Target Details
| UniProt AC | P11362 |
|---|---|
| Gene Symbol | FGFR1 |
| Protein Name | Fibroblast growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 3,320
- Clinical molecules 348
- Avg pChEMBL 7.53
KEGG Pathways (18)
- Adherens junction
- Breast cancer
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- IgSF CAM signaling
- MAPK signaling pathway
- Melanoma
- PI3K-Akt signaling pathway
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
- Thermogenesis
Associated Diseases (8)
Active Molecules (3,320)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FVBNNGBLKUMCEF
|
8.8 | IC50 | 3 | — | |
HWWONGHTSRGZJQ
|
8.8 | IC50 | 2 | — | |
JZMMRIIMJLFYOI
|
8.8 | IC50 | 2 | — | |
KCIGGSIEQASIPY
|
8.8 | IC50 | 2 | — | |
LNCJTAGAWGYDHX
|
8.8 | IC50 | 2 | — | |
MQNZARJVRSNEJL
|
8.8 | IC50 | 2 | — | |
NDXXZPUMKRBNQB
|
8.8 | IC50 | 3 | — | |
NRTLSZJUKLLLCA
|
8.8 | IC50 | 2 | — | |
OWLHHVGNWXMBFF
|
8.8 | IC50 | 2 | — | |
SENVOZNIDWYYED
|
8.8 | IC50 | 4 | — | |
TVWOUPGUUIDZET
|
8.8 | IC50 | 6 | — | |
WNUXYTTWUXBQMA
|
8.8 | IC50 | 2 | — | |
AHAHQLJJHZPGFT
|
8.8 | IC50 | 5 | — | |
FWUSQYKXFMDVPH
|
8.8 | IC50 | 5 | — | |
DDHPDOGCZLIDPA
|
8.8 | IC50 | 4 | — | |
DXVWDCOHXAEMCI
|
8.8 | IC50 | 3 | — | |
KJAJDINGBBZCDE
|
8.8 | IC50 | 2 | — | |
MBFNJGNWXZAXKI
|
8.8 | IC50 | 2 | — | |
OOIYXPLQGGEDGS
|
8.8 | IC50 | 2 | — | |
QQOOENCAPIWETQ
|
8.8 | IC50 | 2 | — | |
SQUVKQUNFNCXMK
|
8.8 | IC50 | 3 | — | |
ZVFYULVCRUAESA
|
8.8 | IC50 | 2 | — | |
JPJVHSSGRZKSDJ
|
8.8 | IC50 | 5 | — | |
QQMCUGWXDVCQJJ
|
8.8 | IC50 | 2 | — | |
RVBIBDGDUFYRME
|
8.8 | IC50 | 2 | — | |
CVQIAUMEBBKXIR
|
8.8 | IC50 | 2 | — | |
DSBGPNZCYAOULK
|
8.8 | IC50 | 2 | — | |
IGHUBVIQSUHAEU
|
8.8 | IC50 | 2 | — | |
KNACLJBHKVSTDL
|
8.8 | Ki | 40 | — | |
OWRCHUPGWMCPME
|
8.8 | IC50 | 2 | — | |
PSRCAUFYXJRQBZ
|
8.8 | IC50 | 2 | — | |
QAXDRNRWTCRTHG
|
8.8 | IC50 | 2 | — | |
QEOFKIKDUSYLPY
|
8.8 | IC50 | 2 | — | |
SLEJFRIKJJZQKL
|
8.8 | IC50 | 5 | — | |
STSJLCHGAYUSER
|
8.8 | IC50 | 2 | — | |
VEFIZLZPHCCAQO
|
8.8 | IC50 | 3 | — | |
XFGMNTTVFYLJIS
|
8.8 | IC50 | 2 | — | |
XWQJWMKIXLWIOD
|
8.8 | IC50 | 2 | — | |
LNSNRKRKVKSAOL
|
8.8 | IC50 | 2 | — | |
LLLHXFXUIWPWMH
|
8.8 | IC50 | 5 | — | |
GVEQLTBABUNRMS
|
8.8 | IC50 | 2 | — | |
KEJHKWDFKQXLMG
|
8.8 | IC50 | 2 | — | |
RGUQNSKUQAYWDB
|
8.8 | IC50 | 2 | — | |
URIOWDLDOGYPLK
|
8.8 | IC50 | 2 | — | |
UWGPKLQEDALKIM
|
8.8 | IC50 | 2 | — | |
YICOQNPWMAVVBP
|
8.8 | IC50 | 2 | — | |
YOMVQFWXFWVVPY
|
8.8 | IC50 | 2 | — | |
ZKKBDZUWZDKUIQ
|
8.8 | IC50 | 2 | — | |
ZQTRKQPFZQBOMV
|
8.8 | IC50 | 2 | — | |
YIKYPGSFLXUTQT
|
8.8 | IC50 | 5 | — |