Target Details
| UniProt AC | P12931 |
|---|---|
| Gene Symbol | SRC |
| Protein Name | Proto-oncogene tyrosine-protein kinase Src |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,978
- Clinical molecules 816
- Avg pChEMBL 7.32
KEGG Pathways (45)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Bladder cancer
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- ErbB signaling pathway
- Estrogen signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- GnRH signaling pathway
- Hepatitis B
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Mitophagy - animal
- Neutrophil extracellular trap formation
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Platelet activation
- Prolactin signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Shigellosis
- Thyroid hormone signaling pathway
- Tight junction
- Tuberculosis
- VEGF signaling pathway
- Viral carcinogenesis
- Yersinia infection
Associated Diseases (2)
Active Molecules (1,978)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ICDKRHFFALYPNE
|
8.2 | IC50 | 2 | — | |
IEUYALOEFWZLQN
|
8.2 | IC50 | 4 | — | |
JXOIAMLUKJBNFR
|
8.2 | IC50 | 4 | Yes | |
OOJMGPZKNVMKBS
|
8.2 | IC50 | 3 | — | |
OTQOZFYTAOFNOL
|
8.2 | IC50 | 3 | — | |
PDQILYUWWBSUJV
|
8.2 | IC50 | 4 | — | |
PELUCDAGCYAICS
|
8.2 | IC50 | 3 | Yes | |
ROHJEIACUNTGFP
|
8.2 | IC50 | 16 | — | |
SSIFHFIRVJXKOP
|
8.2 | IC50 | 4 | — | |
SXEJPJAKKSSHHC
|
8.2 | IC50 | 4 | — | |
VTQGLZJCCQHUJG
|
8.2 | IC50 | 4 | — | |
XZCLCFIAUCVNJF
|
8.2 | IC50 | 4 | — | |
YHHHJKZCRBUOTD
|
8.2 | IC50 | 2 | — | |
ZIQFYVPVJZEOFS
|
8.2 | IC50 | 9 | Yes | |
DSOWZXLTTGDSAK
|
8.2 | IC50 | 2 | Yes | |
FWVUUGWQEZWWHV
|
8.2 | IC50 | 6 | Yes | |
FRKWMLCUONAHJH
|
8.2 | IC50 | 13 | Yes | |
DEUUCYCGMWGKGM
|
8.2 | IC50 | 2 | — | |
HUMIGOFJWQKXPY
|
8.2 | IC50 | 3 | — | |
LXRITECWUGVGTD
|
8.2 | IC50 | 6 | — | |
UMBIRSZUCJNBHB
|
8.2 | IC50 | 18 | — | |
ZVVNPLLNFALAOH
|
8.2 | IC50 | 2 | — | |
KIHQVERTLRHJED
|
8.2 | IC50 | 3 | Yes | |
PDEWZRGITAXNMH
|
8.2 | IC50 | 2 | — | |
PUJPRSYMMNNGBM
|
8.2 | IC50 | 2 | — | |
PWKWAGIBTGYEHC
|
8.2 | IC50 | 2 | — | |
BCAHGWFHBBMPHP
|
8.2 | IC50 | 2 | — | |
IWODHENDABKBRB
|
8.2 | IC50 | 6 | — | |
NYBNNHFUSGTOBH
|
8.2 | IC50 | 2 | — | |
CJMMCIXRPVLDBH
|
8.2 | IC50 | 12 | Yes | |
AMKRSTDSNXNZMY
|
8.2 | IC50 | 4 | — | |
BBDYTNGLQLQTOV
|
8.2 | IC50 | 4 | — | |
COAQRADEUYYCDG
|
8.2 | IC50 | 12 | Yes | |
CQKMMXFWQMPMFC
|
8.2 | IC50 | 3 | — | |
CWIGGHRHBFIADD
|
8.2 | IC50 | 3 | — | |
DGDQMZKPMBIFOF
|
8.2 | IC50 | 4 | — | |
DPLQMNPQGDUUNM
|
8.2 | IC50 | 3 | Yes | |
FEFIXEMJIYHFAZ
|
8.2 | IC50 | 4 | — | |
GRFBNEAPKLWFPA
|
8.2 | IC50 | 4 | — | |
GWOFQUMBWYKHFL
|
8.2 | IC50 | 5 | — | |
HJRJXYSRPDUZLG
|
8.2 | IC50 | 2 | — | |
LJMCZWSDLQFAMA
|
8.2 | IC50 | 2 | — | |
MMEJLCRBNBQORJ
|
8.2 | IC50 | 3 | — | |
PCZISKGDXHGYTI
|
8.2 | IC50 | 3 | — | |
QGRUEQPBBBTRPN
|
8.2 | IC50 | 4 | — | |
QZGNMSFUFGRNIV
|
8.2 | Ki | 2 | — | |
STYBOAPFAFDXGS
|
8.2 | IC50 | 3 | — | |
TXAYKQMEBQBGLR
|
8.2 | IC50 | 4 | Yes | |
XVVANFOECICSLK
|
8.2 | IC50 | 4 | — | |
YJSFAHMGDRBZGH
|
8.2 | IC50 | 16 | Yes |