Target Details
| UniProt AC | P12497 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate NY5) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 454
- Clinical molecules 0
- Avg pChEMBL 8.33
Active Molecules (454)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GIJVOAULRYJRGU
|
7.2 | IC50 | 2 | — | |
KWDFBFZCEVNAHE
|
7.2 | Ki | 2 | — | |
RVHWPGAHEOLZNT
|
7.2 | IC50 | 2 | — | |
JADNFEPHYDBRDW
|
7.2 | Ki | 2 | — | |
HZUCRWWOEVMAPC
|
7.2 | Ki | 2 | — | |
IAXLWGCXGGUUOU
|
7.2 | IC50 | 2 | — | |
LLVJVNVNDLXYES
|
7.2 | IC50 | 2 | — | |
MQGFJXIGONAWLT
|
7.2 | Ki | 2 | — | |
WWJIOVFCXOTDHG
|
7.2 | Ki | 2 | — | |
RGTBPOJAPDHIJT
|
7.2 | IC50 | 2 | — | |
VASWCZNNYHXDLS
|
7.2 | IC50 | 2 | — | |
JGNJWIIHVZPCLO
|
7.2 | IC50 | 2 | — | |
KPWCKNINNOIZFO
|
7.2 | IC50 | 2 | — | |
OQICOQSTWCHGKT
|
7.1 | IC50 | 2 | — | |
XWGIKPIIQBFYGG
|
7.1 | IC50 | 2 | — | |
IKUFDUQKHKVTGZ
|
7.1 | IC50 | 2 | — | |
SJLKQIOVIJCRQA
|
7.1 | IC50 | 2 | — | |
KMGABVMIQPZZHU
|
7.1 | IC50 | 2 | — | |
VZLVYEBEUCOLCO
|
7.1 | IC50 | 2 | — | |
CRSBLGVQVRTNCO
|
7.1 | IC50 | 2 | — | |
GVGIURATDJMDNM
|
7.1 | IC50 | 2 | — | |
SGSVELRCCSUWEU
|
7.1 | IC50 | 2 | — | |
WVVSZAZDAIVXOJ
|
7.1 | Ki | 2 | — | |
AWHVBBSGHXQION
|
7.0 | Ki | 2 | — | |
CKXAPPBTNSDDKV
|
7.0 | IC50 | 2 | — | |
MMKHYVMEYOSGDI
|
7.0 | IC50 | 2 | — | |
NHMIHQZMBYIQSR
|
7.0 | IC50 | 2 | — | |
OQHZMGOXOOOFEE
|
7.0 | IC50 | 2 | — | |
QVGOLNUEBCOLGS
|
7.0 | IC50 | 2 | — | |
RCFQGEMHANXIRS
|
7.0 | IC50 | 2 | — | |
YDXWVSNLNBSYOF
|
7.0 | IC50 | 2 | — | |
ICTQRPRKGRPVHA
|
7.0 | Ki | 2 | — | |
GHXMNIYXDTYJRJ
|
7.0 | Ki | 2 | — | |
SDOJFPSFHFRQPP
|
7.0 | IC50 | 2 | — | |
BHYLXIUVVRJDMP
|
6.9 | IC50 | 2 | — | |
IWDXCNVEWVCNBM
|
6.9 | IC50 | 2 | — | |
GAAOWWZYXBJCRW
|
6.9 | IC50 | 2 | — | |
SCFUZBGSNDDHBF
|
6.9 | IC50 | 2 | — | |
SFUSYMKBUIQBHK
|
6.9 | IC50 | 2 | — | |
DKGUABRGUNATNU
|
6.9 | IC50 | 2 | — | |
DSQIWNUFPPHLBD
|
6.8 | IC50 | 2 | — | |
ZJWOSCDRPXZBJU
|
6.8 | IC50 | 2 | — | |
QQMCQOZEGIKRSY
|
6.8 | Ki | 2 | — | |
IHUPSDHNUJCYBF
|
6.8 | Ki | 2 | — | |
OWCCZVZPRSKALT
|
6.8 | Ki | 2 | — | |
GJUACQHGCKQUSS
|
6.8 | IC50 | 2 | — | |
ZWVMLEVADZPJBJ
|
6.8 | IC50 | 2 | — | |
DXXWPNILFQDFMJ
|
6.8 | Ki | 2 | — | |
KFGIHCFGDLBYGM
|
6.8 | IC50 | 2 | — | |
QPKRELCYQDFLQW
|
6.8 | IC50 | 2 | — |