Target Details
| UniProt AC | P12931 |
|---|---|
| Gene Symbol | SRC |
| Protein Name | Proto-oncogene tyrosine-protein kinase Src |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,978
- Clinical molecules 816
- Avg pChEMBL 7.32
KEGG Pathways (45)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Bladder cancer
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- ErbB signaling pathway
- Estrogen signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- GnRH signaling pathway
- Hepatitis B
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Mitophagy - animal
- Neutrophil extracellular trap formation
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Platelet activation
- Prolactin signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Shigellosis
- Thyroid hormone signaling pathway
- Tight junction
- Tuberculosis
- VEGF signaling pathway
- Viral carcinogenesis
- Yersinia infection
Associated Diseases (2)
Active Molecules (1,978)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UBPYILGKFZZVDX
|
8.7 | IC50 | 130 | Yes | |
UDVSRXQVDHWZAL
|
8.7 | IC50 | 4 | — | |
VXMFHVFTECVHPF
|
8.7 | IC50 | 4 | — | |
WSBZFFNSBMBYQA
|
8.7 | IC50 | 9 | — | |
XGOUHJLISKQBDN
|
8.7 | IC50 | 4 | — | |
XHBVYDAKJHETMP
|
8.7 | IC50 | 24 | Yes | |
YCWQIUKZOZXDEM
|
8.7 | IC50 | 3 | — | |
YOVKYZJMWCAPJA
|
8.7 | IC50 | 3 | Yes | |
ZDUVJFVCYPQWGC
|
8.7 | IC50 | 2 | — | |
ZFAJIINWCGZNAM
|
8.7 | IC50 | 3 | — | |
ZGECDOGOLBHKSC
|
8.7 | IC50 | 3 | — | |
ZGVCPFSIDNPESN
|
8.7 | IC50 | 2 | — | |
KQEWHGHWFIFGMR
|
8.7 | IC50 | 2 | Yes | |
ZTQOHJNXDAUMOA
|
8.7 | IC50 | 13 | Yes | |
VCIZYTQJDGPPDJ
|
8.6 | IC50 | 6 | — | |
QRCADIJQEQMSLL
|
8.6 | IC50 | 2 | — | |
IHWCITLWMVRUQP
|
8.6 | IC50 | 2 | Yes | |
MEBNSJCLFXPYII
|
8.6 | IC50 | 3 | Yes | |
OUKYUETWWIPKQR
|
8.6 | IC50 | 31 | Yes | |
QXWCRBMAGJJKTO
|
8.6 | IC50 | 4 | Yes | |
DKNHELJFXSXKQW
|
8.5 | IC50 | 2 | — | |
LXJWUNONOVIADV
|
8.5 | IC50 | 2 | Yes | |
BEMAXRGCROABFF
|
8.5 | IC50 | 4 | — | |
CNPBEBBPEAKVJZ
|
8.5 | IC50 | 3 | — | |
GOMLJGVTZFYKJG
|
8.5 | IC50 | 3 | — | |
JCSZOMMQIMMAMS
|
8.5 | IC50 | 4 | — | |
JSEJMGKNQGRPEI
|
8.5 | IC50 | 3 | — | |
JTERLHICJVJIRK
|
8.5 | IC50 | 3 | — | |
JVEOZYRULRDCNQ
|
8.5 | IC50 | 3 | — | |
LYADGAGFYYXXIO
|
8.5 | IC50 | 82 | — | |
MBWHJBDHRADERX
|
8.5 | IC50 | 4 | — | |
NMCRRFLWJZUPRE
|
8.5 | IC50 | 5 | Yes | |
NMSHJWKGPWRUSI
|
8.5 | IC50 | 2 | — | |
NXTAONONNMIHOO
|
8.5 | IC50 | 3 | — | |
OGPRLOXNJCGODW
|
8.5 | IC50 | 2 | Yes | |
OGQDHXGPFCDXGA
|
8.5 | IC50 | 4 | — | |
POOFOKSCEYCHJC
|
8.5 | IC50 | 3 | — | |
RCPBXCJRKDXEGJ
|
8.5 | IC50 | 4 | — | |
RPFSNCZTTYGYDI
|
8.5 | IC50 | 3 | — | |
SBPZUKWJUJSFQT
|
8.5 | IC50 | 2 | Yes | |
TYCSETQHBQUZAZ
|
8.5 | IC50 | 3 | — | |
URRPWKVYUYOQBW
|
8.5 | IC50 | 3 | — | |
VARYUMXVRFFXLR
|
8.5 | IC50 | 3 | — | |
YBFJEMNJNCMXOO
|
8.5 | IC50 | 3 | — | |
YGZKTIVAVURWEZ
|
8.5 | IC50 | 3 | — | |
YHVHYWYQEFELOW
|
8.5 | IC50 | 44 | — | |
ZJPSMPSDMNGXHT
|
8.5 | IC50 | 2 | — | |
GPTPEUDRFUOZSX
|
8.5 | IC50 | 2 | — | |
HUZDGCVNDDSQGA
|
8.5 | IC50 | 6 | Yes | |
ZMNWFTYYYCSSTF
|
8.5 | Ki | 18 | — |