Target Details
| UniProt AC | P13612 |
|---|---|
| Gene Symbol | ITGA4 |
| Protein Name | Integrin alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01839 (FG-GAP) PF08441 (Integrin_A_Ig_1) PF20805 (Integrin_A_Ig_2) PF20806 (Integrin_A_Ig_3) |
Summary
- Multi-target molecules 1,260
- Clinical molecules 0
- Avg pChEMBL 7.82
KEGG Pathways (17)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Hematopoietic cell lineage
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- IgSF CAM signaling
- Integrin signaling
- Intestinal immune network for IgA production
- Leishmaniasis
- Leukocyte transendothelial migration
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Yersinia infection
Active Molecules (1,260)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZGVUZPIYOSOTEU
|
8.2 | Ki | 2 | — | |
NCNWVDNQQKXAAM
|
8.2 | IC50 | 2 | — | |
DRSJLVGDSNWQBI
|
8.2 | IC50 | 4 | — | |
FKEVPOLPQDCFDG
|
8.2 | IC50 | 2 | — | |
LPPNDFOQUKQERO
|
8.2 | IC50 | 3 | — | |
NSAOFDPAHXXLPO
|
8.2 | IC50 | 3 | — | |
WLAAYHAUMYPKQO
|
8.2 | IC50 | 2 | — | |
HUPHLMZTLJGDRG
|
8.2 | IC50 | 3 | — | |
QNNJFNWDUBNNHS
|
8.2 | IC50 | 2 | — | |
YSEPKFBFYZRCEF
|
8.2 | IC50 | 2 | — | |
CVUCMYLZXBNVCH
|
8.2 | IC50 | 2 | — | |
VGPJOSHXOYLLDR
|
8.2 | IC50 | 2 | — | |
VVWWYYCPGHVEKY
|
8.2 | IC50 | 3 | — | |
AUDWOIGHJBJWAG
|
8.2 | IC50 | 2 | — | |
BTYSVIBSJVRJTA
|
8.2 | Ki | 2 | — | |
CPWXAEABNBAWBW
|
8.2 | IC50 | 2 | — | |
FQJKZZROWKIEKJ
|
8.2 | IC50 | 2 | — | |
FXNUCHXDIULYQS
|
8.2 | IC50 | 2 | — | |
IFGOZIQVZFBABB
|
8.2 | IC50 | 2 | — | |
PMVWESVPNZPORP
|
8.2 | IC50 | 2 | — | |
PUJRKGKDIKCRSV
|
8.2 | Ki | 2 | — | |
QWYIHLODVGFLLG
|
8.2 | IC50 | 2 | — | |
SATRONDTGPPWOY
|
8.2 | IC50 | 3 | — | |
UZDJXPGRSXEUQF
|
8.2 | IC50 | 2 | — | |
YDWZFLXHAFVVPG
|
8.2 | Ki | 2 | — | |
ZSKXPSIETQZQJF
|
8.2 | Ki | 2 | — | |
FMEWWQCJNULALH
|
8.1 | IC50 | 2 | — | |
LWMXBHHAGNVCLL
|
8.1 | IC50 | 3 | — | |
UIJGLNLFNCUJOR
|
8.1 | IC50 | 2 | — | |
AEMBNJITTWJYBV
|
8.1 | IC50 | 3 | — | |
BMWLPSHBOYUODM
|
8.1 | IC50 | 2 | — | |
CNEQPYAXDOPBOW
|
8.1 | IC50 | 2 | — | |
WPFUDMYSAIKMKF
|
8.1 | IC50 | 2 | — | |
XFEBZCPSSQZCEA
|
8.1 | IC50 | 3 | — | |
YOCCTHZQHRBDCH
|
8.1 | IC50 | 3 | — | |
RIEZNKPULWYALL
|
8.1 | IC50 | 2 | — | |
FJQOIVAGPXCDDW
|
8.1 | Ki | 2 | — | |
JSQYTWAPRPJKPW
|
8.1 | IC50 | 2 | — | |
LYNBJSJVJXRVTC
|
8.1 | IC50 | 2 | — | |
UAWIVFLVAQKETC
|
8.1 | IC50 | 3 | — | |
VSPGOHCWYWVAIX
|
8.1 | IC50 | 2 | — | |
ZNPQPNSOQCGUTL
|
8.1 | IC50 | 2 | — | |
BNQXJYCZJDLJRE
|
8.1 | IC50 | 2 | — | |
CJASQSIGTKSMFJ
|
8.1 | IC50 | 3 | — | |
DGRUTRGOEXGZIA
|
8.1 | IC50 | 2 | — | |
KGDZUGSBEBVXKQ
|
8.1 | IC50 | 3 | — | |
NCNWVDNQQKXAAM
|
8.1 | IC50 | 2 | — | |
UGZHFBYZXYHYQD
|
8.1 | IC50 | 2 | — | |
QFKSUZWCKIXRSF
|
8.1 | IC50 | 2 | — | |
GMXFUNCMCRRVSE
|
8.1 | IC50 | 2 | — |