Target Details
| UniProt AC | P11586 |
|---|---|
| Gene Symbol | MTHFD1 |
| Protein Name | C-1-tetrahydrofolate synthase, cytoplasmic |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01268 (FTHFS) PF00763 (THF_DHG_CYH) PF02882 (THF_DHG_CYH_C) |
Summary
- Multi-target molecules 3
- Clinical molecules 0
- Avg pChEMBL 6.77
KEGG Pathways (4)
Associated Diseases (2)
Active Molecules (3)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MWKSRKSEWLRPBL
|
7.1 | Kd | 1075 | — | |
JSNFRYBHBVDHSG
|
7.0 | IC50 | 2 | — | |
OQKAKSSZSQPTDZ
|
6.2 | IC50 | 2 | — |