Target Details
UniProt ACP12497
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate NY5)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 454
  • Clinical molecules 0
  • Avg pChEMBL 8.33
Top Co-occurrence Targets
Active Molecules (454)
InChIKey pChEMBL Type Targets Clinical
FDYJWNQORWMJFP 8.8 IC50 2
WKVUZGXALWGBQC 8.8 Ki 2
CSUKPQVMRKQBSB 8.8 Ki 2
MEMPZWYMKIENFT 8.8 Ki 2
WVPSCZBMYQIZMS 8.8 IC50 2
HQARCNFWJWVJSV 8.8 IC50 2
SPTXJZHACPMACC 8.8 Ki 2
RRHNFHNXWMHGQP 8.8 Ki 2
FIWNNAIJMGZTNA 8.7 IC50 2
FXXCOXGHNXZQPW 8.7 Ki 2
WQFIXFLIBHKDSR 8.7 Ki 2
LLRKKARNQCFJDO 8.7 IC50 3
BYLKXTBRJNXJAX 8.7 Ki 2
KEYGVCKWMFAJLI 8.7 IC50 2
VQMZYQKMPARVIQ 8.7 Ki 2
GURZXAWQZSNWCW 8.7 Ki 2
JCRRNSCPFUQUFN 8.7 Ki 2
KDYPVPWYOGIVQF 8.7 Ki 2
NNOAGIUJEAGRGK 8.7 Ki 2
QIZKEGQOQMEFPD 8.7 Ki 2
VORGFXCNNGFWSP 8.7 Ki 2
LLMTYJLMNZMATO 8.7 Ki 2
UJHPSSIRIQYFHE 8.7 Ki 2
UZZNRAUXEFSJJZ 8.7 Ki 2
DIVWCYHNQIMLLP 8.7 IC50 2
IPFUGNDHFBFCLN 8.7 IC50 2
MMXGPKYYNISCHB 8.7 IC50 2
POTILZIEQCOPAG 8.7 Ki 2
AOZZDVARVHBKHM 8.6 Ki 2
OSVARXBLQYUJJF 8.6 IC50 2
KMUAFILYGKAKHD 8.6 Ki 2
UNUPWGPCVBPXQE 8.6 Ki 2
VGAVLLKXJGUABN 8.6 IC50 2
WIUDTZXSQKGXHD 8.6 IC50 3
ZVSTVGCGZDZJQW 8.6 IC50 2
CUTWMGRMTNRFHO 8.6 Ki 2
FHAJFFRLMGECJB 8.6 Ki 2
DBSUAMMVSYETMT 8.6 IC50 2
FKUHCZHJZWOCRL 8.6 Ki 2
FQWCTMAHSVLUKL 8.6 Ki 2
YQNOXGAZMZYQEE 8.6 Ki 2
COOPLUBZYCIUFU 8.5 IC50 2
PHRPVVBORYLBTD 8.5 IC50 2
RUWNNMYCDLXNBR 8.5 Ki 2
MTBIKTXGJMGCBP 8.5 IC50 2
UPWOUZDRKCEYPI 8.5 IC50 2
NFHZJXYEEPTVBN 8.5 Ki 2
ZOMNPGWFMCUJBM 8.5 IC50 2
BZDQGKJBMUHQGC 8.5 Ki 2
VDAMGRGIJMNRLL 8.5 Ki 3
2D structure