Target Details
UniProt ACP12497
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate NY5)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 454
  • Clinical molecules 0
  • Avg pChEMBL 8.33
Top Co-occurrence Targets
Active Molecules (454)
InChIKey pChEMBL Type Targets Clinical
DXBMQQLBQTVBBQ 8.1 IC50 2
MMCLAFJWSPFWJN 8.1 Ki 2
XGJBWTYWJMOKBK 8.1 Ki 2
AYZGBDUXVJCUNJ 8.0 Ki 2
GWFKFFPLSALKEY 8.0 Ki 2
AUTHLCQFZJFGMT 8.0 Ki 2
AHMPQPOFMWFJEZ 8.0 IC50 3
FTSVRSRPVCKWHD 8.0 Ki 2
IHQOLDBRNQEINO 8.0 IC50 2
VOQZQCYEDQCVHB 8.0 Ki 2
BZKSWCPXTIIOKX 8.0 Ki 2
CGBDAHCDSVOMCF 8.0 Ki 2
CLDRSJNLDPCRJL 8.0 Ki 2
FDBMQZFGLNMCLV 8.0 Ki 2
ISGIGDDPEZVQPE 8.0 IC50 2
MHLNARDQQWONOV 8.0 IC50 2
ZWBLHWHBSYSDFK 7.9 IC50 2
AQMCGYBGJJWMDS 7.9 Ki 2
DWSUULFDMUNPJU 7.9 IC50 2
FACAUYLYCYUNSS 7.9 IC50 2
NKGCIFOXPWDDMH 7.9 IC50 2
CHZGNAXNHGNYFW 7.9 IC50 2
KHIFVRGSAUWJBP 7.9 Ki 2
TUHVTOYYHANQMW 7.9 Ki 2
KIUZLKJJOFIWAW 7.9 IC50 2
JMVUOXLBVAOZCN 7.8 Ki 2
UFCZJNJTAXXEEG 7.8 IC50 2
YLIMGTGTLQYCAA 7.8 IC50 2
NTNXTIVVNYYALB 7.8 IC50 2
XWYIBXKLXLXYMK 7.8 IC50 2
CUBGMDXVITWRSB 7.8 IC50 2
JLBJKFNEWPIYQA 7.8 IC50 2
QOWUCUBSJPNTJS 7.8 Ki 2
SEUIMKBYBKTVTL 7.8 Ki 2
SYHMSAYQDYUEPQ 7.8 IC50 2
BXHKUQJOWIKKIH 7.8 IC50 3
KPHRDRFCGGZQJY 7.8 Ki 2
LIQUANAIMCXRJS 7.7 Ki 2
MSPKBDSHENZXSJ 7.7 Ki 2
TYICRGMXQPUREK 7.7 Ki 2
LZNQWTXLCBDEDL 7.7 IC50 2
NLFFAUCKMYMCIL 7.7 IC50 2
PFVKUKWMVXMJNL 7.7 Ki 2
PYVYPFLWULRSGG 7.7 IC50 2
CMBBYMMNBCVVGO 7.7 IC50 2
OKLXJRBROSFVFX 7.7 IC50 2
RHMWHSCIEZRMHZ 7.7 IC50 2
XPOQHMRABVBWPR 7.7 IC50 5
MEWAZRJLRMEJDV 7.7 IC50 3
PRRJHDLIZGFHHO 7.7 IC50 2
2D structure