Target Details
| UniProt AC | P12931 |
|---|---|
| Gene Symbol | SRC |
| Protein Name | Proto-oncogene tyrosine-protein kinase Src |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,978
- Clinical molecules 816
- Avg pChEMBL 7.32
KEGG Pathways (45)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Bladder cancer
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- ErbB signaling pathway
- Estrogen signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- GnRH signaling pathway
- Hepatitis B
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Mitophagy - animal
- Neutrophil extracellular trap formation
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Platelet activation
- Prolactin signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Shigellosis
- Thyroid hormone signaling pathway
- Tight junction
- Tuberculosis
- VEGF signaling pathway
- Viral carcinogenesis
- Yersinia infection
Associated Diseases (2)
Active Molecules (1,978)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QXWLCWKPJNSRRJ
|
7.8 | IC50 | 3 | — | |
UFDZZHKLIUCKGW
|
7.8 | IC50 | 3 | — | |
UMUNUYQBNZSRHV
|
7.8 | IC50 | 3 | — | |
VLRRDESRPRRNAD
|
7.8 | IC50 | 4 | — | |
WHPSRWXDXFWLHF
|
7.8 | IC50 | 3 | Yes | |
WLFMHNCEKPWCEA
|
7.8 | IC50 | 3 | Yes | |
XNODQMMIMXSTMX
|
7.8 | IC50 | 12 | Yes | |
YIDJUDDEOGSZCB
|
7.8 | IC50 | 2 | — | |
YVVSDMPVUOIAOS
|
7.8 | IC50 | 3 | — | |
ZNHAPHKYMMDRQX
|
7.8 | IC50 | 3 | — | |
BOQLSYBMPFBUNE
|
7.8 | IC50 | 4 | — | |
SSDFTYWIYVWCIE
|
7.8 | IC50 | 17 | — | |
AFFDEZDCXSAKBU
|
7.8 | IC50 | 4 | — | |
CLRSATALQPIPQY
|
7.8 | IC50 | 3 | — | |
DBSYRDKFSIDUKG
|
7.8 | IC50 | 2 | — | |
FAWGCSGOLCHXBH
|
7.8 | IC50 | 11 | Yes | |
FHNLPTRXVQOXQO
|
7.8 | IC50 | 11 | Yes | |
FLJSOYXRJCMRAE
|
7.8 | IC50 | 3 | — | |
FZHGLIPWYYRIRD
|
7.8 | IC50 | 3 | — | |
GGARDPUFELXEBN
|
7.8 | IC50 | 4 | — | |
HAVMBPZPTGEWPJ
|
7.8 | IC50 | 4 | — | |
HNDIVAFUXDXTDZ
|
7.8 | IC50 | 3 | — | |
JKRIGGIUXGQZRW
|
7.8 | IC50 | 2 | Yes | |
KEYJNCXZEKAAGP
|
7.8 | IC50 | 3 | — | |
KQSYWWGVMIWNOM
|
7.8 | IC50 | 3 | — | |
LJAUTNHJCPVWDZ
|
7.8 | IC50 | 3 | — | |
LJWVFWLHDDCALO
|
7.8 | IC50 | 3 | — | |
MDMCYZGIXLRATE
|
7.8 | IC50 | 4 | — | |
MWYBBCLGEHZSCP
|
7.8 | IC50 | 11 | Yes | |
PAZVWIGCRYUCKP
|
7.8 | IC50 | 4 | — | |
QEXJMEVOCZLJQX
|
7.8 | IC50 | 3 | — | |
QJLFDDXFGSEKEP
|
7.8 | IC50 | 3 | — | |
UFLGKZDFVFEGCP
|
7.8 | IC50 | 6 | Yes | |
VIFMVQBVAVNATG
|
7.8 | IC50 | 4 | — | |
VRCBGBBYFHLJRE
|
7.8 | IC50 | 5 | — | |
ZOJJTNITQOBIGV
|
7.8 | IC50 | 3 | — | |
ZGYGQOBLWQGUEB
|
7.8 | IC50 | 2 | — | |
AJOLXGKMRXNPKQ
|
7.8 | IC50 | 4 | — | |
AWWZYQVCCFNGQX
|
7.8 | IC50 | 2 | Yes | |
BLQYVHBZHAISJM
|
7.8 | IC50 | 54 | — | |
DAXMIVDYBBFSGN
|
7.8 | IC50 | 4 | — | |
DFSRCPBSJAXTNU
|
7.8 | IC50 | 3 | — | |
HWLWBINIXVPIHY
|
7.8 | IC50 | 3 | — | |
HZKOUKPIDXDOOI
|
7.8 | IC50 | 4 | — | |
JJHRHADNFSGPGT
|
7.8 | IC50 | 2 | — | |
MHCPAORAYMTGCZ
|
7.8 | Ki | 37 | — | |
ODPFOHRTWMCIJT
|
7.8 | IC50 | 3 | — | |
OJWPICIEUSPJKT
|
7.8 | IC50 | 3 | Yes | |
OOLMBUKZNOBEOR
|
7.8 | IC50 | 3 | — | |
PTMVPXQFPYJIMN
|
7.8 | IC50 | 4 | — |