Target Details
| UniProt AC | P12497 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate NY5) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 454
- Clinical molecules 0
- Avg pChEMBL 8.33
Active Molecules (454)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WZRBCRPZAJNYRP
|
6.8 | IC50 | 2 | — | |
WEFMCBSODKDJFB
|
6.8 | IC50 | 2 | — | |
UXIVWMINNPGARX
|
6.7 | IC50 | 3 | — | |
LUICRMGYHPZLQE
|
6.7 | IC50 | 2 | — | |
QPKRELCYQDFLQW
|
6.7 | IC50 | 2 | — | |
KOHJMQXAUBCBFT
|
6.7 | IC50 | 2 | — | |
VKHXZIVZQNBARO
|
6.7 | Ki | 2 | — | |
CFKNTKGMEUMOTC
|
6.7 | IC50 | 2 | — | |
JGNJWIIHVZPCLO
|
6.7 | IC50 | 2 | — | |
LCUWRKGCTXXCBV
|
6.7 | Ki | 2 | — | |
KFGIHCFGDLBYGM
|
6.7 | IC50 | 2 | — | |
SFUSYMKBUIQBHK
|
6.7 | IC50 | 2 | — | |
ZLYKUIUJEAYAOR
|
6.7 | IC50 | 2 | — | |
HZUCRWWOEVMAPC
|
6.6 | Ki | 2 | — | |
JRGKTJWRQVHKOO
|
6.6 | IC50 | 2 | — | |
PKNSWTXTLSKLHZ
|
6.6 | Ki | 2 | — | |
JYCRZVGDFQMBST
|
6.6 | IC50 | 2 | — | |
PIVCSFQAABPVOR
|
6.6 | IC50 | 2 | — | |
SYMCBBYJOYFSNB
|
6.5 | IC50 | 2 | — | |
VERMKZUVUYNLHI
|
6.5 | IC50 | 2 | — | |
WAQDMMDIFOJGCP
|
6.5 | IC50 | 2 | — | |
XCSQTRCCSZFEKV
|
6.5 | IC50 | 2 | — | |
XOMLSGLFNOYRSP
|
6.5 | IC50 | 2 | — | |
WNDVEZVRDLTINH
|
6.5 | IC50 | 2 | — | |
WSMLOMCZUGUJEP
|
6.5 | IC50 | 2 | — | |
ZOYPQZASFVMBOQ
|
6.5 | Ki | 2 | — | |
PYGWGZALEOIKDF
|
6.4 | IC50 | 5 | — | |
MXNDJZKEFYGXNY
|
6.4 | IC50 | 2 | — | |
OJWIIEFLUZBLJI
|
6.4 | IC50 | 2 | — | |
HFYNRTHTPCWYOT
|
6.4 | IC50 | 2 | — | |
QPXSFMLHUCDSGF
|
6.4 | IC50 | 2 | — | |
WAHBCPQDHASNLU
|
6.4 | IC50 | 2 | — | |
XFVAZZZKQWGAJJ
|
6.4 | IC50 | 2 | — | |
PCEGWKGFACRWOO
|
6.4 | IC50 | 2 | — | |
ZIUYNDNWGWCFJI
|
6.4 | IC50 | 2 | — | |
AAYIGYNCAMMVQJ
|
6.3 | IC50 | 2 | — | |
LHQZYXZCDMXJLV
|
6.3 | Ki | 2 | — | |
OAXPPAUXOZJCFF
|
6.3 | Ki | 2 | — | |
XWEQBHNRDFTICX
|
6.3 | IC50 | 2 | — | |
DPYHGUIDBOZDPO
|
6.3 | IC50 | 2 | — | |
NIBXFUBAUTVIGY
|
6.3 | Ki | 2 | — | |
CCPGCKQLIHGSCJ
|
6.2 | Ki | 2 | — | |
HZUCRWWOEVMAPC
|
6.2 | Ki | 2 | — | |
PCZZRLMYGNFQOV
|
6.2 | Ki | 2 | — | |
UAWPOYVQIDXTLH
|
6.2 | Ki | 2 | — | |
BNDPDYQQAJUJPY
|
6.2 | IC50 | 2 | — | |
CKOGZEIBYRMITE
|
6.2 | IC50 | 2 | — | |
ZLSNKTCBGPUFEX
|
6.2 | IC50 | 2 | — | |
BPEXGZSFDTVMDJ
|
6.2 | IC50 | 2 | — | |
ATVGQDPVWYFCCA
|
6.1 | IC50 | 2 | — |