Target Details
| UniProt AC | P11802 |
|---|---|
| Gene Symbol | CDK4 |
| Protein Name | Cyclin-dependent kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,896
- Clinical molecules 538
- Avg pChEMBL 7.72
KEGG Pathways (28)
- AGE-RAGE signaling pathway in diabetic complications
- Bladder cancer
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Endocrine resistance
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human T-cell leukemia virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- T cell receptor signaling pathway
- Tight junction
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (4)
Active Molecules (2,896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VAPFBPVHSQVGMQ
|
8.9 | Ki | 4 | — | |
VHKPWKUJIHDGJJ
|
8.9 | IC50 | 2 | — | |
AGIIDJZSMZSLJN
|
8.9 | IC50 | 9 | Yes | |
FHUULRWYKIDOHF
|
8.9 | IC50 | 3 | — | |
DHQTVQLYTCGZPM
|
8.9 | IC50 | 2 | — | |
LSXXISAPRYZBDC
|
8.9 | IC50 | 2 | — | |
MLLWORSXSDVTQA
|
8.9 | IC50 | 2 | — | |
ROVFHHODJNANCC
|
8.9 | IC50 | 2 | — | |
VXXZEWXBMJSADU
|
8.9 | IC50 | 3 | — | |
WUNBOTQFUIFMPU
|
8.9 | Ki | 4 | — | |
XPMRMPBWKVMUTB
|
8.9 | Ki | 5 | — | |
JKKUZTDMJDZHEB
|
8.9 | IC50 | 7 | — | |
UEYQVGAFBVFHAU
|
8.9 | pIC50 | 3 | Yes | |
QXBRBWDRQIISAT
|
8.9 | IC50 | 6 | — | |
SXVVQLGGDQUNKQ
|
8.9 | IC50 | 5 | — | |
UGMXVKWXOFIULK
|
8.9 | IC50 | 5 | — | |
QIEKHLDZKRQLLN
|
8.9 | Ki | 9 | — | |
SDAWBLGFXWXOCC
|
8.9 | IC50 | 3 | — | |
VNRANBWAFHAFQG
|
8.9 | IC50 | 2 | — | |
XKPZMRRASYJBKC
|
8.9 | IC50 | 3 | — | |
AUIRGOWAROZXCR
|
8.8 | IC50 | 6 | — | |
CNEMATMUMUNODK
|
8.8 | IC50 | 2 | — | |
DNYGSWNXJXELOX
|
8.8 | Ki | 5 | — | |
FAEZGBZGTZNWMS
|
8.8 | Ki | 4 | — | |
FAEZGBZGTZNWMS
|
8.8 | Ki | 4 | — | |
MFFUZTBYSYJSTO
|
8.8 | IC50 | 3 | — | |
NDQPEKJCVSIVHE
|
8.8 | IC50 | 4 | — | |
QDFRMUUVZQGYCN
|
8.8 | IC50 | 2 | — | |
RLSSWKHNBFFPTF
|
8.8 | IC50 | 3 | — | |
RSJIUPFUDJRJNK
|
8.8 | Ki | 4 | — | |
SIMJTPTVYRLFAT
|
8.8 | IC50 | 3 | — | |
VZRDHFCDSYWOHQ
|
8.8 | Ki | 4 | — | |
WBMDZLSDTLNSBE
|
8.8 | Ki | 4 | — | |
YTNZPCAMOLEZQS
|
8.8 | IC50 | 2 | — | |
DHFGHSZKOLMKGI
|
8.8 | IC50 | 2 | — | |
IRHOQMGOYMQRJB
|
8.8 | IC50 | 3 | — | |
SSIOYGMEKCPFAV
|
8.8 | IC50 | 5 | — | |
SXMLFYVKHGTDIW
|
8.8 | IC50 | 5 | Yes | |
WWPOWSOSERGQKM
|
8.8 | IC50 | 3 | — | |
FEBXDTFBHZJUJT
|
8.8 | IC50 | 5 | — | |
NCAQSQYHTSCOCV
|
8.8 | IC50 | 7 | — | |
OPZCPKBSWZFNRM
|
8.8 | IC50 | 3 | — | |
XHCXEGJOAXJLFH
|
8.8 | IC50 | 3 | — | |
BAUPLMMFMLNKKB
|
8.8 | IC50 | 3 | — | |
BRBJCJHJBAMBPR
|
8.8 | IC50 | 12 | — | |
COALBSOMQOGPKG
|
8.8 | IC50 | 3 | — | |
DTBQJHPUJVUHNS
|
8.8 | Ki | 7 | — | |
FBUYSZWFYRBPBV
|
8.8 | IC50 | 4 | — | |
FHEQFUUMLHFZOS
|
8.8 | IC50 | 3 | — | |
GCELNWHYDYQJHB
|
8.8 | IC50 | 3 | — |