Target Details
| UniProt AC | P12931 |
|---|---|
| Gene Symbol | SRC |
| Protein Name | Proto-oncogene tyrosine-protein kinase Src |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,978
- Clinical molecules 816
- Avg pChEMBL 7.32
KEGG Pathways (45)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Bladder cancer
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- ErbB signaling pathway
- Estrogen signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- GnRH signaling pathway
- Hepatitis B
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Mitophagy - animal
- Neutrophil extracellular trap formation
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Platelet activation
- Prolactin signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Shigellosis
- Thyroid hormone signaling pathway
- Tight junction
- Tuberculosis
- VEGF signaling pathway
- Viral carcinogenesis
- Yersinia infection
Associated Diseases (2)
Active Molecules (1,978)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PXOGHMDWJDTSBR
|
7.8 | IC50 | 2 | — | |
QAKIGHBHPHZCJC
|
7.8 | IC50 | 4 | — | |
RBXYGQNZRVPDNB
|
7.8 | Ki | 34 | — | |
SCDTVQOOFJOJPO
|
7.8 | IC50 | 2 | — | |
SUCOEVXSLGWMLL
|
7.8 | IC50 | 3 | — | |
TWRMMAAINFMTFO
|
7.8 | IC50 | 3 | — | |
UDYNZGINEPJGRE
|
7.8 | IC50 | 2 | — | |
UUWNXFJBBYAMDT
|
7.8 | Ki | 46 | — | |
VAUWNNIXFMIEBF
|
7.8 | IC50 | 3 | — | |
VDYAAIDBWJMZBD
|
7.8 | IC50 | 3 | — | |
VSXCXKDGHBAKDZ
|
7.8 | IC50 | 3 | — | |
YKDLGDBIORZVLP
|
7.8 | IC50 | 10 | Yes | |
ZSUZNPQSAQRXJP
|
7.8 | IC50 | 4 | — | |
AFZKXALTXCNQAZ
|
7.8 | IC50 | 2 | Yes | |
LSTCMOOVQGRKHL
|
7.8 | IC50 | 2 | — | |
SLCFEJAMCRLYRG
|
7.8 | IC50 | 8 | Yes | |
DGUSFVFTIHATAT
|
7.8 | IC50 | 5 | Yes | |
FPWCREKHIZDTGO
|
7.8 | IC50 | 3 | — | |
GACWECUHBHHMBL
|
7.8 | IC50 | 3 | — | |
ICRKLHQKHODTLD
|
7.8 | IC50 | 4 | — | |
IPRGOVMOQCIUFP
|
7.8 | IC50 | 2 | — | |
IWGIXRMJMSKLGP
|
7.8 | IC50 | 4 | Yes | |
KIPZYDCBLYBUMY
|
7.8 | IC50 | 4 | — | |
KLCRZBNGDBKHFA
|
7.8 | IC50 | 4 | — | |
KUUKOPMICNKRGE
|
7.8 | IC50 | 12 | Yes | |
KWQYOKQSJYMUAF
|
7.8 | IC50 | 2 | — | |
LRJOPQDEHYLGQF
|
7.8 | Ki | 3 | — | |
LTNUJJDDRIVIPZ
|
7.8 | IC50 | 2 | — | |
LVURDXDDOIWLAP
|
7.8 | IC50 | 2 | — | |
MMBUUNLZGRAVKE
|
7.8 | IC50 | 3 | — | |
OXTMWMXCNQWAGP
|
7.8 | IC50 | 4 | — | |
RDUBHIVRDVFUBN
|
7.8 | IC50 | 2 | — | |
VPSLBUMYCILBRD
|
7.8 | IC50 | 8 | Yes | |
VYSNYHPSOJCNIW
|
7.8 | IC50 | 3 | — | |
ZSAJPWOGVMFXHN
|
7.8 | IC50 | 10 | Yes | |
HVKVREKLPAMYHA
|
7.8 | IC50 | 2 | Yes | |
NDUAHACMVSARNG
|
7.8 | IC50 | 4 | — | |
DAXOOIRHYYCDDH
|
7.8 | IC50 | 10 | Yes | |
JQGBWSRCIMCMTI
|
7.8 | IC50 | 2 | — | |
OUHRROUUMISCGY
|
7.8 | IC50 | 2 | — | |
BYRBUVTUGSOTSC
|
7.7 | IC50 | 7 | Yes | |
DANMJMQROKKATM
|
7.7 | IC50 | 3 | — | |
FZBVNCFBCNXULH
|
7.7 | IC50 | 18 | — | |
GPYGSYSPXHEXTJ
|
7.7 | IC50 | 3 | — | |
HKSWAIDHHZHZTD
|
7.7 | IC50 | 6 | — | |
KFXHPWUOUVDXSQ
|
7.7 | IC50 | 3 | — | |
MACKJBHSMLAAGO
|
7.7 | IC50 | 7 | Yes | |
NUCRGYCYHSHHCH
|
7.7 | IC50 | 3 | — | |
ORJLWELEFZSDSZ
|
7.7 | IC50 | 2 | — | |
RPHZNUQELARGGG
|
7.7 | IC50 | 3 | — |