Target Details
| UniProt AC | P12931 |
|---|---|
| Gene Symbol | SRC |
| Protein Name | Proto-oncogene tyrosine-protein kinase Src |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,978
- Clinical molecules 816
- Avg pChEMBL 7.32
KEGG Pathways (45)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Bladder cancer
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- ErbB signaling pathway
- Estrogen signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- GnRH signaling pathway
- Hepatitis B
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Mitophagy - animal
- Neutrophil extracellular trap formation
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Platelet activation
- Prolactin signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Shigellosis
- Thyroid hormone signaling pathway
- Tight junction
- Tuberculosis
- VEGF signaling pathway
- Viral carcinogenesis
- Yersinia infection
Associated Diseases (2)
Active Molecules (1,978)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YMXZIONZPMRKQD
|
8.2 | IC50 | 5 | — | |
URNMUIDFWOJTPW
|
8.1 | Ki | 7 | Yes | |
WJOMVKXZFSMUMB
|
8.1 | IC50 | 3 | — | |
LYJIVFCOOJRVBF
|
8.1 | IC50 | 4 | — | |
XQBYDVRVYRYLCH
|
8.1 | IC50 | 3 | Yes | |
FCIILWHQWNLPJU
|
8.1 | IC50 | 4 | Yes | |
AJNZDFUREDKURT
|
8.1 | IC50 | 3 | — | |
AOEVEOHCGZVHSB
|
8.1 | IC50 | 3 | — | |
AUQUDEKRNSXTHR
|
8.1 | IC50 | 2 | — | |
CSZJFFGJPPIFRZ
|
8.1 | IC50 | 2 | — | |
FPSYUXXLCHMFRU
|
8.1 | IC50 | 4 | — | |
GPPNXVDUQMDEAO
|
8.1 | IC50 | 3 | — | |
HMMIVTXSLFBBHC
|
8.1 | IC50 | 4 | — | |
IMHCVVDKOFKZKX
|
8.1 | IC50 | 3 | — | |
ITLNVPRPOQCABR
|
8.1 | IC50 | 2 | — | |
JQVRXEMLYFQYRR
|
8.1 | IC50 | 3 | — | |
JSDGKSMNPHJDFK
|
8.1 | Ki | 35 | — | |
LSEQHHCLNCHKNO
|
8.1 | IC50 | 3 | — | |
MFPLYINPSNJRRI
|
8.1 | IC50 | 3 | — | |
MIAZWLXBNITBFW
|
8.1 | IC50 | 4 | — | |
MRCFTWAYZAHAFA
|
8.1 | IC50 | 12 | Yes | |
ULMCFLZUGRSEQA
|
8.1 | Ki | 17 | — | |
URPHWXWGWHZRLT
|
8.1 | IC50 | 3 | — | |
USUSRWRXNKNUGL
|
8.1 | IC50 | 3 | — | |
VGHUYLNQBPEVLC
|
8.1 | IC50 | 2 | — | |
WDZOSPABBUJVMV
|
8.1 | IC50 | 3 | — | |
WQDGYGJFEUAXKW
|
8.1 | IC50 | 3 | — | |
XLYVQVWMTOLDNL
|
8.1 | IC50 | 21 | — | |
XLYVQVWMTOLDNL
|
8.1 | IC50 | 21 | — | |
XTASITJXTTXPJS
|
8.1 | IC50 | 3 | — | |
YGZNOUTVUALXEX
|
8.1 | IC50 | 3 | — | |
ZWVZORIKUNOTCS
|
8.1 | Ki | 69 | — | |
MXBRHEFPFHSZLC
|
8.1 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
8.1 | Kd | 220 | — | |
RFSFIDGEFVXSQM
|
8.1 | IC50 | 12 | Yes | |
ZJVPEIBBMXWONH
|
8.1 | IC50 | 3 | — | |
HYEHPKUGAXUAGD
|
8.1 | IC50 | 3 | — | |
KBHJOYQXMRWUFC
|
8.1 | IC50 | 3 | — | |
VKNSWNWSJODLGL
|
8.1 | IC50 | 2 | — | |
DMZBGGYSGOPZET
|
8.1 | IC50 | 4 | — | |
GHRBLHUQTOTLMU
|
8.1 | IC50 | 2 | — | |
GYAOYHATHSUFRX
|
8.1 | IC50 | 3 | — | |
HSODWQGVXRNOEV
|
8.1 | IC50 | 3 | — | |
HYEOMJSVLMONGY
|
8.1 | IC50 | 4 | — | |
IFPPYSWJNWHOLQ
|
8.1 | IC50 | 52 | Yes | |
IHERTXREJRKYHR
|
8.1 | IC50 | 2 | — | |
MKEMSFNHLLMWNR
|
8.1 | IC50 | 2 | — | |
MXWHSGSOZDOVLL
|
8.1 | IC50 | 4 | Yes | |
PEDMIJDFAWDUDE
|
8.1 | IC50 | 3 | — | |
QBHJVCQCWMYGAJ
|
8.1 | IC50 | 3 | — |