Target Details
| UniProt AC | P13612 |
|---|---|
| Gene Symbol | ITGA4 |
| Protein Name | Integrin alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 1,260
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Intestinal immune network for IgA production
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Yersinia infection
Active Molecules (1,260)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YZZMJHSHQYXEFZ
|
8.8 | IC50 | 2 | — | |
ZPYVSGYLDUOOIZ
|
8.8 | IC50 | 2 | — | |
LAVKEKZSIBZMRJ
|
8.8 | IC50 | 3 | — | |
LYEWIWRMQRJNFS
|
8.8 | IC50 | 2 | — | |
UDEOSPCGCDINCC
|
8.8 | IC50 | 2 | — | |
HJWCBRDYEUTPNN
|
8.8 | IC50 | 2 | — | |
RYQVJWYRMJZFAD
|
8.8 | IC50 | 2 | — | |
WUAFZBANWSFBSP
|
8.8 | IC50 | 2 | — | |
CWIZGCPRLPKGAW
|
8.7 | IC50 | 2 | — | |
KCHWAIVFBMDFOL
|
8.7 | IC50 | 2 | — | |
OEJOIHNKFVHVEB
|
8.7 | IC50 | 3 | — | |
UTLDJUNUIMQLSJ
|
8.7 | IC50 | 3 | — | |
VNCVFIISPZFYCK
|
8.7 | IC50 | 2 | — | |
WOZSUXNJFSSYJW
|
8.7 | IC50 | 3 | — | |
ZSLLAAOZAJPOMZ
|
8.7 | IC50 | 2 | — | |
DHLWZPYEINGBFR
|
8.7 | IC50 | 3 | — | |
FSIOKPLPDOYRFJ
|
8.7 | IC50 | 2 | — | |
LBTMUQGNXSWGSG
|
8.7 | IC50 | 3 | — | |
BRXOSTDCWWZMCS
|
8.7 | IC50 | 2 | — | |
QYLJBVNSXNPXCO
|
8.7 | IC50 | 3 | — | |
BYORRPJZRWMSCK
|
8.7 | IC50 | 2 | — | |
IHZDVSSJVCEYBR
|
8.7 | Ki | 2 | — | |
JEBRWBXEAHSNTF
|
8.7 | Ki | 2 | — | |
JGCUUCXMZKFRKP
|
8.7 | IC50 | 3 | — | |
JHBJKRQQEIQKHE
|
8.7 | IC50 | 2 | — | |
JMRHAIGRROKJRA
|
8.7 | IC50 | 2 | — | |
MWICRKHXHXGESF
|
8.7 | IC50 | 3 | — | |
QTTOUXZPHJSBFZ
|
8.7 | IC50 | 2 | — | |
SJHWRZBMMCDJDX
|
8.7 | IC50 | 2 | — | |
UOCOERCBTSGDPC
|
8.7 | IC50 | 2 | — | |
UOQRUCISSASGLE
|
8.7 | IC50 | 2 | — | |
VBHVOJJDISNENC
|
8.7 | IC50 | 3 | — | |
VVZGYMGXVWZKDS
|
8.7 | IC50 | 2 | — | |
YWUYPMUCGBFZKX
|
8.7 | IC50 | 2 | — | |
YECQPPDRORMNRX
|
8.7 | IC50 | 3 | — | |
CXSIVJHZBHTFAQ
|
8.7 | IC50 | 3 | — | |
MXTOSAOISBOVCI
|
8.7 | IC50 | 3 | — | |
MZVLJIIBEREKBQ
|
8.7 | IC50 | 2 | — | |
UMSYINVARMBJFW
|
8.7 | IC50 | 2 | — | |
UNPABXBAJICLTA
|
8.7 | IC50 | 2 | — | |
WRHKZVFBIZOZCV
|
8.7 | IC50 | 2 | — | |
CBLWZZPATNWACH
|
8.7 | IC50 | 2 | — | |
GRSVHAPJHOVVNB
|
8.7 | IC50 | 2 | — | |
HZKMGPCRORUHHA
|
8.7 | IC50 | 2 | — | |
VPJJESVGYJPWNF
|
8.7 | IC50 | 2 | — | |
WDRNJLLLEXRYOE
|
8.7 | IC50 | 2 | — | |
YPBWVSWHQCEYGY
|
8.7 | IC50 | 2 | — | |
DZZGWIOPCRAELG
|
8.7 | IC50 | 2 | — | |
RYYQCANRHNEFSA
|
8.7 | Ki | 2 | — | |
HJBLGUARYIQSOP
|
8.6 | IC50 | 2 | — |