC50 | 2 | — | |
BRPCXPCQFDLQMG
|
8.4 | IC50 | 2 | — | |
DGTPDOWNYVTTSD
|
8.4 | IC50 | 2 | — | |
HXCSQLRXMBOJCE
|
8.4 | IC50 | 3 | — | |
KDBWXBVKPMEHLY
|
8.4 | IC50 | 2 | — | |
RBYPTCVDQLQTJV
|
8.4 | IC50 | 3 | — | |
VHVHUZLIYQWAJK
|
8.4 | IC50 | 2 | — | |
AHCTUJXINUDHPY
|
8.4 | IC50 | 2 | — | |
BYRKTALPFLWGRH
|
8.4 | IC50 | 2 | — | |
LUQNTQZWQQXMQY
|
8.4 | IC50 | 3 | — | |
MKIFLEJHQVJUHQ
|
8.4 | IC50 | 2 | — |