Target Details
| UniProt AC | P12931 |
|---|---|
| Gene Symbol | SRC |
| Protein Name | Proto-oncogene tyrosine-protein kinase Src |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,978
- Clinical molecules 816
- Avg pChEMBL 7.32
KEGG Pathways (45)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Bladder cancer
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- ErbB signaling pathway
- Estrogen signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- GnRH signaling pathway
- Hepatitis B
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Mitophagy - animal
- Neutrophil extracellular trap formation
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Platelet activation
- Prolactin signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Shigellosis
- Thyroid hormone signaling pathway
- Tight junction
- Tuberculosis
- VEGF signaling pathway
- Viral carcinogenesis
- Yersinia infection
Associated Diseases (2)
Active Molecules (1,978)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VKEOUSNQAFAOAA
|
7.6 | IC50 | 3 | — | |
YNSRIXGBOYZSBO
|
7.6 | IC50 | 3 | — | |
YVMCTVCGSKMRCI
|
7.6 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
7.6 | Kd | 154 | — | |
FWXVGKSWZJEPQI
|
7.6 | IC50 | 5 | — | |
JDAQJEHWJCXAFI
|
7.6 | IC50 | 4 | — | |
JOUPQTNCMDHNRF
|
7.6 | IC50 | 4 | — | |
KDECLMGBTBGDLA
|
7.6 | IC50 | 3 | — | |
KUMLEJXITHSWSP
|
7.6 | IC50 | 9 | Yes | |
SHEWRCTXFWSZHA
|
7.6 | IC50 | 3 | — | |
YQWRDEHPSFGGHV
|
7.6 | IC50 | 4 | Yes | |
YRRHAVKHTFWTLV
|
7.6 | IC50 | 3 | Yes | |
ZAPMLUQRTGRJST
|
7.6 | IC50 | 3 | — | |
BSTCRUFJLBKYMG
|
7.6 | IC50 | 4 | — | |
JBJNZQXRYXXLDI
|
7.6 | IC50 | 3 | — | |
MCCCQFAOMZMZKE
|
7.6 | Ki | 52 | — | |
QGDUHRXRHUCXIQ
|
7.6 | IC50 | 3 | — | |
RXNGGTYNZUEFOM
|
7.6 | IC50 | 8 | Yes | |
ULHGAQSVFPOUDY
|
7.6 | Ki | 43 | — | |
UOOZSMNSBYVUGZ
|
7.6 | Ki | 32 | — | |
XKZINYYXWJEYEL
|
7.6 | Ki | 37 | — | |
YJNVZAXZUDOAAI
|
7.6 | IC50 | 10 | Yes | |
BHNGTBAKKDCSHZ
|
7.6 | IC50 | 3 | — | |
NEKBJPNERWJTIC
|
7.6 | IC50 | 2 | — | |
OVTSFQUFYKJILE
|
7.6 | IC50 | 3 | Yes | |
RVVLIQXYHHNLCN
|
7.6 | IC50 | 3 | — | |
VWGMFKBQYRNIIN
|
7.6 | IC50 | 3 | — | |
XHHRGYCOEVNAKV
|
7.6 | Ki | 6 | Yes | |
DOMOLNAWFSVTTI
|
7.6 | IC50 | 3 | — | |
FWBIASCKMYRNDJ
|
7.6 | IC50 | 3 | — | |
NSVUVPGLZGFORM
|
7.6 | IC50 | 3 | — | |
OKFFBZNIDUDHDR
|
7.6 | IC50 | 3 | — | |
RPKWQQFQJOCDPR
|
7.6 | IC50 | 2 | — | |
XHHBBSIBRLADLF
|
7.6 | IC50 | 3 | Yes | |
XHKFYFCKCXKVPO
|
7.6 | IC50 | 5 | — | |
XSINXQGWUBFCGP
|
7.6 | IC50 | 3 | — | |
YSFGCARYACLFDS
|
7.6 | Ki | 7 | Yes | |
AHJRPTVABKSPBA
|
7.6 | IC50 | 3 | — | |
MMXSCACHGJJWPP
|
7.6 | IC50 | 2 | Yes | |
BJJRLHLFUBMTBH
|
7.5 | IC50 | 3 | — | |
NTRGHFKSGIJGAD
|
7.5 | IC50 | 3 | — | |
OUROWULXWNIHIF
|
7.5 | IC50 | 4 | — | |
PQZDDSNPXGLODE
|
7.5 | IC50 | 3 | Yes | |
RXXPIRGHDOIFNF
|
7.5 | IC50 | 3 | — | |
UPDASDRUBVHIJS
|
7.5 | IC50 | 4 | — | |
UYBFGBPGWZDBPF
|
7.5 | IC50 | 3 | — | |
XFVXNAQMQOCOEI
|
7.5 | IC50 | 2 | — | |
ZBQANXLXZIWFJV
|
7.5 | IC50 | 3 | — | |
AEQLIHRFVYSWGR
|
7.5 | IC50 | 4 | — | |
DDNCDVXLOZYMSA
|
7.5 | IC50 | 3 | — |