Target Details
| UniProt AC | P11802 |
|---|---|
| Gene Symbol | CDK4 |
| Protein Name | Cyclin-dependent kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,896
- Clinical molecules 538
- Avg pChEMBL 7.72
KEGG Pathways (28)
- AGE-RAGE signaling pathway in diabetic complications
- Bladder cancer
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Endocrine resistance
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human T-cell leukemia virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- T cell receptor signaling pathway
- Tight junction
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (4)
Active Molecules (2,896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GFUYDGPHKDLMHQ
|
8.5 | IC50 | 2 | — | |
UZGLLJQDQDOFFE
|
8.5 | IC50 | 2 | — | |
VCEVKRSWGMXHPO
|
8.5 | IC50 | 2 | — | |
WJENEGQQOQWXTQ
|
8.5 | IC50 | 3 | — | |
YUTSNVSLGLNUDW
|
8.5 | IC50 | 3 | — | |
HLOKDQHOCMHLLI
|
8.5 | IC50 | 7 | — | |
ISWNVTVWJJQFQV
|
8.5 | IC50 | 3 | — | |
AKEMXASAMBDUOC
|
8.5 | pIC50 | 3 | Yes | |
AMPDZRFNHCTPTF
|
8.5 | Ki | 10 | — | |
AZXYPCBAGCXZPP
|
8.5 | IC50 | 4 | — | |
BBUVDDPUURMFOX
|
8.5 | IC50 | 4 | — | |
BBUVDDPUURMFOX
|
8.5 | IC50 | 3 | — | |
BHQZGGSZRHDQFZ
|
8.5 | pIC50 | 13 | Yes | |
CQMZJAORBQTGTR
|
8.5 | IC50 | 4 | — | |
CZPQAZKLLINYQE
|
8.5 | IC50 | 2 | — | |
DLYVGVOGPLQZFG
|
8.5 | pIC50 | 2 | Yes | |
DSYAGVYPTCYGKP
|
8.5 | IC50 | 5 | — | |
DUHXDQPGUINDGD
|
8.5 | IC50 | 3 | — | |
GBVXPZRKGCHAIL
|
8.5 | IC50 | 6 | — | |
GTQSNWXKTIFPBY
|
8.5 | IC50 | 5 | — | |
HFMQOFFEBHLBLK
|
8.5 | IC50 | 3 | — | |
HOKDQPMWTBQYHL
|
8.5 | IC50 | 8 | — | |
HOWIXJOUKWURJN
|
8.5 | IC50 | 2 | — | |
HZORGXNHDYOIAL
|
8.5 | IC50 | 3 | — | |
ICVHMFOFVOYFPB
|
8.5 | IC50 | 3 | — | |
IEPWMLWPYJPPOJ
|
8.5 | IC50 | 3 | — | |
IHNQNVXNYQNXFW
|
8.5 | IC50 | 3 | — | |
KLULGLOBJXRRAM
|
8.5 | IC50 | 4 | — | |
MGLCYKLRRMBDTH
|
8.5 | IC50 | 3 | — | |
MRPVMOCAEFVNTQ
|
8.5 | IC50 | 3 | — | |
NWIPTENCWQPQTO
|
8.5 | Ki | 4 | Yes | |
ONYDIUVHLRZYJB
|
8.5 | IC50 | 3 | — | |
PJAZUKUXPBWWHG
|
8.5 | IC50 | 2 | — | |
PLZQIHPAODEDGT
|
8.5 | IC50 | 3 | — | |
POFVJRKJJBFPII
|
8.5 | Ki | 8 | — | |
QTNFANVRKMXUKB
|
8.5 | IC50 | 3 | — | |
RATTVJZQLHAPSM
|
8.5 | IC50 | 3 | — | |
RBMBLJOYIGVBNO
|
8.5 | IC50 | 6 | — | |
RFAFNLAEMWZQJI
|
8.5 | IC50 | 3 | — | |
RKGAIIIRLQHASS
|
8.5 | IC50 | 3 | — | |
RLWUWLYKPWQOFL
|
8.5 | IC50 | 3 | — | |
RNHRCKQJHFBOKM
|
8.5 | IC50 | 2 | — | |
RVBOIHXTZQGXRV
|
8.5 | pIC50 | 3 | Yes | |
SHEPFXMPLORKLW
|
8.5 | Ki | 8 | — | |
TUVPQAXSMZXTMF
|
8.5 | IC50 | 2 | — | |
TWBKRUBZYHTJIT
|
8.5 | IC50 | 3 | — | |
USXJKWQIDCWKGZ
|
8.5 | Ki | 10 | — | |
VCQXPLQAUTUUTC
|
8.5 | IC50 | 3 | — | |
VFNJLPYDAYDGKC
|
8.5 | IC50 | 5 | — | |
VISMKLIGDLCELE
|
8.5 | IC50 | 3 | — |