Target Details
UniProt ACP12497
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate NY5)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 454
  • Clinical molecules 0
  • Avg pChEMBL 8.33
Top Co-occurrence Targets
Active Molecules (454)
InChIKey pChEMBL Type Targets Clinical
UDNCOTKJZZVWPV 8.5 Ki 2
YXDSUTZGWOOLTI 8.5 Ki 2
JRBCRNGAKHIIBU 8.4 Ki 2
BGTODZAMNVMTGT 8.4 IC50 2
DLCNQKKUXRFUON 8.4 IC50 2
FHAHURNGIVLDQN 8.4 Ki 2
QMJIUGVUFJPDBZ 8.4 Ki 2
WPGHMMPZJWGJEU 8.4 Ki 2
ZNEZCXJJIUHKKH 8.4 Ki 2
FJCFRXMLYMDVAR 8.4 IC50 2
KHHLYBOHRSWBOZ 8.4 Ki 2
LKWOENQGRXKRQP 8.4 Ki 2
DQHWWSRQFWBYKQ 8.4 Ki 2
SRNDLXYVYKGRFI 8.4 Ki 2
SRJPSKNGOVFEQC 8.4 IC50 2
AOYXHSKLMZDHPN 8.3 Ki 2
DWFBAIALVWQHRX 8.3 Ki 2
RNBNABRBLMLESP 8.3 IC50 2
VXOVWUYDWPEXBD 8.3 Ki 2
NDDPZDNJJKSILL 8.3 Ki 2
VIWOOVZGEDFUGH 8.3 Ki 2
LDOHVDYPFKGCAF 8.3 IC50 2
NOYADQYONLFGMN 8.3 Ki 2
CGFVYUGIPISJQG 8.3 Ki 2
PDXABVTZQPAMBI 8.3 Ki 2
ONTDUWVAEQZOGD 8.3 IC50 2
HKLUQPHPQBDWEO 8.3 IC50 2
OCXOYYFOGHBUKE 8.2 Ki 2
PXMJLFGIXDKOBX 8.2 Ki 2
QGJOHLVESASOJB 8.2 Ki 2
IEBXGLCCSIIGCP 8.2 Ki 2
HNOFSZGMHUZHEV 8.2 Ki 2
SSDHDCHQNPWZLQ 8.2 IC50 2
UNWFMMQOIDKTHK 8.2 Ki 2
YFSQZXVVXXIXQG 8.2 IC50 2
RHMWHSCIEZRMHZ 8.2 IC50 2
SCVGALCLJNKWJI 8.2 IC50 2
WINNFDUWGPPOBZ 8.2 Ki 2
FSFMSQDLEGJAJG 8.2 Ki 2
DXPPSGZWDKIKAH 8.2 Ki 2
CDWYOPDREJTKQH 8.2 Ki 2
MOCWEQREIHGFDD 8.2 IC50 2
YNTKPAFJCHPPOK 8.2 IC50 2
YFQXDMQSJQFILP 8.1 IC50 2
ZOQHQYKHUNCUNU 8.1 IC50 2
JPNYRBVKJYFOBV 8.1 Ki 2
LLIXCTOZLODPSK 8.1 Ki 2
MBNPLZRTGOAFGX 8.1 Ki 2
QCZIGGBDUSMTIJ 8.1 Ki 2
JNBVLGDICHLLTN 8.1 IC50 3
2D structure