Target Details
| UniProt AC | P11802 |
|---|---|
| Gene Symbol | CDK4 |
| Protein Name | Cyclin-dependent kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,896
- Clinical molecules 538
- Avg pChEMBL 7.72
KEGG Pathways (28)
- AGE-RAGE signaling pathway in diabetic complications
- Bladder cancer
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Endocrine resistance
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human T-cell leukemia virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- T cell receptor signaling pathway
- Tight junction
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (4)
Active Molecules (2,896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VRIWWBXFSKWVDK
|
9.0 | IC50 | 3 | — | |
VWQIQPRBMMSYCE
|
9.0 | IC50 | 6 | — | |
VYYVSGBSHKYYPS
|
9.0 | IC50 | 2 | — | |
XANUTEQSZWRXHI
|
9.0 | IC50 | 3 | — | |
XCJRUIHXLFTUNW
|
9.0 | IC50 | 3 | — | |
XNFJUHZLDMOZHP
|
9.0 | IC50 | 2 | — | |
XVRFIUSGDOJQMI
|
9.0 | IC50 | 3 | — | |
YCOFHJMLYTXYAJ
|
9.0 | IC50 | 3 | — | |
YPJRHEKCFKOVRT
|
9.0 | IC50 | 12 | — | |
YRSCDRTXWYUNBB
|
9.0 | pIC50 | 4 | Yes | |
YUBKIQYQCNIXLH
|
9.0 | IC50 | 2 | — | |
YWCKVLPHEKWBJP
|
9.0 | IC50 | 3 | — | |
ZFNZZKVYLDBWRD
|
9.0 | Ki | 8 | — | |
ZQHZICOJSNIGEO
|
9.0 | IC50 | 2 | — | |
BAPMZESGRJMZNL
|
9.0 | IC50 | 5 | — | |
FTFHCSWIOVPGGS
|
9.0 | IC50 | 6 | — | |
LCDCVRYMEWMBEV
|
9.0 | IC50 | 5 | — | |
LQHMJVOJVOLFTJ
|
9.0 | IC50 | 7 | — | |
PUXKEKPYASIYGT
|
9.0 | IC50 | 7 | — | |
CZQMPFCNIINMMC
|
9.0 | IC50 | 8 | — | |
APLCQEOLIQVWQN
|
9.0 | Ki | 7 | — | |
PMCGYDRAUVMLBE
|
9.0 | IC50 | 3 | — | |
POTKDJWRAMHALZ
|
9.0 | IC50 | 9 | — | |
CGMYNNHQYROWEE
|
9.0 | IC50 | 2 | — | |
GZVZVBKIIIOOOF
|
9.0 | Ki | 4 | — | |
GZVZVBKIIIOOOF
|
9.0 | Ki | 4 | — | |
KEYGZUKDLFNALV
|
9.0 | Ki | 4 | — | |
LIJUCWLALFXGCL
|
9.0 | IC50 | 7 | — | |
RKILQDBEPHSTGP
|
9.0 | IC50 | 4 | — | |
SMJIOBIBQNQQMH
|
9.0 | Ki | 4 | — | |
XSAQISWEGTUJBT
|
9.0 | IC50 | 7 | — | |
AKGTYSYXMRZPBV
|
8.9 | IC50 | 9 | — | |
IVKYJVDFJKEXIH
|
8.9 | IC50 | 6 | — | |
KGMVZSJAPXYTKH
|
8.9 | IC50 | 23 | — | |
PFGMZHAOYLGYMA
|
8.9 | Ki | 8 | — | |
TWNUIDQVTSUXKY
|
8.9 | IC50 | 3 | — | |
ZJXAYHKSLDKUOY
|
8.9 | IC50 | 3 | — | |
AAVOJGZMGDAVNM
|
8.9 | IC50 | 6 | — | |
IWSDTEGBQVXXON
|
8.9 | IC50 | 7 | — | |
PBDNNWWYSHCMCH
|
8.9 | IC50 | 7 | — | |
QPSCTAMMABVQIH
|
8.9 | IC50 | 3 | — | |
UVMVCEDKKHGTIW
|
8.9 | IC50 | 7 | — | |
XHCXEGJOAXJLFH
|
8.9 | IC50 | 3 | — | |
DHDRSDPRAQJACL
|
8.9 | IC50 | 4 | — | |
KABOFUDSOMJKKL
|
8.9 | Ki | 4 | — | |
LFWRZTGKNXDMJU
|
8.9 | IC50 | 5 | — | |
MNPXDFVGSLMIRV
|
8.9 | IC50 | 2 | — | |
NWMOJGWJNSLCBU
|
8.9 | IC50 | 3 | — | |
RHMZROQDZHOQQS
|
8.9 | IC50 | 2 | — | |
RLTCKGIEOKUCSQ
|
8.9 | IC50 | 3 | — |