Target Details
| UniProt AC | P13612 |
|---|---|
| Gene Symbol | ITGA4 |
| Protein Name | Integrin alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 1,260
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Intestinal immune network for IgA production
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Yersinia infection
Active Molecules (1,260)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LBTMUQGNXSWGSG
|
8.6 | IC50 | 3 | — | |
LTMQOAYQBDWTIQ
|
8.6 | IC50 | 3 | — | |
ULYHJYGNJKWWDI
|
8.6 | IC50 | 2 | — | |
IVFXLUZQXMJCNS
|
8.6 | IC50 | 2 | — | |
QARMMTGRKYICJC
|
8.6 | IC50 | 2 | — | |
AESXNYDCOYLGAH
|
8.6 | IC50 | 2 | — | |
AQGOTKCWRZAUIP
|
8.6 | IC50 | 3 | — | |
CANDGDJMWTWWGD
|
8.6 | IC50 | 2 | — | |
KFNKHVGWGQDFPY
|
8.6 | IC50 | 3 | — | |
LETDUXBWZBQZEK
|
8.6 | IC50 | 2 | — | |
NFMHJWOVOIOOTE
|
8.6 | IC50 | 3 | — | |
QLSFJHYLUVSHEA
|
8.6 | IC50 | 2 | — | |
YEIXEKIUHATHCQ
|
8.6 | IC50 | 2 | — | |
ZIPHKIDWZBDOSS
|
8.6 | IC50 | 3 | — | |
KCLSGFBGNSDHCC
|
8.6 | IC50 | 2 | — | |
UMWNDCFZURLHDU
|
8.6 | IC50 | 2 | — | |
ZUYLZBWPGTXZOO
|
8.6 | IC50 | 3 | — | |
BQGQVBGSESRXLR
|
8.6 | Ki | 2 | — | |
DGVLWIGCRQYUHB
|
8.6 | IC50 | 2 | — | |
PLGLSICIZNTCPX
|
8.6 | IC50 | 2 | — | |
VMDLUIBMPQVKHH
|
8.6 | IC50 | 2 | — | |
XGSTWXJCKPYTLE
|
8.6 | IC50 | 2 | — | |
MCAIXYIMLUUTHW
|
8.6 | IC50 | 3 | — | |
MMIPQFQYOLUDRE
|
8.6 | IC50 | 3 | — | |
MUMCFXBPBDMRQQ
|
8.6 | IC50 | 2 | — | |
VXONPVFJSPELTA
|
8.6 | IC50 | 2 | — | |
ZNCWUXZNXWDVRM
|
8.6 | IC50 | 2 | — | |
BYRKTALPFLWGRH
|
8.6 | IC50 | 2 | — | |
JOZJWMSTRAKGKY
|
8.6 | IC50 | 2 | — | |
KFKKFCVUQZXZEI
|
8.6 | IC50 | 2 | — | |
BKYBRLBEBOMPJQ
|
8.6 | IC50 | 3 | — | |
CTRIJHIVZHRDHX
|
8.6 | IC50 | 2 | — | |
ILIJAAWQIUXHNY
|
8.6 | IC50 | 2 | — | |
INVXYDDFZYTUMS
|
8.6 | IC50 | 2 | — | |
YKDBMBISKSKBIS
|
8.6 | IC50 | 2 | — | |
ZLNBTVYNXDCEPU
|
8.6 | IC50 | 2 | — | |
AAJPBIDYTZACLA
|
8.5 | IC50 | 2 | — | |
FZMHKLISSNPJKF
|
8.5 | IC50 | 2 | — | |
KHZVLOYNGSJKBU
|
8.5 | IC50 | 2 | — | |
LYIQTSRHBZHIPH
|
8.5 | IC50 | 2 | — | |
YDWJHQASZKEBFD
|
8.5 | IC50 | 2 | — | |
GGUXLECBDJKACP
|
8.5 | IC50 | 2 | — | |
XAVTVDBSJQZNHA
|
8.5 | IC50 | 2 | — | |
BNMACLPLFKEEMT
|
8.5 | IC50 | 2 | — | |
FOABJUOBCGOTCS
|
8.5 | IC50 | 2 | — | |
ILKTTWKSRXZSRE
|
8.5 | IC50 | 2 | — | |
MKCISCXMJCFWLW
|
8.5 | IC50 | 2 | — | |
MONYNIRDTFXWKB
|
8.5 | IC50 | 2 | — | |
NOEWSRIYUKZVEG
|
8.5 | IC50 | 3 | — | |
QMHTXRUDZGHUND
|
8.5 | IC50 | 2 | — |