Target Details
| UniProt AC | P13612 |
|---|---|
| Gene Symbol | ITGA4 |
| Protein Name | Integrin alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 1,260
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Intestinal immune network for IgA production
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Yersinia infection
Active Molecules (1,260)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UWDSAWYVWRSKPP
|
9.4 | IC50 | 3 | — | |
FILAPYMFTPTZNJ
|
9.4 | IC50 | 2 | — | |
WRHKZVFBIZOZCV
|
9.4 | IC50 | 2 | — | |
XVFGXBXVSHPQNQ
|
9.4 | IC50 | 3 | — | |
GRIXHDLHYDUGHP
|
9.4 | IC50 | 2 | — | |
JSMSAVCWGLIOCE
|
9.4 | IC50 | 2 | — | |
MMKDEARGHIPLGR
|
9.4 | IC50 | 2 | — | |
QPZMNXQBHCXEKU
|
9.4 | IC50 | 2 | — | |
AHUFAXIJOQGUOY
|
9.4 | IC50 | 2 | — | |
HLDVFPCKENBYRZ
|
9.4 | IC50 | 2 | — | |
RUTGLWCLWPBBMZ
|
9.4 | IC50 | 2 | — | |
TZHPMUDTJGJDTC
|
9.4 | IC50 | 2 | — | |
ZFEZMZIUQXOHHJ
|
9.4 | IC50 | 2 | — | |
KLRZAJNROFRNBT
|
9.3 | IC50 | 2 | — | |
FJTPRDFOASDXPB
|
9.3 | IC50 | 3 | — | |
NAKHAAQWKXWRKS
|
9.3 | IC50 | 2 | — | |
GYUQWZWCORBSLX
|
9.3 | IC50 | 2 | — | |
HLUUKMWLLADVRH
|
9.3 | IC50 | 2 | — | |
CQLHRAHQMMCYBN
|
9.3 | IC50 | 2 | — | |
MOQBCMVOFUTVHS
|
9.3 | Ki | 2 | — | |
XDGSCLZNDKEXAE
|
9.3 | IC50 | 3 | — | |
YHFWYPZHVJZULG
|
9.3 | IC50 | 2 | — | |
WIBDJDYXWICGSX
|
9.3 | IC50 | 2 | — | |
JZNIXBUMPQZIJY
|
9.3 | IC50 | 2 | — | |
YXPCBCHWUVICEH
|
9.3 | IC50 | 2 | — | |
KAGRGOJSNNEPTP
|
9.3 | IC50 | 2 | — | |
QPBVMPSYTAHRNI
|
9.3 | IC50 | 2 | — | |
BXXARJACSOMMKX
|
9.3 | IC50 | 2 | — | |
WFNCDDGCGNUXLG
|
9.3 | IC50 | 2 | — | |
RXOAYEHOAAHUMM
|
9.2 | IC50 | 2 | — | |
WNKRETACHGJVKC
|
9.2 | IC50 | 3 | — | |
NWQAJABKOGMVNQ
|
9.2 | IC50 | 2 | — | |
DDXWRMMINAREGF
|
9.2 | IC50 | 3 | — | |
BRZKFEHVZLVFIJ
|
9.2 | IC50 | 2 | — | |
MGKZYWCSUHALDJ
|
9.2 | IC50 | 3 | — | |
PWDOMNUZQXPHIM
|
9.2 | IC50 | 2 | — | |
IYTTUCDELWMTPJ
|
9.2 | IC50 | 2 | — | |
LPPNDFOQUKQERO
|
9.2 | IC50 | 3 | — | |
SITGJFUZUFHSHU
|
9.2 | IC50 | 3 | — | |
LDWAIULYHJTVQT
|
9.2 | IC50 | 3 | — | |
XQYVKXLNFSIYBI
|
9.2 | IC50 | 2 | — | |
AKXPOHLUWJPKQY
|
9.2 | IC50 | 2 | — | |
OSOUXNDWVSWDJT
|
9.2 | IC50 | 2 | — | |
OPJBDVVJACDHPY
|
9.1 | IC50 | 3 | — | |
SALKSINYSDSNQB
|
9.1 | IC50 | 2 | — | |
XTGPAZFJJAYMMR
|
9.1 | IC50 | 2 | — | |
ASYDYYRPDBLCFU
|
9.1 | IC50 | 3 | — | |
ASYDYYRPDBLCFU
|
9.1 | IC50 | 3 | — | |
DXZXXIJEZVYUJW
|
9.1 | IC50 | 3 | — | |
QPBGCQHXTQTQCH
|
9.1 | IC50 | 2 | — |