Target Details
| UniProt AC | P11362 |
|---|---|
| Gene Symbol | FGFR1 |
| Protein Name | Fibroblast growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 3,320
- Clinical molecules 348
- Avg pChEMBL 7.53
KEGG Pathways (18)
- Adherens junction
- Breast cancer
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- IgSF CAM signaling
- MAPK signaling pathway
- Melanoma
- PI3K-Akt signaling pathway
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
- Thermogenesis
Associated Diseases (8)
Active Molecules (3,320)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YTDWYXQAKOWNAV
|
8.5 | IC50 | 3 | — | |
YTDWYXQAKOWNAV
|
8.5 | IC50 | 4 | — | |
HAMQGTWNMUEACH
|
8.5 | IC50 | 5 | — | |
SISPBNWXCLKBKE
|
8.5 | IC50 | 5 | — | |
ULHGAQSVFPOUDY
|
8.5 | Ki | 43 | — | |
GYXODBZTJVUDOH
|
8.5 | IC50 | 4 | — | |
JFRMAVZKDFQNCB
|
8.5 | IC50 | 2 | — | |
LLBFRCVAASUZPB
|
8.5 | IC50 | 2 | — | |
PCUPJGFLZXOSJC
|
8.5 | IC50 | 2 | — | |
QIXCNXNXARCJIU
|
8.5 | IC50 | 3 | — | |
XZWWCRJOEPEAFT
|
8.5 | IC50 | 3 | — | |
FVUYKZNGSHSNBI
|
8.5 | IC50 | 5 | — | |
IZIDHKRDFQGCMR
|
8.5 | IC50 | 2 | — | |
JKEDZMIFSJMZHH
|
8.5 | IC50 | 2 | — | |
JMGHVRJQMLUCCL
|
8.5 | IC50 | 3 | — | |
JVHRYVZNKJPNLU
|
8.5 | IC50 | 5 | — | |
NVVLHTUQGYXRPA
|
8.5 | IC50 | 2 | — | |
YYBZWPUIOONRPU
|
8.5 | IC50 | 2 | — | |
AZOXWOCICFEBCQ
|
8.5 | IC50 | 11 | — | |
UAHJXPBYRPDINJ
|
8.5 | IC50 | 2 | — | |
UHSDGQHRNMRTLI
|
8.5 | IC50 | 5 | — | |
UZZUQDLJRHRISA
|
8.5 | Kd | 3 | — | |
WHBOZVVJRXLYLP
|
8.5 | IC50 | 2 | — | |
KONCHEYJKNSRJF
|
8.5 | IC50 | 5 | — | |
NXQWBKIKMLKVOS
|
8.5 | IC50 | 5 | — | |
OYJDTEBZSGLLNC
|
8.5 | IC50 | 2 | — | |
XNRZJGZKJIEPIW
|
8.5 | IC50 | 3 | — | |
BYJMQCNNDWXBRA
|
8.4 | IC50 | 5 | — | |
CCWQRQKDZAKBBS
|
8.4 | IC50 | 6 | — | |
FBJRJSLJQISKRR
|
8.4 | IC50 | 5 | — | |
PDCHXVOBVIQUEZ
|
8.4 | IC50 | 5 | — | |
POMPWDXYMSRSAW
|
8.4 | IC50 | 4 | — | |
AMXKOAUPVJWSGA
|
8.4 | IC50 | 3 | — | |
CEYCXVCSPGUEPS
|
8.4 | IC50 | 2 | — | |
FLXIGSCPROLWAB
|
8.4 | IC50 | 2 | — | |
HQKHKYBURJLEMV
|
8.4 | IC50 | 5 | — | |
KEIPNCCJPRMIAX
|
8.4 | IC50 | 5 | — | |
KNPLSRBVKFTLQU
|
8.4 | IC50 | 3 | — | |
MYFRXSIWRAGTKV
|
8.4 | IC50 | 5 | — | |
QAGLJDWYCCJEHH
|
8.4 | pIC50 | 7 | Yes | |
SRAFQIWHQBJFJJ
|
8.4 | IC50 | 2 | — | |
AYMIOSAGFUFSMC
|
8.4 | IC50 | 4 | — | |
DNVFTXQYIYFQBW
|
8.4 | IC50 | 4 | — | |
DXIOQMYZLOTSFT
|
8.4 | IC50 | 2 | — | |
GLYUIGNYFSCICA
|
8.4 | IC50 | 2 | — | |
LQLFCORECOTJTQ
|
8.4 | IC50 | 2 | — | |
MXMLJQCILGAGCP
|
8.4 | IC50 | 5 | — | |
QIEVSBKOXPAREF
|
8.4 | IC50 | 5 | — | |
HLRISBLSHWIQBN
|
8.4 | IC50 | 2 | — | |
HNXJXOXKHKFGNB
|
8.4 | IC50 | 2 | — |