Target Details
| UniProt AC | P11387 |
|---|---|
| Gene Symbol | TOP1 |
| Protein Name | DNA topoisomerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14370 (Topo_C_assoc) PF01028 (Topoisom_I) PF02919 (Topoisom_I_N) |
Summary
- Multi-target molecules 6
- Clinical molecules 0
- Avg pChEMBL 7.11
Active Molecules (6)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MWKSRKSEWLRPBL
|
8.2 | Kd | 1075 | — | |
RPFYDENHBPRCTN
|
7.5 | IC50 | 2 | — | |
AJTBUWMKUOLMNM
|
7.4 | IC50 | 5 | — | |
ZCCPLJOKGAACRT
|
7.4 | Kd | 599 | — | |
VSJKWCGYPAHWDS
|
6.2 | IC50 | 19 | — | |
FJHBVJOVLFPMQE
|
6.0 | IC50 | 2 | — |