Target Details
| UniProt AC | P11474 |
|---|---|
| Gene Symbol | ESRRA |
| Protein Name | Steroid hormone receptor ERR1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 40
- Clinical molecules 10
- Avg pChEMBL 7.34
Active Molecules (40)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VWUXBMIQPBEWFH
|
8.7 | IC50 | 8 | Yes | |
RYBHKLZSHRZGQK
|
8.5 | IC50 | 2 | — | |
UHDQHUPIXKORDL
|
8.4 | IC50 | 2 | — | |
XRUZUCBHVAMRMC
|
8.4 | IC50 | 6 | Yes | |
MJJDANHWHHWHME
|
8.3 | IC50 | 6 | Yes | |
VOXZDWNPVJITMN
|
8.3 | IC50 | 8 | — | |
BEPBQWCCVBVLGI
|
8.2 | IC50 | 2 | — | |
IIJORMBEWMYDEN
|
8.1 | IC50 | 2 | — | |
TZBJGXHYKVUXJN
|
8.0 | IC50 | 12 | Yes | |
SDQIIVSWOGDEKO
|
7.7 | IC50 | 2 | — | |
LGNJPIOPTLOFKV
|
7.5 | IC50 | 6 | Yes | |
XCPJWYKWACPRGL
|
7.5 | IC50 | 2 | — | |
GLVQMSCCFOGRRG
|
7.5 | Ki | 4 | — | |
LHEAAXNLFNVCGK
|
7.5 | IC50 | 2 | — | |
AWCSWPAAFIXQFA
|
7.5 | IC50 | 2 | — | |
TYWJUKOBNZCZNP
|
7.4 | Ki | 2 | — | |
OGDCTCUVBBYZTK
|
7.3 | IC50 | 2 | — | |
JHGHNHLKUJDBRE
|
7.3 | IC50 | 6 | Yes | |
NFDYBNVVFHAKIV
|
7.3 | IC50 | 2 | — | |
MPGOJACGGLDRIE
|
7.2 | IC50 | 6 | Yes | |
KGZZMTWCVOBJOB
|
7.2 | Ki | 4 | — | |
FSCSPCCXODGFCH
|
7.1 | Ki | 3 | — | |
LZRCWCHYOCKNED
|
7.1 | IC50 | 4 | Yes | |
SAQPECWWGZJCNM
|
7.1 | IC50 | 2 | — | |
GKRORYXGWZWHID
|
7.0 | IC50 | 2 | — | |
VZSCCCSZIQBCNZ
|
7.0 | Ki | 2 | — | |
DWTNKXOQSZYRNO
|
7.0 | IC50 | 2 | — | |
QAGWYKCFYYZWRQ
|
7.0 | Ki | 4 | — | |
YPLWXUBAJNIFDO
|
7.0 | IC50 | 2 | — | |
UQJVSWJIGSWDBK
|
6.9 | Ki | 4 | — | |
BMIUOILMANDNSR
|
6.9 | IC50 | 2 | — | |
LIAQMIXVDMWARY
|
6.8 | IC50 | 2 | — | |
BTKBDYIATAATDW
|
6.8 | IC50 | 2 | — | |
OBBIOCQFTMNSJI
|
6.8 | IC50 | 4 | Yes | |
ASVAJAKZUJMJRU
|
6.8 | IC50 | 2 | — | |
OWWNFHKDBPGHSM
|
6.8 | IC50 | 2 | — | |
NKANXQFJJICGDU
|
6.7 | IC50 | 35 | Yes | |
UZCGSEMPWJYIKG
|
6.7 | Ki | 4 | — | |
DVBSYBFWHRYTSH
|
6.2 | IC50 | 2 | — | |
BIUDJVBDYHJCCR
|
6.0 | Ki | 4 | — |