Target Details
| UniProt AC | P12497 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate NY5) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 454
- Clinical molecules 0
- Avg pChEMBL 8.33
Active Molecules (454)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JORVRJNILJXMMG
|
13.8 | Ki | 2 | — | |
KTXGTJRUYOGULA
|
11.4 | Ki | 2 | — | |
UFSMRNQSQSGJII
|
11.2 | Ki | 2 | — | |
QPVWMQXBTCSLCB
|
11.0 | Ki | 3 | — | |
QPVWMQXBTCSLCB
|
10.9 | Ki | 3 | — | |
AHWCYDXQIXZVRK
|
10.8 | Ki | 2 | — | |
CWAPFPHVCGEYRK
|
10.7 | IC50 | 3 | — | |
IBJYNRZEQITOHY
|
10.7 | IC50 | 2 | — | |
JBMUJPIOBHXTBM
|
10.7 | IC50 | 2 | — | |
QWXPUMULWMMLKL
|
10.7 | IC50 | 2 | — | |
XZQIZKWFXZKEAV
|
10.7 | IC50 | 2 | — | |
ZGWLZLXBDWVOBP
|
10.6 | Ki | 2 | — | |
HVEBASXMVUNVTR
|
10.5 | IC50 | 2 | — | |
JHXAGQHXTOUOAK
|
10.5 | IC50 | 2 | — | |
KWQSZJFNIYQWFS
|
10.5 | Ki | 2 | — | |
PKJPLBXKJRGYRL
|
10.5 | IC50 | 2 | — | |
PRPIEBUSWYMLSB
|
10.5 | IC50 | 3 | — | |
WSSCUQOFDGTCKU
|
10.5 | IC50 | 2 | — | |
HRYSVKPTFVWINZ
|
10.5 | Ki | 2 | — | |
QCBGCIMPJCAVDQ
|
10.4 | Ki | 2 | — | |
APIPLLBUSGFYKP
|
10.4 | IC50 | 2 | — | |
JHLHCZGWXCUYAR
|
10.4 | IC50 | 2 | — | |
LFTMEZYTSNGORM
|
10.4 | Ki | 2 | — | |
NQBHHXONDCQLRN
|
10.4 | IC50 | 2 | — | |
RLJQWYVDXNSZRV
|
10.4 | Ki | 2 | — | |
RTAOSKPTWQTCBX
|
10.4 | IC50 | 2 | — | |
TWZWSIXDZUIEIJ
|
10.4 | IC50 | 3 | — | |
VFIIEWPPQLSHRX
|
10.4 | Ki | 2 | — | |
DQRSUYGZTXMPLM
|
10.4 | Ki | 2 | — | |
IBYKYUOLRZSYBB
|
10.3 | Ki | 2 | — | |
HSNYTGTZBQKMTG
|
10.3 | Ki | 2 | — | |
GBGNQOSPNHQALW
|
10.3 | IC50 | 3 | — | |
ANNUMOOPAZTSPK
|
10.3 | IC50 | 2 | — | |
DYKNOWOXJACNMI
|
10.3 | IC50 | 2 | — | |
HSRYXNOZZMLYGS
|
10.3 | IC50 | 2 | — | |
JIINVZHJRITJBO
|
10.3 | IC50 | 2 | — | |
MDIRMTMAUIDUHR
|
10.3 | IC50 | 2 | — | |
SWPBTKCAQDJKSO
|
10.3 | IC50 | 3 | — | |
UMKGIYRNMMTPJS
|
10.3 | Ki | 2 | — | |
WUIIVYZPUDLMGE
|
10.3 | IC50 | 3 | — | |
BIHYGUVPMSZAHD
|
10.2 | IC50 | 2 | — | |
BKEXZOJHHKGPBQ
|
10.2 | IC50 | 2 | — | |
ZXMNXYSILSXVSY
|
10.2 | Ki | 2 | — | |
NJBBLOIWMSYVCQ
|
10.2 | Ki | 3 | — | |
VCNRITFCECGWNQ
|
10.2 | IC50 | 3 | — | |
WWYHZIBXQFYYRM
|
10.2 | Ki | 2 | — | |
AROGOLUHMWJZII
|
10.2 | IC50 | 2 | — | |
OEBPYTHAFYTQCV
|
10.2 | IC50 | 2 | — | |
QCDSMEFLKXHFKV
|
10.2 | IC50 | 2 | — | |
MGHDILCKBXOROX
|
10.1 | IC50 | 2 | — |