Target Details
| UniProt AC | P11802 |
|---|---|
| Gene Symbol | CDK4 |
| Protein Name | Cyclin-dependent kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,896
- Clinical molecules 538
- Avg pChEMBL 7.72
KEGG Pathways (28)
- AGE-RAGE signaling pathway in diabetic complications
- Bladder cancer
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Endocrine resistance
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human T-cell leukemia virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- T cell receptor signaling pathway
- Tight junction
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (4)
Active Molecules (2,896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HCEVZIBGQRWFCG
|
8.8 | IC50 | 9 | — | |
JBYFOPPGLVHSDJ
|
8.8 | IC50 | 3 | — | |
JINXSJRUNKRAKJ
|
8.8 | IC50 | 3 | — | |
KLYIOUNPTCQBFR
|
8.8 | IC50 | 2 | — | |
MHBAURANSRCGRJ
|
8.8 | IC50 | 2 | — | |
NRMCNHRZOLZAMB
|
8.8 | IC50 | 2 | — | |
OLYGYSAFCXIBIB
|
8.8 | IC50 | 3 | — | |
PQWACVUXFPZERA
|
8.8 | IC50 | 5 | — | |
QXBRBWDRQIISAT
|
8.8 | IC50 | 6 | — | |
QYJLBHRAPDJOSO
|
8.8 | Ki | 4 | — | |
RWXWFEVRTCVSJO
|
8.8 | Ki | 4 | — | |
SAKHMWHBWMDUMO
|
8.8 | IC50 | 7 | — | |
YGZQAQIWZFMADC
|
8.8 | IC50 | 12 | — | |
ZKCDHUYJDPLBTG
|
8.8 | Ki | 4 | — | |
ZZJRRZQQOYYZCO
|
8.8 | IC50 | 4 | — | |
ANELMUPUYRZVHZ
|
8.8 | IC50 | 7 | — | |
BENAWDZPBLPFCU
|
8.8 | IC50 | 3 | — | |
DVAPMYJVUZJNDK
|
8.8 | Ki | 8 | — | |
HQNCNCFOTIHEJU
|
8.8 | IC50 | 3 | — | |
MDLZFWHQTJGZMT
|
8.8 | IC50 | 3 | — | |
QCCNJYPQBCTGGP
|
8.8 | IC50 | 3 | — | |
XKPZMRRASYJBKC
|
8.8 | IC50 | 7 | — | |
XXBMNYHUMYIUIC
|
8.8 | IC50 | 3 | — | |
YFRIHUMUDOXHTG
|
8.8 | IC50 | 5 | — | |
BWIZOFRKIJFPNB
|
8.8 | IC50 | 2 | — | |
CGHADMRBCNGDHX
|
8.8 | IC50 | 8 | Yes | |
DSNHCXNKKZEERJ
|
8.8 | IC50 | 2 | — | |
HTNZLGGHWZIRJC
|
8.8 | IC50 | 3 | — | |
IEYXXFUMUXPXFO
|
8.8 | Ki | 4 | — | |
JUQKGEXKBSXXHM
|
8.8 | IC50 | 2 | — | |
LWCQVHGNSZVWQE
|
8.8 | IC50 | 3 | — | |
PWVOSYHMZXNMBQ
|
8.8 | IC50 | 2 | — | |
SLORTXJSOVPUPP
|
8.8 | IC50 | 3 | — | |
TVXXLAJWEQEGRC
|
8.8 | IC50 | 2 | — | |
URASAXYDDZARND
|
8.8 | IC50 | 2 | — | |
VBGIUUAJXDRAPC
|
8.8 | Ki | 4 | — | |
WWTFYOIDRQEIOZ
|
8.8 | IC50 | 3 | — | |
IHSJJFRMGGAMME
|
8.8 | IC50 | 5 | — | |
SSVSKCKWUAPYHI
|
8.8 | IC50 | 8 | — | |
YYJMURXYXPOIDU
|
8.8 | Ki | 7 | — | |
IIHKFIWSMAISST
|
8.8 | IC50 | 3 | — | |
JAZHDXRHOSJZHB
|
8.8 | IC50 | 3 | — | |
DWVMFMWELQFMNJ
|
8.8 | IC50 | 3 | — | |
GKYNYPYSGJOBRE
|
8.8 | IC50 | 2 | — | |
GYDXFTMHNUETBY
|
8.8 | IC50 | 5 | — | |
HWUQUQZRNDZMLC
|
8.8 | IC50 | 3 | — | |
PXVCFDHPZYVHEG
|
8.8 | IC50 | 3 | — | |
QCALUKUBCRTVRC
|
8.8 | Ki | 4 | — | |
SKRUYIPFBIYOHZ
|
8.8 | IC50 | 2 | — | |
SZRKXCASACKTFU
|
8.8 | IC50 | 3 | — |