Target Details
| UniProt AC | P12497 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate NY5) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 454
- Clinical molecules 0
- Avg pChEMBL 8.33
Active Molecules (454)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NUZHSQZGCWZLGP
|
10.1 | IC50 | 2 | — | |
ULZQPXCCYGSIEK
|
10.1 | Ki | 2 | — | |
ACDSTTDXRYHRGH
|
10.0 | IC50 | 2 | — | |
CRGBWRPKHYQBLG
|
10.0 | IC50 | 2 | — | |
FOBRXMROTNVGST
|
10.0 | Ki | 2 | — | |
IHWHGUPQQYJEJX
|
10.0 | IC50 | 2 | — | |
ZJBRKIRKNPBADJ
|
10.0 | IC50 | 2 | — | |
FOVRWBMYYSFRJC
|
10.0 | Ki | 2 | — | |
JZWIKLUJPPKQIL
|
10.0 | Ki | 2 | — | |
PUWGCBYRYTWKFB
|
10.0 | IC50 | 2 | — | |
QHMRYQPPHBYFRG
|
10.0 | IC50 | 2 | — | |
XZKOCRLLAUYWLK
|
10.0 | Ki | 2 | — | |
QPVWMQXBTCSLCB
|
9.9 | Ki | 2 | — | |
MGUCDSPLDUZWFB
|
9.9 | IC50 | 2 | — | |
GBCDOYQRVNSPPY
|
9.9 | IC50 | 2 | — | |
XSAZXCCZKMWBKB
|
9.9 | IC50 | 2 | — | |
BFKBFXHIZWPEIZ
|
9.8 | IC50 | 2 | — | |
KQOVSEYTSQWNCB
|
9.8 | IC50 | 2 | — | |
QWXVAJISGYODFJ
|
9.8 | Ki | 2 | — | |
LGMBHWQZEHFJOS
|
9.8 | IC50 | 2 | — | |
CNNKZGRBCPFNKW
|
9.8 | IC50 | 2 | — | |
KECQKQUDKBXADS
|
9.8 | IC50 | 2 | — | |
QAEDTXWPNADCED
|
9.8 | IC50 | 2 | — | |
CEXRANZMBATAHS
|
9.8 | IC50 | 2 | — | |
JHOFCODADOCEIF
|
9.8 | IC50 | 2 | — | |
LCKITJOWWCXRAD
|
9.8 | IC50 | 2 | — | |
LGYBUYUKEZVHLQ
|
9.8 | IC50 | 2 | — | |
POIJPWBGRRKOEC
|
9.8 | Ki | 2 | — | |
BJSDYSQDZIOQOY
|
9.8 | IC50 | 2 | — | |
CEJZVKZLVAQAHB
|
9.8 | IC50 | 2 | — | |
VGMPZEPIRBEORD
|
9.8 | IC50 | 2 | — | |
DYYJWDSYFDXNOW
|
9.8 | IC50 | 5 | — | |
PGBOPLATAWOMRE
|
9.7 | IC50 | 2 | — | |
INMQYOIMKNCOOR
|
9.7 | IC50 | 2 | — | |
GRZXUXXLRTYPJR
|
9.7 | Ki | 2 | — | |
AXEUVBCBVIQZCZ
|
9.7 | IC50 | 2 | — | |
POTVKRBLAIMCGT
|
9.7 | Ki | 2 | — | |
YQGGCSWNCZJMOG
|
9.7 | IC50 | 2 | — | |
ZGLNLADIKLQLDI
|
9.7 | Ki | 2 | — | |
IBEFZWIXMAEVAT
|
9.6 | Ki | 2 | — | |
NPEMYFWDGCYISM
|
9.6 | IC50 | 2 | — | |
TVPZOFNHBJUMNP
|
9.6 | Ki | 2 | — | |
JRADSVKTKARKBE
|
9.5 | IC50 | 2 | — | |
NMIMFKATLFLNPM
|
9.5 | Ki | 2 | — | |
ZGQZLXSZBYZZLN
|
9.5 | Ki | 2 | — | |
MAMJAUDDHCPYJQ
|
9.5 | IC50 | 3 | — | |
OLRXMFAOSDZYQZ
|
9.5 | Ki | 2 | — | |
UMNROTOYYWSPDV
|
9.5 | IC50 | 3 | — | |
IUVJUTKIAUWSDH
|
9.5 | Ki | 2 | — | |
ZFZABTBOHOLXDC
|
9.4 | IC50 | 2 | — |