Target Details
| UniProt AC | P12931 |
|---|---|
| Gene Symbol | SRC |
| Protein Name | Proto-oncogene tyrosine-protein kinase Src |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,978
- Clinical molecules 816
- Avg pChEMBL 7.32
KEGG Pathways (45)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Bladder cancer
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- ErbB signaling pathway
- Estrogen signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- GnRH signaling pathway
- Hepatitis B
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Mitophagy - animal
- Neutrophil extracellular trap formation
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Platelet activation
- Prolactin signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Shigellosis
- Thyroid hormone signaling pathway
- Tight junction
- Tuberculosis
- VEGF signaling pathway
- Viral carcinogenesis
- Yersinia infection
Associated Diseases (2)
Active Molecules (1,978)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YWBUMBUFDDSLCR
|
9.0 | IC50 | 4 | — | |
DCIXGXIYPVJPIL
|
9.0 | IC50 | 2 | Yes | |
SUGCHLACYQMXHH
|
9.0 | IC50 | 2 | Yes | |
WJNXCARNBUNEMQ
|
9.0 | IC50 | 2 | Yes | |
JTWMOWRMSZZHDR
|
8.9 | IC50 | 13 | — | |
SWPUVWWNIQGBGY
|
8.9 | IC50 | 2 | Yes | |
YZLLDEHDOHFUOU
|
8.9 | IC50 | 2 | Yes | |
DFYOVMKHYAWORB
|
8.9 | IC50 | 3 | Yes | |
NSUVVSKQZKQXTP
|
8.9 | IC50 | 2 | Yes | |
ZCWXCBKGPJOAFQ
|
8.9 | IC50 | 13 | — | |
MFDCEMLTTQCDTH
|
8.8 | IC50 | 3 | Yes | |
UZWNDXWGPCUGGI
|
8.8 | IC50 | 2 | Yes | |
ZHRFIVBJJFVCEO
|
8.8 | IC50 | 2 | Yes | |
OLGSVSPNJXGSAD
|
8.8 | IC50 | 5 | Yes | |
QAMUWRFOZKONDU
|
8.8 | IC50 | 7 | — | |
ZWEHYQSGMOUIRZ
|
8.8 | IC50 | 3 | — | |
AQSSMEORRLJZLU
|
8.8 | IC50 | 34 | Yes | |
GJTWFSFZLIOXFD
|
8.8 | IC50 | 2 | Yes | |
KSCBSHLEWGZVON
|
8.8 | IC50 | 4 | — | |
XSYZCQDIHCJKAQ
|
8.8 | IC50 | 2 | — | |
HMQAQKDHRMARNF
|
8.8 | IC50 | 2 | Yes | |
KIHQVERTLRHJED
|
8.8 | IC50 | 2 | — | |
ZMNWHIBSNZMHFB
|
8.7 | IC50 | 2 | Yes | |
ALNFKLJYTICTCF
|
8.7 | IC50 | 4 | — | |
BMHCYYLFLWTPHZ
|
8.7 | IC50 | 4 | Yes | |
BPJALVMFXXJAJS
|
8.7 | IC50 | 3 | — | |
CEINQDWSZHAZSK
|
8.7 | IC50 | 2 | — | |
CGXCGLMVTWFROO
|
8.7 | IC50 | 4 | — | |
CLESKVZBGDCDJJ
|
8.7 | IC50 | 3 | — | |
COAQRADEUYYCDG
|
8.7 | IC50 | 12 | Yes | |
CZZVNONIDUMKCY
|
8.7 | IC50 | 2 | — | |
DQLUUNQMRQJPAL
|
8.7 | IC50 | 3 | — | |
DVMBLTDKHALLLH
|
8.7 | IC50 | 6 | Yes | |
DVRSTRMZTAPMKO
|
8.7 | IC50 | 10 | Yes | |
GWYGTWXYFRMPAH
|
8.7 | IC50 | 3 | Yes | |
HFGUPJNHEPCEHX
|
8.7 | IC50 | 3 | — | |
JOEZGPVMIDNCJZ
|
8.7 | IC50 | 5 | Yes | |
KNARVZUUCLIBGV
|
8.7 | Ki | 33 | — | |
LGACHOLIGNCDSQ
|
8.7 | IC50 | 4 | — | |
LHYKFLNJIXCRLM
|
8.7 | IC50 | 4 | — | |
LQSGDXCDNZWTJN
|
8.7 | IC50 | 17 | — | |
LUNIPUNUORVVSN
|
8.7 | IC50 | 4 | — | |
NEXHUYYIABFLMP
|
8.7 | IC50 | 2 | — | |
OCGMYHIDTHTZSV
|
8.7 | IC50 | 4 | — | |
OJKGJLKJOICLKA
|
8.7 | IC50 | 4 | — | |
OKERWTBOFAFQQV
|
8.7 | IC50 | 3 | — | |
OOVTWDNYKGHGHW
|
8.7 | IC50 | 2 | — | |
QJIXTISVQSBZTF
|
8.7 | IC50 | 3 | — | |
RIQXNLIRMOIENV
|
8.7 | IC50 | 4 | — | |
RNGNGIHVGNTTHO
|
8.7 | IC50 | 3 | — |