Target Details
UniProt ACP11473
Gene SymbolVDR
Protein NameVitamin D3 receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00104 (Hormone_recep) PF00105 (zf-C4)
Summary
  • Multi-target molecules 87
  • Clinical molecules 1
  • Avg pChEMBL 8.88
Associated Diseases (2)
Top Co-occurrence Targets
Active Molecules (87)
InChIKey pChEMBL Type Targets Clinical
KVQQVUQXVQANFT 8.7 Ki 4
OJONWBFOVMXDLK 8.7 Ki 4
LBCLWNAKMLUAKD 8.7 Ki 4
HYUZMDKRIBTARX 8.7 Ki 4
APCSKDZXHMFZBO 8.6 Ki 4
YRESHCJSCNXCIP 8.6 Ki 4
QXEYNUWHIAFPHP 8.6 Ki 4
WVNDCOIKWKQPDK 8.6 Ki 4
WNBAUVLDXSOKMM 8.5 Ki 4
KBFMOHUYUYNYGP 8.5 Ki 4
AXFCFTMMGTUXSG 8.4 Ki 4
PDADFIJOFSWDJB 8.4 Ki 4
QPVGNXJYLPJOIQ 8.4 Ki 4
GLRWZEISUAIVMI 8.4 Ki 4
ULGYNCVBFLQVPX 8.4 Ki 4
VZHORDSFYCKLRO 8.4 Ki 4
YOQMDXGCJSLBBS 8.3 Ki 4
PPOMMOPYGUOVFS 8.3 Ki 4
XMADFSDPKTZGLY 8.2 Ki 4
SWZJPLIVZNKLDQ 8.2 Ki 4
VQHDFSMAHHFXEB 8.2 Ki 4
GUBYHCIYOBESBX 8.2 Ki 4
NQIFYNGRQPWASE 8.2 Ki 4
FJGIJPVLRUOQFB 8.1 Ki 4
MYMAOKWDKYVIOY 8.1 Ki 4
GKXKKYAXVMCURJ 8.1 Ki 4
SPBIQVBLOPVLFL 8.0 Ki 4
QVVUXZWJNUQUIQ 8.0 Ki 4
ZHVCTZIFHMKHHU 7.9 Ki 4
AIKLCYAFOOBGEV 7.9 Ki 2
QOEMKJVIXGOYHR 7.1 IC50 2
RTKIYFITIVXBLE 7.1 IC50 17 Yes
UBDHJEXXHMTARH 6.8 Kd 4
XCVIXZRNZRDCKE 6.7 Kd 4
AIKLCYAFOOBGEV 6.5 Ki 2
SMEROWZSTRWXGI 6.5 Kd 2
GFUKCIXVOZBJQK 6.2 IC50 2
2D structure