Target Details
| UniProt AC | P12497 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate NY5) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 454
- Clinical molecules 0
- Avg pChEMBL 8.33
Active Molecules (454)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VMKIRLPDTOOXPM
|
7.7 | IC50 | 2 | — | |
NHGJCQDJVVIEHB
|
7.7 | Ki | 2 | — | |
BAEPUUWETTZONO
|
7.7 | Ki | 2 | — | |
HPNWNQXCBHLAEF
|
7.7 | IC50 | 2 | — | |
IJMLLSKOKKJLBX
|
7.7 | Ki | 2 | — | |
VEXRXPAIHVICKW
|
7.7 | Ki | 2 | — | |
SCVGALCLJNKWJI
|
7.7 | IC50 | 2 | — | |
DBZLZNFYSDUNIS
|
7.6 | Ki | 2 | — | |
UPWOUZDRKCEYPI
|
7.6 | IC50 | 2 | — | |
GFJUQXPENVFSPL
|
7.5 | Ki | 2 | — | |
UDBQSHPMEQJBIA
|
7.5 | Ki | 2 | — | |
IJBPAVCQGVFAKL
|
7.5 | IC50 | 2 | — | |
AEJMIBHXONFIJT
|
7.5 | IC50 | 2 | — | |
DDHUVWKEFAMGRB
|
7.5 | IC50 | 2 | — | |
SQBOSZXDOHQFAA
|
7.5 | IC50 | 2 | — | |
CLIJYYKSHOUGGU
|
7.5 | Ki | 2 | — | |
OOAVNTQEOJWXBW
|
7.5 | Ki | 2 | — | |
NNIGRBMKHHHZSZ
|
7.5 | Ki | 2 | — | |
NRHQSCBNXQVHDR
|
7.5 | IC50 | 2 | — | |
SJRFWBCULLJDGA
|
7.5 | Ki | 2 | — | |
VPXDKZOIMQMIRC
|
7.5 | Ki | 2 | — | |
YSNCNINOHAXGEF
|
7.4 | Ki | 2 | — | |
JQBRNXDUXTYTKY
|
7.4 | IC50 | 2 | — | |
JXCRNYYHOBWABD
|
7.4 | Ki | 2 | — | |
QOXURAUXAXPSPD
|
7.4 | IC50 | 2 | — | |
WGUDWHYBVHSPSU
|
7.4 | IC50 | 2 | — | |
XHDOJHIGYFGOND
|
7.4 | IC50 | 2 | — | |
BFFIPVLTEGEZDJ
|
7.4 | IC50 | 2 | — | |
GTGPHAUFYVHIIY
|
7.4 | Ki | 2 | — | |
HGZGSIWZDXBMDK
|
7.4 | IC50 | 2 | — | |
ITOFMHXYOAGPKK
|
7.4 | IC50 | 2 | — | |
SGPZLDNIZDMEIK
|
7.4 | IC50 | 2 | — | |
HIJDADBORWRDJP
|
7.4 | IC50 | 2 | — | |
RTXCQPDBXIDIQX
|
7.4 | Ki | 2 | — | |
NTNXTIVVNYYALB
|
7.3 | IC50 | 2 | — | |
SPEPPPKXFJRIFN
|
7.3 | IC50 | 2 | — | |
ZVWSWYSIMOZTTG
|
7.3 | IC50 | 2 | — | |
UPWOUZDRKCEYPI
|
7.3 | IC50 | 2 | — | |
VVYUNBWXGPXGBU
|
7.3 | IC50 | 2 | — | |
XGSPSWMOULVMMN
|
7.3 | IC50 | 2 | — | |
YTVUVKHREDAUGZ
|
7.3 | IC50 | 2 | — | |
NDRULGXLEDZQGT
|
7.3 | Ki | 2 | — | |
WZRBCRPZAJNYRP
|
7.3 | IC50 | 2 | — | |
DHQTXGHHAQJESR
|
7.3 | IC50 | 2 | — | |
JSHJDJSZOFESCN
|
7.2 | IC50 | 2 | — | |
SCXIXUQUBGZHMQ
|
7.2 | IC50 | 2 | — | |
KQBXKNMHEJHPCA
|
7.2 | IC50 | 2 | — | |
OFSZIOSVMKUCOI
|
7.2 | IC50 | 2 | — | |
SJFIXPJVPGUFKR
|
7.2 | Ki | 2 | — | |
DHGYJQQCTRWFTI
|
7.2 | IC50 | 2 | — |