Target Details
| UniProt AC | P11802 |
|---|---|
| Gene Symbol | CDK4 |
| Protein Name | Cyclin-dependent kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,896
- Clinical molecules 538
- Avg pChEMBL 7.72
KEGG Pathways (28)
- AGE-RAGE signaling pathway in diabetic complications
- Bladder cancer
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Endocrine resistance
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human T-cell leukemia virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- T cell receptor signaling pathway
- Tight junction
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (4)
Active Molecules (2,896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SZRLOUJSZUQGCD
|
8.8 | IC50 | 3 | — | |
YWCRCIBLGLRDHR
|
8.8 | IC50 | 2 | — | |
DYNVDYWVVYCHHR
|
8.8 | IC50 | 3 | — | |
GZAGBRPFBCDRDL
|
8.8 | IC50 | 4 | — | |
JDIAYVMOUUKPNK
|
8.8 | IC50 | 5 | — | |
JLIDFAZKTWWWCN
|
8.8 | IC50 | 5 | — | |
PEMNVVTZKGRLSX
|
8.8 | IC50 | 7 | — | |
ZAFJPCZWYDCVJT
|
8.8 | IC50 | 3 | — | |
GNEARXSVRDSWKT
|
8.8 | IC50 | 7 | — | |
BAYGKMGZGJYXFQ
|
8.7 | Ki | 4 | — | |
CGMYFNOVLBOMQH
|
8.7 | Ki | 4 | — | |
CGMYFNOVLBOMQH
|
8.7 | Ki | 4 | — | |
CXOZYBPVDKRPHI
|
8.7 | IC50 | 2 | — | |
JRHOBEGXOYAOBM
|
8.7 | Ki | 4 | — | |
KUXCGTVJRJBHEO
|
8.7 | Ki | 4 | — | |
PAXKGQZKOJPPEG
|
8.7 | pIC50 | 5 | Yes | |
QDVDCIIBNIJIPH
|
8.7 | IC50 | 4 | — | |
RGNVSYDAMGOPSH
|
8.7 | Ki | 4 | — | |
STJKLSZICWMZSS
|
8.7 | IC50 | 3 | — | |
UTDIUAOBXDHROL
|
8.7 | IC50 | 5 | — | |
VQBVWRIVPOILKH
|
8.7 | Ki | 3 | — | |
ZBNQMLROFDKTHM
|
8.7 | IC50 | 2 | — | |
ZDJLCMWGZIMCAQ
|
8.7 | Ki | 4 | — | |
GOWOIXBMOFKIQJ
|
8.7 | IC50 | 4 | Yes | |
ZEWPRVBMQMQROZ
|
8.7 | IC50 | 4 | — | |
ZTXZICVBZWFLGQ
|
8.7 | IC50 | 3 | — | |
AWZRGPIFBNJODY
|
8.7 | IC50 | 3 | — | |
CFZGMAQTSTWGSI
|
8.7 | IC50 | 2 | — | |
FDNONPIMUKKMQB
|
8.7 | IC50 | 2 | — | |
HCAPKVUYVLOOHA
|
8.7 | IC50 | 3 | — | |
KWTCGLLOWQHMIN
|
8.7 | IC50 | 2 | — | |
LMABWMJUORCNEW
|
8.7 | Ki | 4 | — | |
NRMCNHRZOLZAMB
|
8.7 | IC50 | 2 | — | |
RHWIDIZNQRAAIU
|
8.7 | IC50 | 7 | — | |
SUEYATVNHWMTSO
|
8.7 | IC50 | 7 | — | |
UBZYDNRWJFPDPN
|
8.7 | IC50 | 2 | — | |
JRGMQQCQWFMKLA
|
8.7 | IC50 | 6 | — | |
YERVFCNDCWMBBO
|
8.7 | IC50 | 3 | — | |
BPMAUJVZZZYXDV
|
8.7 | IC50 | 3 | — | |
CFZGMAQTSTWGSI
|
8.7 | IC50 | 2 | — | |
CPJXTPZMRAOYPN
|
8.7 | IC50 | 2 | — | |
CWRTWFWDDAJOMG
|
8.7 | pIC50 | 4 | Yes | |
DKTHMZUTCUNQAZ
|
8.7 | IC50 | 5 | — | |
DUROZRXTLVHYHX
|
8.7 | IC50 | 2 | — | |
DYYOXQSHYDLEFT
|
8.7 | IC50 | 2 | — | |
FJPAQWZAYUMSQZ
|
8.7 | Ki | 4 | — | |
FKVVNZDMHAHADF
|
8.7 | Ki | 4 | — | |
FTWLELHFVFNVSG
|
8.7 | IC50 | 3 | — | |
GBNWWXHUOVAUHT
|
8.7 | pIC50 | 4 | Yes | |
GFXPNXYGBQGEGI
|
8.7 | Ki | 4 | — |