Target Details
| UniProt AC | P11802 |
|---|---|
| Gene Symbol | CDK4 |
| Protein Name | Cyclin-dependent kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,896
- Clinical molecules 538
- Avg pChEMBL 7.72
KEGG Pathways (28)
- AGE-RAGE signaling pathway in diabetic complications
- Bladder cancer
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Endocrine resistance
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human T-cell leukemia virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- T cell receptor signaling pathway
- Tight junction
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (4)
Active Molecules (2,896)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YJGGMTJSWVEDCJ
|
8.7 | IC50 | 4 | — | |
KZZDDXBCJROTIP
|
8.7 | IC50 | 8 | — | |
UEGPMXKTKCKXOK
|
8.7 | IC50 | 3 | — | |
VTLCELVAADXYMP
|
8.7 | IC50 | 2 | — | |
AXTXGXVLRKZCFY
|
8.7 | Ki | 4 | — | |
DSUXSBZUWGKTQG
|
8.7 | IC50 | 2 | — | |
DZWLTXLJZHDQOP
|
8.7 | IC50 | 2 | — | |
HGFLDVQTDYSNRS
|
8.7 | IC50 | 4 | Yes | |
HVTYFANOGPVRAE
|
8.7 | IC50 | 3 | — | |
IUYLNMPIDQAYSG
|
8.7 | IC50 | 7 | — | |
KNRZSSHNVWPHLG
|
8.7 | IC50 | 2 | — | |
LMIPCDJYZXYYLQ
|
8.7 | IC50 | 5 | — | |
LNUMMPBBRBTMNM
|
8.7 | IC50 | 3 | — | |
NBSJZWFDNFWQDN
|
8.7 | IC50 | 29 | — | |
OAWKAAOUONBYOS
|
8.7 | IC50 | 2 | — | |
SFFBXSHJSYMDGI
|
8.7 | Ki | 4 | — | |
SVXDTIUTCGVODS
|
8.7 | IC50 | 3 | — | |
BRROKWAZCDMWEU
|
8.7 | IC50 | 3 | — | |
DHMHGKLKKIGMHX
|
8.7 | IC50 | 3 | — | |
QHCHMOFMVBOPSK
|
8.7 | IC50 | 3 | — | |
VCPXSBULBDYRLT
|
8.7 | pIC50 | 4 | Yes | |
WIAMCDYCLOMHKF
|
8.7 | IC50 | 6 | — | |
ZUOVZWHQGAJGQA
|
8.7 | IC50 | 3 | — | |
CGHADMRBCNGDHX
|
8.6 | IC50 | 4 | — | |
CGHADMRBCNGDHX
|
8.6 | IC50 | 5 | Yes | |
COALBSOMQOGPKG
|
8.6 | IC50 | 2 | — | |
CPTPRZGRXQWAQQ
|
8.6 | Ki | 4 | — | |
RECJWFRRTNLZDX
|
8.6 | Ki | 4 | — | |
UZGLLJQDQDOFFE
|
8.6 | IC50 | 3 | — | |
VEBBZRVCYCERII
|
8.6 | IC50 | 2 | — | |
ZSNPHFWSNIDXSN
|
8.6 | IC50 | 3 | — | |
AVKHUGZDSUKIKQ
|
8.6 | IC50 | 3 | — | |
JNZTWAOEOYBNNP
|
8.6 | IC50 | 5 | — | |
KSHZWPCJWQWIST
|
8.6 | IC50 | 2 | — | |
SOHOEERULHWXJB
|
8.6 | IC50 | 5 | — | |
SQAZXWOTKSSCBZ
|
8.6 | IC50 | 3 | — | |
WEIJWGUXTMLFKT
|
8.6 | IC50 | 3 | — | |
YYWWXDBYEUYMKM
|
8.6 | IC50 | 3 | — | |
ICCWQZQHILTVNE
|
8.6 | Ki | 4 | — | |
KYEMOBSMSCIMFC
|
8.6 | IC50 | 2 | — | |
LLFOBMRPWNABCB
|
8.6 | IC50 | 11 | — | |
LLMVPGIWVUJSPH
|
8.6 | IC50 | 2 | — | |
LTJSYFAVWOFESN
|
8.6 | Ki | 4 | — | |
OIQZLVBXHSEFQP
|
8.6 | IC50 | 6 | — | |
PPCNFXQXVGAXIF
|
8.6 | IC50 | 2 | — | |
QELIOBZBBHRBAA
|
8.6 | Ki | 4 | — | |
ROMAHJZEHBXJSU
|
8.6 | IC50 | 7 | — | |
TWBXLKWAYLBJOV
|
8.6 | IC50 | 3 | — | |
UQNXGQYESHUBBX
|
8.6 | IC50 | 3 | — | |
WTKYHVUVQSLNBW
|
8.6 | IC50 | 6 | — |