Target Details
UniProt ACP12497
Gene Symbolgag-pol
Protein NameGag-Pol polyprotein
OrganismHuman immunodeficiency virus type 1 group M subtype B (isolate NY5)
Entry Name
Organism Category Pathogen
Pfam Domains PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC)
Summary
  • Multi-target molecules 454
  • Clinical molecules 0
  • Avg pChEMBL 8.33
Top Co-occurrence Targets
Active Molecules (454)
InChIKey pChEMBL Type Targets Clinical
NNOFYWJFSHHUJW 9.4 Ki 3
COYUFXKETXXNHC 9.4 IC50 2
GHXMNIYXDTYJRJ 9.4 Ki 2
KYTSIVAPHUFMRI 9.4 Ki 2
VZNNJZGVQVNHCM 9.4 Ki 2
ZSYJEFDOEYIEPI 9.4 Ki 2
GTKXWDRHECRXIZ 9.4 IC50 2
WRNVKZZCUAPYRR 9.4 IC50 2
IVSJEGKVUYYFNA 9.4 IC50 2
PSHUCZKRZJVSPI 9.4 Ki 2
ZAVBVWUMKMZPAI 9.4 Ki 2
VJEYRJGOROCIKW 9.3 IC50 2
IBGSYHZPJOAHDT 9.3 IC50 2
OBRPRLIEMNDOGJ 9.3 Ki 2
QPDCJMXOIJUAPY 9.3 Ki 2
FVXGZVWGOFVUIM 9.3 Ki 2
MURCDOXDAHPNRQ 9.3 IC50 2
WGUDWHYBVHSPSU 9.3 IC50 2
SWJSIAZKWPALMA 9.3 IC50 2
RITIXPBLKVIIFG 9.3 Ki 2
GJFDHKMKAAWPPS 9.3 IC50 2
RRSJFIZKJZRETD 9.2 Ki 2
UOHMQWQGAJAUGT 9.2 Ki 4
ZOMNPGWFMCUJBM 9.2 IC50 2
YHKWCKXVLPYUKQ 9.2 Ki 2
LJMLRDFXBGZNOB 9.2 IC50 4
FVCKWPQMLLACPQ 9.2 Ki 2
SMDNSMSAGVSMIP 9.2 Ki 2
UZBJXXZZZVEMND 9.2 IC50 2
IRQGWRXNIWWMMU 9.1 Ki 2
SMABGRXWDGFPEH 9.1 Ki 2
OKNWBOKCZOFVKS 9.0 Ki 2
GYFHTEOWKRLODY 9.0 IC50 2
IMXXWUHDQINZEB 9.0 Ki 2
LGQICAULOIAVMN 9.0 Ki 2
QMNHBQAFCJWMJT 9.0 Ki 2
RVRZGUWLTBTUQV 9.0 Ki 2
QZBGFQPYINAGJE 8.9 Ki 2
CPUYSKJCJDRZOR 8.9 Ki 2
OAYKABVVJPVGJQ 8.9 IC50 2
PFYXADIWLAQFKJ 8.9 IC50 2
AJPKIPJBVMYDNN 8.9 Ki 2
YLEGWYXZMZBAFY 8.9 Ki 2
MBCZMDSALKGQPM 8.9 IC50 2
AHSQZQWEKNDRIX 8.8 Ki 2
CSWRAOHDICNMPU 8.8 Ki 2
RKKXLJSFTPRDSM 8.8 Ki 2
TZKGOSNDFIBVER 8.8 IC50 2
WBZOUMUPXZAPEF 8.8 Ki 2
BMLVFCSZGJVQSQ 8.8 Ki 2
2D structure