Target Details
| UniProt AC | P11362 |
|---|---|
| Gene Symbol | FGFR1 |
| Protein Name | Fibroblast growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 3,320
- Clinical molecules 348
- Avg pChEMBL 7.53
KEGG Pathways (18)
- Adherens junction
- Breast cancer
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- IgSF CAM signaling
- MAPK signaling pathway
- Melanoma
- PI3K-Akt signaling pathway
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
- Thermogenesis
Associated Diseases (8)
Active Molecules (3,320)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JCQODDIJVHORMY
|
8.8 | IC50 | 5 | — | |
PVEPJQQWAOPNNQ
|
8.8 | IC50 | 2 | — | |
UOWDVWIHJKFQPY
|
8.8 | IC50 | 5 | — | |
BYVRSERQASVMIN
|
8.7 | IC50 | 3 | — | |
DSFNDCSGZPQFHC
|
8.7 | IC50 | 2 | — | |
DXQAUQWASZIRTJ
|
8.7 | IC50 | 2 | — | |
GWOHWBYOVFLZGM
|
8.7 | IC50 | 2 | — | |
GZRXWBJYUJUZNW
|
8.7 | IC50 | 3 | — | |
HGUFBZQRVSFTRA
|
8.7 | IC50 | 2 | — | |
HXKRTTRYDVNOTH
|
8.7 | IC50 | 2 | — | |
LTKSJPZMTYBCRM
|
8.7 | IC50 | 2 | — | |
LYDRTKDNCXYTQA
|
8.7 | IC50 | 5 | — | |
SUXYGJZMCWKJJI
|
8.7 | IC50 | 26 | Yes | |
WJZSUSVUKVZGLF
|
8.7 | pIC50 | 7 | Yes | |
ZZDKMIARNROCNG
|
8.7 | IC50 | 2 | — | |
UHPWIGXTFQRPCG
|
8.7 | IC50 | 5 | — | |
WITKAEIQNFPTFS
|
8.7 | IC50 | 5 | — | |
ZXKALWYYLPSYSO
|
8.7 | IC50 | 2 | — | |
AISWQGLURAAAKE
|
8.7 | IC50 | 7 | — | |
CMMUVKONDKDCCZ
|
8.7 | IC50 | 5 | — | |
FONDQLCAYMUQPO
|
8.7 | IC50 | 2 | — | |
HKMTYQNMRIBAHX
|
8.7 | IC50 | 4 | — | |
YLUAUDRMSFJFJJ
|
8.7 | IC50 | 4 | — | |
SYQCXJZLWMRWKD
|
8.7 | IC50 | 5 | — | |
CQDRTFWUDOIACC
|
8.7 | IC50 | 5 | — | |
DCWCFKXCIYCNTA
|
8.7 | IC50 | 3 | — | |
FHDKNSAADPLWFU
|
8.7 | IC50 | 2 | — | |
FZFKBDZAXOFANZ
|
8.7 | IC50 | 2 | — | |
HWEVEQFMAGTKGM
|
8.7 | IC50 | 3 | — | |
HZIAJKJBTRYTIC
|
8.7 | IC50 | 2 | — | |
HZPFRBXNIBOLLW
|
8.7 | IC50 | 2 | — | |
JQYPWJCACYTKIC
|
8.7 | IC50 | 5 | — | |
MCJDCDKCTQBUDW
|
8.7 | IC50 | 2 | — | |
MUWNBQMOGBRDAG
|
8.7 | IC50 | 2 | — | |
MZEOWSVWCPCLAR
|
8.7 | pIC50 | 2 | Yes | |
NYEZHXSUIICMSA
|
8.7 | IC50 | 5 | — | |
ONAZMIGCNRUYHT
|
8.7 | IC50 | 5 | — | |
PHXJVRSECIGDHY
|
8.7 | IC50 | 59 | — | |
UCSSQROSBFPVKH
|
8.7 | pIC50 | 7 | Yes | |
VRQMAABPASPXMW
|
8.7 | Kd | 10 | — | |
WIAGFLYJODEJMC
|
8.7 | IC50 | 2 | — | |
XXRQVZDYLNBSMD
|
8.7 | IC50 | 2 | — | |
UEOZGCZDSDHALE
|
8.7 | IC50 | 5 | — | |
CHZKEAYTNKCUEF
|
8.7 | IC50 | 2 | — | |
GHEIOFQIMGYHML
|
8.7 | IC50 | 5 | — | |
HZZGQUIDAUEOSV
|
8.7 | IC50 | 2 | — | |
IVQXFJNVCKJIHX
|
8.7 | IC50 | 5 | — | |
OACFIPDTGXZIQH
|
8.7 | IC50 | 2 | — | |
OSPKANQURMXUIE
|
8.7 | pIC50 | 7 | Yes | |
PBYKDTVBNNMWRF
|
8.7 | IC50 | 2 | — |