Target Details
| UniProt AC | P12931 |
|---|---|
| Gene Symbol | SRC |
| Protein Name | Proto-oncogene tyrosine-protein kinase Src |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,978
- Clinical molecules 816
- Avg pChEMBL 7.32
KEGG Pathways (45)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Bladder cancer
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- ErbB signaling pathway
- Estrogen signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- GnRH signaling pathway
- Hepatitis B
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Mitophagy - animal
- Neutrophil extracellular trap formation
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Platelet activation
- Prolactin signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Shigellosis
- Thyroid hormone signaling pathway
- Tight junction
- Tuberculosis
- VEGF signaling pathway
- Viral carcinogenesis
- Yersinia infection
Associated Diseases (2)
Active Molecules (1,978)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XIJQHLBJFSYQQB
|
7.9 | IC50 | 2 | — | |
YBQBWKIOPABUPG
|
7.9 | IC50 | 2 | — | |
YDEDKRCWCCZXBE
|
7.9 | IC50 | 2 | — | |
YXGPQZLIIOQQAZ
|
7.9 | IC50 | 2 | — | |
ZOJRUPGIRXZFTR
|
7.9 | IC50 | 3 | — | |
ZPKGDYKWVKCDJQ
|
7.9 | IC50 | 4 | Yes | |
NYCMTZDIVLFLKV
|
7.9 | IC50 | 3 | — | |
TXIHQMLNWLFVHM
|
7.9 | IC50 | 6 | Yes | |
ZDZUIAHQMAWKQF
|
7.9 | IC50 | 2 | — | |
LGMDJFPPNVPECO
|
7.9 | IC50 | 3 | Yes | |
SRUYMJRFVGLQDV
|
7.9 | Ki | 37 | — | |
UGEJLCNSVIVALC
|
7.9 | Ki | 41 | — | |
WQACVRFKZIYHIM
|
7.9 | IC50 | 3 | Yes | |
FJCORFQIRVXPCY
|
7.9 | IC50 | 4 | — | |
HUNGUWOZPQBXGX
|
7.9 | IC50 | 4 | — | |
IBRPSHUYWHRYQA
|
7.9 | IC50 | 4 | Yes | |
IRXWZAWSUMZCBD
|
7.9 | IC50 | 3 | — | |
KBDMNNVCGCQHGS
|
7.9 | IC50 | 3 | — | |
KFKOANBFFZCCOA
|
7.9 | IC50 | 2 | — | |
KKYYLKPGILUPOA
|
7.9 | IC50 | 2 | — | |
KPESYVJNOVNDGE
|
7.9 | IC50 | 4 | — | |
KSCDJRWPBJOREH
|
7.9 | IC50 | 3 | — | |
MAXZESONWXTISA
|
7.9 | IC50 | 3 | — | |
MCPXUGGNYXHTMJ
|
7.9 | IC50 | 2 | — | |
PSPWDUMROPJEGG
|
7.9 | IC50 | 3 | — | |
QSECCHMWSVTBKZ
|
7.9 | IC50 | 4 | Yes | |
RPZCFPLDPHTRPE
|
7.9 | Ki | 3 | — | |
URFCMVULTIAJNO
|
7.9 | IC50 | 2 | — | |
VSQDAQJVIALSGZ
|
7.9 | IC50 | 3 | — | |
YAFBWUKWKZZPIF
|
7.9 | IC50 | 4 | Yes | |
YTFOAGDDMAAOPC
|
7.9 | IC50 | 3 | — | |
ZAAKPRKYIFTIIV
|
7.9 | IC50 | 3 | — | |
ZZUSFIPRLCGKQL
|
7.9 | IC50 | 4 | — | |
BLQYVHBZHAISJM
|
7.8 | IC50 | 21 | Yes | |
DFMFALRCABNVBW
|
7.8 | IC50 | 3 | — | |
DSQCTESAPJCINY
|
7.8 | IC50 | 3 | — | |
DTFJTXRGYIXMMS
|
7.8 | IC50 | 5 | — | |
DTGGTIWRYHDYPL
|
7.8 | IC50 | 4 | — | |
FCHGXFUOVXKORC
|
7.8 | IC50 | 2 | — | |
HYWXBDQAYLPMIX
|
7.8 | IC50 | 3 | Yes | |
ICOQLVRSRCFGJB
|
7.8 | IC50 | 3 | — | |
IEHFKZAAIWSDQM
|
7.8 | IC50 | 3 | — | |
MRZVUZUMBCEAGI
|
7.8 | IC50 | 11 | Yes | |
NVRXTLZYXZNATH
|
7.8 | IC50 | 47 | Yes | |
OFTHCDFOVLVBTL
|
7.8 | IC50 | 3 | — | |
ONBCGBVSJRMMHE
|
7.8 | IC50 | 2 | — | |
PUDBISUVQGIKBD
|
7.8 | IC50 | 4 | — | |
QFXFIEVXAUEHEV
|
7.8 | IC50 | 6 | — | |
QGMACHJORMNYMR
|
7.8 | IC50 | 3 | Yes | |
QVJHVQPCRIXTMX
|
7.8 | IC50 | 3 | — |