Target Details
| UniProt AC | P12931 |
|---|---|
| Gene Symbol | SRC |
| Protein Name | Proto-oncogene tyrosine-protein kinase Src |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,978
- Clinical molecules 816
- Avg pChEMBL 7.32
KEGG Pathways (45)
- Adherens junction
- Axon guidance
- Bacterial invasion of epithelial cells
- Bladder cancer
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- ErbB signaling pathway
- Estrogen signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- GABAergic synapse
- Gap junction
- GnRH signaling pathway
- Hepatitis B
- Herpes simplex virus 1 infection
- Hormone signaling
- Human cytomegalovirus infection
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Mitophagy - animal
- Neutrophil extracellular trap formation
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Platelet activation
- Prolactin signaling pathway
- Proteoglycans in cancer
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Shigellosis
- Thyroid hormone signaling pathway
- Tight junction
- Tuberculosis
- VEGF signaling pathway
- Viral carcinogenesis
- Yersinia infection
Associated Diseases (2)
Active Molecules (1,978)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UDUPSRWUDACGIS
|
9.9 | IC50 | 13 | Yes | |
ANWHQLGKGDJLJO
|
9.7 | IC50 | 6 | — | |
BPLTVYXMXOYIBK
|
9.7 | IC50 | 9 | — | |
BPLTVYXMXOYIBK
|
9.7 | IC50 | 6 | — | |
HJVDQPRJANOXIX
|
9.7 | IC50 | 10 | — | |
VYEYNLSRVXXGPW
|
9.6 | Ki | 2 | — | |
IWBVZILESKBVJL
|
9.4 | IC50 | 6 | — | |
DOBZFFWLHXORTB
|
9.3 | Ki | 2 | — | |
UNZHPVUBBKLAJR
|
9.3 | IC50 | 6 | Yes | |
PQRFMBAACAPZPP
|
9.3 | IC50 | 12 | Yes | |
QQHSTSLAVGUPKP
|
9.2 | IC50 | 3 | — | |
SYWUIAOLWMUYTP
|
9.2 | IC50 | 3 | — | |
RWKFWKPIQLFUQP
|
9.2 | IC50 | 6 | — | |
ZTNMLIDOCZAAEX
|
9.2 | IC50 | 2 | Yes | |
CSXVLYGUGWXOAL
|
9.2 | IC50 | 2 | — | |
GCFYFSXVZCZHBK
|
9.1 | IC50 | 2 | Yes | |
XHRFFDAZHQMDPM
|
9.1 | IC50 | 3 | Yes | |
ANUHLKPVOXDYSK
|
9.1 | IC50 | 5 | Yes | |
BIEFBSIFAKMKOT
|
9.1 | IC50 | 2 | Yes | |
ZKQTVBGLURSDIR
|
9.1 | Ki | 2 | — | |
CXBBWVXSZINRCS
|
9.1 | Ki | 41 | — | |
GMPQGWXPDRNCBL
|
9.1 | Ki | 4 | — | |
JYRRZNYFIFNIGM
|
9.1 | IC50 | 2 | Yes | |
QGFOJZMDPXDGSA
|
9.1 | IC50 | 3 | — | |
ZBNZXTGUTAYRHI
|
9.1 | IC50 | 102 | Yes | |
WFQCEVIDLOLEDG
|
9.1 | IC50 | 5 | — | |
JCNVRKBMXOPADG
|
9.1 | Ki | 2 | — | |
BMJIPGXVDYVSGD
|
9.1 | IC50 | 4 | — | |
HHOVYYSFRMBKPP
|
9.1 | IC50 | 3 | Yes | |
CZCGARLOFSDTBA
|
9.0 | Ki | 2 | — | |
RDTFOUQPUVOZQZ
|
9.0 | IC50 | 2 | Yes | |
UUDPUQDMSHQSKH
|
9.0 | IC50 | 3 | — | |
BAIXSQGNLALLTR
|
9.0 | IC50 | 4 | — | |
BRACWNNBDWUPJC
|
9.0 | IC50 | 2 | — | |
CHWHVQUNCYDPDK
|
9.0 | IC50 | 6 | Yes | |
CRLZGLXSANQWFT
|
9.0 | IC50 | 6 | — | |
FFPDTHQSUMBEBA
|
9.0 | IC50 | 2 | — | |
HKBVCGJVIFGBEX
|
9.0 | IC50 | 6 | Yes | |
HOBGSWDBYMRRJR
|
9.0 | IC50 | 4 | — | |
KKBSRZBNVASLTJ
|
9.0 | IC50 | 3 | — | |
MBPKPSDAPFPECJ
|
9.0 | IC50 | 12 | Yes | |
NJKRMPNUGZAMJN
|
9.0 | IC50 | 5 | — | |
PVVFFEVERRIBNR
|
9.0 | IC50 | 3 | — | |
QRDWGUVCGQETNO
|
9.0 | IC50 | 4 | Yes | |
RASCHEQRJMEENP
|
9.0 | IC50 | 4 | — | |
VOURYMYVBGIOOG
|
9.0 | IC50 | 2 | — | |
VSJXTUFWPAOYLC
|
9.0 | IC50 | 11 | Yes | |
WCTNEALHPXRJMI
|
9.0 | IC50 | 3 | — | |
WJSCDYSIDGEWEB
|
9.0 | IC50 | 5 | Yes | |
XUIJEFBUBZVZFL
|
9.0 | IC50 | 4 | — |