Target Details
| UniProt AC | P12931 |
|---|---|
| Gene Symbol | SRC |
| Protein Name | Proto-oncogene tyrosine-protein kinase Src |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,978
- Clinical molecules 816
- Avg pChEMBL 7.32
KEGG Pathways (45)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Bladder cancer
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- ErbB signaling pathway
- Estrogen signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- GnRH signaling pathway
- Hepatitis B
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Mitophagy - animal
- Neutrophil extracellular trap formation
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Platelet activation
- Prolactin signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Shigellosis
- Thyroid hormone signaling pathway
- Tight junction
- Tuberculosis
- VEGF signaling pathway
- Viral carcinogenesis
- Yersinia infection
Associated Diseases (2)
Active Molecules (1,978)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BGKZQFXBRTXGLE
|
8.5 | IC50 | 2 | — | |
JVMXFXGOSURYQL
|
8.5 | IC50 | 3 | — | |
QONHZAOUSLDLOE
|
8.5 | Ki | 3 | — | |
KNGAOBKKLCKYNZ
|
8.5 | IC50 | 5 | — | |
QHESHAOBGKRAPW
|
8.5 | IC50 | 2 | Yes | |
CPKWNMKGJMCCPZ
|
8.5 | IC50 | 2 | — | |
GFPDOXWFWOKWOV
|
8.5 | IC50 | 2 | — | |
KNTPBVJWLVSQOV
|
8.5 | IC50 | 2 | — | |
PLZOWXHKTJJSQR
|
8.5 | IC50 | 3 | Yes | |
VWDNDBICKRVFCP
|
8.5 | IC50 | 4 | — | |
DNLQIFRJOZJGCU
|
8.4 | IC50 | 6 | Yes | |
HBMCAYMASSWIBL
|
8.4 | IC50 | 3 | Yes | |
ZBRROTSBDAODQD
|
8.4 | IC50 | 7 | Yes | |
CDRJTNGWNAODES
|
8.4 | IC50 | 3 | Yes | |
NPWDRTZQIHHHNK
|
8.4 | IC50 | 2 | — | |
YISMQBFJYDFMAL
|
8.4 | IC50 | 46 | — | |
GCDSDVNITVBCDW
|
8.4 | IC50 | 17 | — | |
HUDVRTTVWXVPMO
|
8.4 | IC50 | 5 | — | |
ZJDFSJYCAFMEGH
|
8.4 | IC50 | 2 | Yes | |
BANXPZGDYGVXOC
|
8.4 | IC50 | 4 | — | |
BZPKVUCAGBEWOQ
|
8.4 | IC50 | 3 | — | |
BZUHVULXCGBRBT
|
8.4 | IC50 | 2 | — | |
CCRFXSGDDYALRL
|
8.4 | IC50 | 3 | — | |
DDKIKSYBXRUQAD
|
8.4 | IC50 | 2 | — | |
DUICXLIDQMBFRK
|
8.4 | IC50 | 3 | — | |
IICSZMDQEOSVKN
|
8.4 | IC50 | 3 | — | |
JBUBKVHDFJCRSZ
|
8.4 | IC50 | 3 | Yes | |
JIFZZVZROIFPKB
|
8.4 | IC50 | 5 | — | |
JLPAYKSYUUUWDC
|
8.4 | IC50 | 2 | — | |
KDRIQANXEFIHCL
|
8.4 | IC50 | 4 | — | |
KSUDUUBCXJUFRL
|
8.4 | Kd | 12 | — | |
KXZHSSMCHVENBJ
|
8.4 | IC50 | 3 | — | |
NJEBMDHGQZGODS
|
8.4 | IC50 | 2 | — | |
NKJNHXKAASJVEM
|
8.4 | IC50 | 3 | — | |
PILZXNUZIFIDSU
|
8.4 | IC50 | 3 | — | |
PITUMGJELDUJEZ
|
8.4 | IC50 | 3 | Yes | |
PRFGCHAHYIAXCL
|
8.4 | IC50 | 3 | Yes | |
QKZKUCIKRGDWHQ
|
8.4 | IC50 | 3 | — | |
RHCMQQAUBJPPPW
|
8.4 | IC50 | 4 | — | |
RHFWTFDTRBFIHU
|
8.4 | IC50 | 13 | Yes | |
SGVBVAOVXTWIJT
|
8.4 | IC50 | 3 | — | |
SUXYGJZMCWKJJI
|
8.4 | IC50 | 26 | Yes | |
UUEYTEZBJWMVIQ
|
8.4 | IC50 | 5 | Yes | |
WLXUDQMWNQFZOR
|
8.4 | IC50 | 2 | — | |
YAQGBNTVJOCPCH
|
8.4 | IC50 | 2 | Yes | |
ZBTLTVIYBHYEHL
|
8.4 | IC50 | 13 | Yes | |
ZUMNLSFJINJANM
|
8.4 | IC50 | 5 | Yes | |
AJVISBGKRJRTQV
|
8.4 | IC50 | 2 | — | |
HVZJCIZSFTWSMN
|
8.4 | IC50 | 2 | — | |
SIUNALDMRGZQBR
|
8.4 | IC50 | 3 | — |