Target Details
| UniProt AC | P13612 |
|---|---|
| Gene Symbol | ITGA4 |
| Protein Name | Integrin alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 1,260
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Intestinal immune network for IgA production
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Yersinia infection
Active Molecules (1,260)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XINCANZSFCTALF
|
9.1 | IC50 | 2 | — | |
BLLLAUHTNAVSQR
|
9.1 | Kd | 5 | — | |
CCBJMQPSBBHXRQ
|
9.1 | IC50 | 2 | — | |
POFWSMHHXSOAAJ
|
9.1 | Ki | 2 | — | |
VOCBDNRGLAJDJJ
|
9.1 | Ki | 2 | — | |
WSJBDILTQGLEQA
|
9.1 | IC50 | 2 | — | |
CRLOUCQPUXMUCD
|
9.1 | IC50 | 2 | — | |
GYRBFYNAOXAEPO
|
9.1 | IC50 | 2 | — | |
RTQDJONLCOQVMI
|
9.1 | IC50 | 2 | — | |
UUXTZGJGBUBTBQ
|
9.1 | IC50 | 2 | — | |
WHAMHFBSIWLDIJ
|
9.1 | IC50 | 2 | — | |
OVAMYRDVZGRBCF
|
9.1 | IC50 | 2 | — | |
SIXJMSJQDGDEAK
|
9.1 | IC50 | 2 | — | |
JPDURLRTQZCKKD
|
9.1 | IC50 | 2 | — | |
PUJRKGKDIKCRSV
|
9.1 | Ki | 2 | — | |
XHCXORPSNPUSKF
|
9.1 | IC50 | 2 | — | |
XRXLVYQWWZTNMN
|
9.1 | IC50 | 2 | — | |
ZSKXPSIETQZQJF
|
9.1 | Ki | 2 | — | |
DVLBSXLUGBCBRC
|
9.0 | IC50 | 3 | — | |
NXAVFGCSONIIII
|
9.0 | IC50 | 2 | — | |
PALKXFSSVDMBNG
|
9.0 | IC50 | 3 | — | |
PUGXPRVUVZGAHB
|
9.0 | IC50 | 2 | — | |
FQKAGOPIYIPBGP
|
9.0 | IC50 | 2 | — | |
IRVJBUBWERQASS
|
9.0 | IC50 | 3 | — | |
UZEJXLHLCJUOKN
|
9.0 | IC50 | 3 | — | |
ZLSOUAKIYFWGAA
|
9.0 | IC50 | 2 | — | |
XAENZKDUGMVTAX
|
9.0 | IC50 | 2 | — | |
BQGQVBGSESRXLR
|
9.0 | Ki | 2 | — | |
FZHRZAHVVNSORE
|
9.0 | IC50 | 2 | — | |
NVHYHKRZUDLBBQ
|
9.0 | IC50 | 3 | — | |
POFWSMHHXSOAAJ
|
9.0 | Ki | 2 | — | |
PQNWKBRBHJLNTG
|
9.0 | IC50 | 2 | — | |
PWMAEWNRSJGUGQ
|
9.0 | IC50 | 2 | — | |
RJALSTOENHOZQV
|
9.0 | IC50 | 3 | — | |
USEDUTJSKDZBGX
|
9.0 | IC50 | 2 | — | |
VOKWLPMZPWNTFX
|
9.0 | IC50 | 2 | — | |
YVTBYYRAVCBZCJ
|
9.0 | IC50 | 2 | — | |
OFKDMFLFKUWHRQ
|
9.0 | IC50 | 2 | — | |
PRUPKWNQAVQPOI
|
9.0 | IC50 | 3 | — | |
GRKQLMXUWWDASB
|
9.0 | IC50 | 2 | — | |
NJWAMCOTWKQQQO
|
9.0 | IC50 | 2 | — | |
OPKAUQAIFQSBOZ
|
9.0 | IC50 | 2 | — | |
WKEYMRCHVPVMOY
|
9.0 | IC50 | 3 | — | |
WVLIGOCMVXCNLK
|
9.0 | IC50 | 2 | — | |
XXMAAHCJSQLUJD
|
9.0 | IC50 | 2 | — | |
PPLDXTMJKAYRSX
|
8.9 | IC50 | 2 | — | |
UTRBTIFHRKMFMU
|
8.9 | IC50 | 3 | — | |
DQNZNDKDCJZRKQ
|
8.9 | IC50 | 2 | — | |
JQZNUGKWTQHGEY
|
8.9 | IC50 | 2 | — | |
OUOYSXSWASMDOM
|
8.9 | IC50 | 2 | — |