Target Details
| UniProt AC | P11362 |
|---|---|
| Gene Symbol | FGFR1 |
| Protein Name | Fibroblast growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 3,320
- Clinical molecules 348
- Avg pChEMBL 7.53
KEGG Pathways (18)
- Adherens junction
- Breast cancer
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- IgSF CAM signaling
- MAPK signaling pathway
- Melanoma
- PI3K-Akt signaling pathway
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
- Thermogenesis
Associated Diseases (8)
Active Molecules (3,320)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PZUMGJXNMDBEIT
|
8.6 | IC50 | 2 | — | |
SEHOCSFHPAZLLH
|
8.6 | IC50 | 2 | — | |
SOSSKSLYRZFQAX
|
8.6 | IC50 | 2 | — | |
WGEUPMAJTYQVEP
|
8.6 | IC50 | 3 | — | |
ZKKMRDODNGIIGF
|
8.6 | IC50 | 2 | — | |
BQCQOBOXMZWHQL
|
8.6 | IC50 | 5 | — | |
KTQNUSVVKAQAIV
|
8.6 | IC50 | 5 | — | |
MSSUJWPHHVXXFT
|
8.6 | IC50 | 5 | — | |
JEYPNCLDZGLRAU
|
8.6 | IC50 | 2 | — | |
JTFVQKRKLOURMQ
|
8.6 | IC50 | 2 | — | |
MQABPWIBJWWDIM
|
8.6 | IC50 | 2 | — | |
MWTKOJWSURZTTH
|
8.6 | IC50 | 2 | — | |
NFYDPTASEPAEMT
|
8.6 | IC50 | 4 | — | |
OWLHHVGNWXMBFF
|
8.6 | IC50 | 2 | — | |
RNLCEYKRDCFQPX
|
8.6 | IC50 | 2 | — | |
ANMVTYAYYHHSTF
|
8.5 | IC50 | 2 | — | |
AVHLETMOCLYGNK
|
8.5 | IC50 | 5 | — | |
FNTYYRMQLQQXEI
|
8.5 | IC50 | 4 | — | |
LJQGHKNSFBSZFJ
|
8.5 | IC50 | 2 | — | |
OTZMRUFJZIGILY
|
8.5 | IC50 | 6 | — | |
SXXLGVGHYVRIAF
|
8.5 | IC50 | 2 | — | |
UXBXBZKCNJEIRO
|
8.5 | IC50 | 2 | — | |
WAKJUGXHBUNUIT
|
8.5 | IC50 | 5 | — | |
WRABCNDMFRHWIR
|
8.5 | IC50 | 6 | — | |
CUMCBEDCPQGOTJ
|
8.5 | IC50 | 5 | — | |
LNZDHCYDEDDMTH
|
8.5 | IC50 | 5 | — | |
ZDPMRTCLIVGQSN
|
8.5 | IC50 | 5 | — | |
BNRXMSGHPVYSDK
|
8.5 | IC50 | 24 | — | |
CSGDFNSJHVTVHD
|
8.5 | pIC50 | 2 | Yes | |
DFYOEDRVJUNFKB
|
8.5 | IC50 | 2 | — | |
FBKIPMHVNJQANW
|
8.5 | IC50 | 3 | — | |
GEKQPARVOXSQNS
|
8.5 | IC50 | 2 | — | |
HCAUEIOBSYOQPN
|
8.5 | pIC50 | 5 | Yes | |
JEQXEBGQZXOOGK
|
8.5 | IC50 | 2 | — | |
JJNUVTXMRDPOPO
|
8.5 | IC50 | 3 | — | |
KTZAHPAGCSCZTG
|
8.5 | IC50 | 3 | — | |
MAXGMZGUSCSCRT
|
8.5 | IC50 | 2 | — | |
MQFRLYRFRPJFEY
|
8.5 | IC50 | 3 | — | |
RQIXEOXMOHDTLC
|
8.5 | IC50 | 2 | — | |
SAHTUCUOJHIHGN
|
8.5 | IC50 | 5 | — | |
VRWGJEGSNQCDOR
|
8.5 | IC50 | 3 | — | |
WNVADWMUVOLRPY
|
8.5 | IC50 | 3 | — | |
WUTMSLAMPQIEAG
|
8.5 | IC50 | 2 | — | |
YXTHFMOUCQZVJH
|
8.5 | IC50 | 3 | — | |
YZRSMWKLOJZVAD
|
8.5 | IC50 | 4 | — | |
AQHXGQTWGFVXTB
|
8.5 | IC50 | 2 | — | |
CYHGHBQCTXVJCN
|
8.5 | IC50 | 3 | — | |
DUZJRGKUZTUIRX
|
8.5 | IC50 | 2 | — | |
HEIWGGHLGABSLB
|
8.5 | Kd | 10 | — | |
QUVMICMHDQTVPB
|
8.5 | IC50 | 5 | — |