Target Details
| UniProt AC | P11362 |
|---|---|
| Gene Symbol | FGFR1 |
| Protein Name | Fibroblast growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 3,320
- Clinical molecules 348
- Avg pChEMBL 7.53
KEGG Pathways (18)
- Adherens junction
- Breast cancer
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- IgSF CAM signaling
- MAPK signaling pathway
- Melanoma
- PI3K-Akt signaling pathway
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
- Thermogenesis
Associated Diseases (8)
Active Molecules (3,320)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OARJPSVHVHBFTL
|
9.1 | IC50 | 2 | — | |
QMXGFRWKHLJTJA
|
9.1 | IC50 | 2 | — | |
QRSKATROTXSCAH
|
9.1 | IC50 | 2 | — | |
UGADWCXPZTYDIJ
|
9.1 | IC50 | 2 | — | |
ZJRVNNZFLXDMBL
|
9.1 | IC50 | 2 | — | |
FXIBXFGZSDZFSP
|
9.0 | IC50 | 5 | — | |
UCWGZZUXJLIYIK
|
9.0 | IC50 | 4 | — | |
YJAREBGBTVFDIK
|
9.0 | IC50 | 5 | — | |
MDPWQSCOLLDWIY
|
9.0 | IC50 | 5 | — | |
VRQMAABPASPXMW
|
9.0 | IC50 | 8 | — | |
XAGAJLBPFOEQPM
|
9.0 | IC50 | 2 | — | |
AKINNIMWOKBQKR
|
9.0 | IC50 | 2 | — | |
AKNCKKKGJAAVEH
|
9.0 | IC50 | 2 | — | |
ARYDDRNBUXLRQZ
|
9.0 | IC50 | 3 | — | |
BAWZESLJEVSFRN
|
9.0 | IC50 | 2 | — | |
BBEVMAFPVMSMEU
|
9.0 | IC50 | 3 | — | |
BCOJIDFRCFXQSL
|
9.0 | IC50 | 3 | — | |
CTUHJNJXPMROFF
|
9.0 | IC50 | 3 | — | |
FJKSLOFTCKXLSC
|
9.0 | IC50 | 2 | — | |
HYTKNUZBKDBMMN
|
9.0 | IC50 | 5 | — | |
JPESTLPEBJPKGA
|
9.0 | IC50 | 2 | — | |
JXMYXVQTSAHUJU
|
9.0 | IC50 | 2 | — | |
LVPNWYGBLSBXLS
|
9.0 | IC50 | 3 | — | |
NAWYNVJDAIYLPP
|
9.0 | IC50 | 2 | — | |
NUMZOUWDKZZHAY
|
9.0 | IC50 | 2 | — | |
OCMFTUJIRAAZFF
|
9.0 | IC50 | 5 | — | |
PHTNPGCZALDYLD
|
9.0 | IC50 | 4 | — | |
PQULTGFDTTYMKA
|
9.0 | IC50 | 2 | — | |
RHIYIXKVGFLFDX
|
9.0 | IC50 | 2 | — | |
SMWFHLHWOOWYAP
|
9.0 | IC50 | 4 | Yes | |
WFLAIALBWODQSL
|
9.0 | IC50 | 2 | — | |
WXRBLSQWDTUDCY
|
9.0 | IC50 | 2 | — | |
XIQQPHOWVZOQQP
|
9.0 | IC50 | 4 | — | |
GUHZQOUGERIFMY
|
9.0 | IC50 | 5 | — | |
OEIJEWDFQMITII
|
9.0 | IC50 | 5 | — | |
HWKKKYKEHLRWPW
|
9.0 | IC50 | 2 | — | |
AOYJOQPVLIISJS
|
9.0 | IC50 | 4 | — | |
BIZAIIWAPNOYPN
|
9.0 | IC50 | 5 | — | |
BYEGVFRRTLAAQA
|
9.0 | IC50 | 2 | — | |
JYQPFNMDHXKRKL
|
9.0 | IC50 | 5 | — | |
KRHJVQBHCYJAPS
|
9.0 | IC50 | 2 | — | |
LTWBXHYYWOPFGA
|
9.0 | IC50 | 2 | — | |
OACFIPDTGXZIQH
|
9.0 | IC50 | 2 | — | |
OCIIUHMXXRNNNL
|
9.0 | IC50 | 2 | — | |
PFTPAJNMFJOUIG
|
9.0 | IC50 | 5 | — | |
PSWCYOAFOKRCAC
|
9.0 | IC50 | 2 | — | |
QBOPLHQHJDUIPC
|
9.0 | IC50 | 4 | — | |
QKLROYVFWRSBCK
|
9.0 | IC50 | 2 | — | |
SDFCBOWBJRMBSN
|
9.0 | IC50 | 2 | — | |
SDGGLMMHOSCYCM
|
9.0 | IC50 | 2 | — |