Target Details
| UniProt AC | P11802 |
|---|---|
| Gene Symbol | CDK4 |
| Protein Name | Cyclin-dependent kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,896
- Clinical molecules 538
- Avg pChEMBL 7.72
KEGG Pathways (28)
- AGE-RAGE signaling pathway in diabetic complications
- Bladder cancer
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Endocrine resistance
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human T-cell leukemia virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- T cell receptor signaling pathway
- Tight junction
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (4)
Active Molecules (2,896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GKTNOVUFHDVNPA
|
8.7 | IC50 | 4 | — | |
GMHSCMWFLYBPIU
|
8.7 | IC50 | 3 | — | |
GPJWAQYXKOYKLZ
|
8.7 | IC50 | 2 | — | |
IIHKFIWSMAISST
|
8.7 | IC50 | 6 | — | |
LTNIHYAIRMIXOL
|
8.7 | IC50 | 3 | — | |
MEERXFXGAAXQOJ
|
8.7 | IC50 | 4 | — | |
NAGFLZVMWVHHLW
|
8.7 | Ki | 2 | — | |
NLHJLMBCNCNHRL
|
8.7 | IC50 | 2 | — | |
NROJANSVZVKJQE
|
8.7 | IC50 | 2 | — | |
OHNWSWSUMDWFSA
|
8.7 | Ki | 6 | — | |
OIQCBGFNCAFMQX
|
8.7 | Ki | 10 | — | |
OIWOJECTXFWECL
|
8.7 | IC50 | 5 | Yes | |
OPJBZLDDGJGVCQ
|
8.7 | IC50 | 5 | — | |
PTUBNTQWBQUBRX
|
8.7 | IC50 | 2 | — | |
QLTMJJAAHXGJMD
|
8.7 | Ki | 10 | — | |
QTTLRBURMUNSGV
|
8.7 | IC50 | 3 | — | |
REZSMOYMCKDNEU
|
8.7 | IC50 | 3 | — | |
SIEQAYSHYKILTK
|
8.7 | IC50 | 3 | — | |
SLHUOQIIOYHUFR
|
8.7 | IC50 | 2 | — | |
UKDNMBIYQCJECP
|
8.7 | IC50 | 2 | — | |
UVEBMCRIHHZDFG
|
8.7 | Ki | 8 | — | |
UZWDCWONPYILKI
|
8.7 | IC50 | 47 | — | |
VASFNXBXECJRSY
|
8.7 | IC50 | 15 | — | |
VSTBDMYJXAWENH
|
8.7 | Ki | 6 | — | |
VWXHIFNNYBTKPP
|
8.7 | IC50 | 3 | — | |
VXBMLLKHEDZLSY
|
8.7 | pIC50 | 4 | Yes | |
YZSCPLGKKMSBMV
|
8.7 | IC50 | 10 | — | |
ZFFPZCADMXKXTH
|
8.7 | IC50 | 3 | — | |
ZRBMKKBZXGSURN
|
8.7 | IC50 | 2 | — | |
ZURIPGCQHWFPSQ
|
8.7 | IC50 | 2 | — | |
AXTGGTFVALFVDO
|
8.7 | IC50 | 6 | — | |
AZENZYQBDCPVQO
|
8.7 | IC50 | 3 | — | |
GIOKUJORFDKSSG
|
8.7 | IC50 | 7 | — | |
OFTAQYQPSSRBOZ
|
8.7 | Ki | 4 | — | |
ZAPGHPQYYDYEQW
|
8.7 | IC50 | 6 | — | |
CVNQRFZZFGTWIK
|
8.7 | IC50 | 3 | — | |
DIJLSYRZXZRGJF
|
8.7 | IC50 | 3 | — | |
DLOAOZHQATYZNK
|
8.7 | IC50 | 2 | — | |
DSMBDRWDECFDNR
|
8.7 | IC50 | 7 | — | |
DZDDEICDXJYDRL
|
8.7 | IC50 | 2 | — | |
FSSQAUUKDWDXEX
|
8.7 | Ki | 4 | — | |
HWUQUQZRNDZMLC
|
8.7 | IC50 | 3 | — | |
IWSXQLKBUPJIBK
|
8.7 | IC50 | 2 | — | |
KIKLVQCDRAYAMG
|
8.7 | IC50 | 2 | — | |
NSWBUBCIZVPAIF
|
8.7 | IC50 | 2 | — | |
OEJRGRXZSULSGO
|
8.7 | IC50 | 2 | — | |
POVBNEVJRAXZQO
|
8.7 | IC50 | 3 | — | |
SAWDJPCFUCEYJD
|
8.7 | Ki | 4 | — | |
VHWYHHQIYHLXIJ
|
8.7 | IC50 | 2 | — | |
XIVVCWMLPOQNDX
|
8.7 | IC50 | 3 | — |