Target Details
| UniProt AC | P11802 |
|---|---|
| Gene Symbol | CDK4 |
| Protein Name | Cyclin-dependent kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,896
- Clinical molecules 538
- Avg pChEMBL 7.72
KEGG Pathways (28)
- AGE-RAGE signaling pathway in diabetic complications
- Bladder cancer
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Endocrine resistance
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human T-cell leukemia virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- T cell receptor signaling pathway
- Tight junction
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (4)
Active Molecules (2,896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IKMLTMFWMJPBIL
|
9.1 | IC50 | 2 | — | |
PDGKHKMBHVFCMG
|
9.1 | IC50 | 5 | — | |
RLRQXKXWZNPYRB
|
9.1 | IC50 | 3 | — | |
VXLAKHWYGRKCGI
|
9.1 | IC50 | 9 | — | |
YPMOBRWHNOTUIL
|
9.1 | IC50 | 7 | — | |
FJVCRQHDTUXVMH
|
9.1 | Ki | 4 | — | |
JFBGPNNZAPXVQS
|
9.1 | Ki | 4 | — | |
JKTDPJGOPWGJLD
|
9.1 | IC50 | 2 | — | |
KBPQIDCZZMLFSH
|
9.1 | Ki | 4 | — | |
LASUSMNDZBNUAS
|
9.1 | Ki | 4 | — | |
LDJNLOZYHRVQME
|
9.1 | IC50 | 2 | — | |
SFINPTBPZGSJQZ
|
9.1 | Ki | 4 | — | |
BONJLZFNDLMWRE
|
9.0 | IC50 | 3 | — | |
DSMBDRWDECFDNR
|
9.0 | IC50 | 6 | — | |
GUYDOLZTUBMZKV
|
9.0 | Ki | 6 | — | |
MSKGFMBSNBBHMB
|
9.0 | IC50 | 2 | — | |
SPKWRLBKVPRPMT
|
9.0 | IC50 | 9 | — | |
BURBSRHEPGFKHA
|
9.0 | IC50 | 2 | — | |
WIAMCDYCLOMHKF
|
9.0 | IC50 | 3 | — | |
PBDNNWWYSHCMCH
|
9.0 | IC50 | 7 | — | |
VUKGJVXJRDQYFA
|
9.0 | IC50 | 9 | — | |
AAOLDQJTTACKSD
|
9.0 | Ki | 4 | Yes | |
AGNLNZIKBGWSFX
|
9.0 | IC50 | 4 | — | |
AJFKYSBQAUFOAW
|
9.0 | IC50 | 3 | — | |
AKDZNPFQMDRCMU
|
9.0 | IC50 | 7 | — | |
AVZIKDOLKKDYPG
|
9.0 | Ki | 4 | — | |
BOQORPXVPMXARS
|
9.0 | pIC50 | 3 | Yes | |
CEIAWFVLEUQXHI
|
9.0 | IC50 | 5 | — | |
FZHZYQRQDGJIBK
|
9.0 | pIC50 | 3 | Yes | |
IYLQAMPBXDBIFL
|
9.0 | IC50 | 2 | — | |
JIYCAEUCAZHFNL
|
9.0 | IC50 | 3 | — | |
JRNJNYBQQYBCLE
|
9.0 | Kd | 40 | Yes | |
JTZWTKLEXMYEMU
|
9.0 | Ki | 6 | — | |
LDHMPOHMNQEDFG
|
9.0 | Ki | 4 | — | |
LDXLQEXLXZCYSR
|
9.0 | pIC50 | 2 | Yes | |
LFGOPXAPKINMIT
|
9.0 | Ki | 4 | — | |
LICJOAWXMPKZSX
|
9.0 | Ki | 10 | — | |
LQLWCEYRAKKEIP
|
9.0 | IC50 | 2 | — | |
LUHGNQLUGTWNCL
|
9.0 | Ki | 12 | — | |
MIZFTGLHDNPPOW
|
9.0 | IC50 | 3 | — | |
NOUVQMCOTSOPTN
|
9.0 | IC50 | 2 | — | |
OCUYCOQPRGFQEV
|
9.0 | pIC50 | 3 | Yes | |
OYBGABJZRRNVII
|
9.0 | Ki | 4 | — | |
PSILLYORWULWQE
|
9.0 | Ki | 4 | — | |
PSWOMNFIVDHMDM
|
9.0 | IC50 | 6 | — | |
UFUZVHSCAUVFOR
|
9.0 | IC50 | 5 | — | |
UHCMUGYUWQCODZ
|
9.0 | Ki | 5 | — | |
UHRJHVJHZMDUJK
|
9.0 | Ki | 5 | — | |
VADHWSWHRRXKCV
|
9.0 | IC50 | 2 | — | |
VGQBMNJRVGPBKT
|
9.0 | IC50 | 3 | — |