Target Details
| UniProt AC | P11362 |
|---|---|
| Gene Symbol | FGFR1 |
| Protein Name | Fibroblast growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 3,320
- Clinical molecules 348
- Avg pChEMBL 7.53
KEGG Pathways (18)
- Adherens junction
- Breast cancer
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- IgSF CAM signaling
- MAPK signaling pathway
- Melanoma
- PI3K-Akt signaling pathway
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
- Thermogenesis
Associated Diseases (8)
Active Molecules (3,320)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SJEVLHTYUBABDJ
|
9.0 | IC50 | 4 | — | |
STINDBVFOPRZHE
|
9.0 | pIC50 | 8 | Yes | |
UQZPQFKVJWOQTM
|
9.0 | IC50 | 4 | — | |
VYULPLQTNFKWPI
|
9.0 | IC50 | 2 | — | |
YHIGPAIFBVOPKV
|
9.0 | IC50 | 4 | — | |
YLMMYYCOZCUKKA
|
8.9 | IC50 | 5 | — | |
FCCSDYKLOXTQPP
|
8.9 | IC50 | 4 | — | |
MKEGPZIMUWZUKO
|
8.9 | IC50 | 4 | — | |
BYCZXBZXUBUKGX
|
8.9 | IC50 | 2 | — | |
CXJITJGGCTWHEG
|
8.9 | IC50 | 3 | — | |
DIDLAUMNKKUFSF
|
8.9 | IC50 | 5 | — | |
IWBVZILESKBVJL
|
8.9 | IC50 | 6 | — | |
MJHFGTHWKHPARC
|
8.9 | IC50 | 5 | — | |
NMODJHIAZMCFBV
|
8.9 | IC50 | 3 | — | |
OLAHOMJCDNXHFI
|
8.9 | IC50 | 6 | — | |
OOJCSNDQUFLDIN
|
8.9 | IC50 | 2 | — | |
VLOPFGZLJSYVCD
|
8.9 | IC50 | 4 | — | |
YWKSYTCBEVSAAX
|
8.9 | IC50 | 3 | — | |
ZELUDNIRCNOVHB
|
8.9 | IC50 | 2 | — | |
ZWDPQCVFSJWCFD
|
8.9 | IC50 | 2 | — | |
QTZWCECBLKRZBR
|
8.9 | IC50 | 4 | — | |
RIDLANJMTSBUSD
|
8.9 | IC50 | 5 | — | |
JTIMRSSBBONYGV
|
8.9 | IC50 | 5 | — | |
OYHDEFFNZNIKPS
|
8.9 | IC50 | 5 | — | |
XWRLHVWTHQFHSY
|
8.9 | IC50 | 5 | — | |
AABHAFTYFDHGCT
|
8.9 | IC50 | 2 | — | |
BQBUDKYPYIHTHV
|
8.9 | IC50 | 2 | — | |
BXJXGGAHIUAWTR
|
8.9 | IC50 | 3 | — | |
GKJCVYLDJWTWQU
|
8.9 | IC50 | 6 | — | |
HOKFABUDYHGQKX
|
8.9 | IC50 | 2 | — | |
IGLSLLWKILRJQQ
|
8.9 | IC50 | 2 | — | |
IWAIRGHIYWNQTE
|
8.9 | IC50 | 2 | — | |
KXKRDLMFFZNYPD
|
8.9 | IC50 | 2 | — | |
MHHLXYGRKUMXPW
|
8.9 | IC50 | 2 | — | |
OCKLCHHQTFDHGO
|
8.9 | IC50 | 2 | — | |
OIAKQMVWXQYUFN
|
8.9 | IC50 | 2 | — | |
OVZKBAUSZIANJA
|
8.9 | IC50 | 5 | — | |
QTGVMULYBGRVHT
|
8.9 | IC50 | 5 | — | |
SRLZJSAQKFBYKX
|
8.9 | IC50 | 2 | — | |
VEGCSHHXEINKOV
|
8.9 | IC50 | 4 | — | |
YRBAKPVAQIOONM
|
8.9 | IC50 | 2 | — | |
KEIPNCCJPRMIAX
|
8.9 | IC50 | 3 | — | |
MNUGHQYUMFMXIC
|
8.9 | IC50 | 5 | — | |
QZUYKKDZNXWNPD
|
8.9 | IC50 | 5 | — | |
ZGLWZSSPPSSMRB
|
8.9 | IC50 | 5 | — | |
GLLVJFAKHOOPKT
|
8.9 | IC50 | 5 | — | |
USCLDZNWLVHDPF
|
8.9 | IC50 | 5 | — | |
VCNJSFBAEBDCKK
|
8.9 | IC50 | 5 | — | |
XUDRPPZFODNIIN
|
8.9 | IC50 | 5 | — | |
DZSUJUOJJJCWGG
|
8.8 | pIC50 | 55 | Yes |